UY30856A1 - NEW DERIVATIVES OF 2,4 DIANILINOPIRIMIDINAS, ITS PREPARATION, AS MEDICINES, PHARMACEUTICAL COMPOSITIONS AND MAINLY AS IKK INHIBITORS - Google Patents
NEW DERIVATIVES OF 2,4 DIANILINOPIRIMIDINAS, ITS PREPARATION, AS MEDICINES, PHARMACEUTICAL COMPOSITIONS AND MAINLY AS IKK INHIBITORSInfo
- Publication number
- UY30856A1 UY30856A1 UY30856A UY30856A UY30856A1 UY 30856 A1 UY30856 A1 UY 30856A1 UY 30856 A UY30856 A UY 30856A UY 30856 A UY30856 A UY 30856A UY 30856 A1 UY30856 A1 UY 30856A1
- Authority
- UY
- Uruguay
- Prior art keywords
- mainly
- dianilinopirimidinas
- medicines
- preparation
- pharmaceutical compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Diabetes (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La invencion se refiere a nuevos derivados de 2,4-dianilinopirimidinas, de formula (I), en todas sus formas isomericas y a sus sales, como medicamento principalmente como inhibidores de IKK, donde los sustituyentes son tales como se especifican en la memoria descriptiva y en las reivindicaciones.The invention relates to new derivatives of 2,4-dianylinopyrimidines, of formula (I), in all its isomeric forms and to its salts, as a medicament mainly as IKK inhibitors, where the substituents are as specified in the specification and in the claims.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0700063A FR2911137B1 (en) | 2007-01-05 | 2007-01-05 | NOVEL 2,4-DIANILINOPYRIMIDE DERIVATIVES, THEIR PREPARATION AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND IN PARTICULAR AS INHIBITORS OF IKK |
Publications (1)
Publication Number | Publication Date |
---|---|
UY30856A1 true UY30856A1 (en) | 2008-09-02 |
Family
ID=38353639
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY30856A UY30856A1 (en) | 2007-01-05 | 2008-01-04 | NEW DERIVATIVES OF 2,4 DIANILINOPIRIMIDINAS, ITS PREPARATION, AS MEDICINES, PHARMACEUTICAL COMPOSITIONS AND MAINLY AS IKK INHIBITORS |
Country Status (11)
Country | Link |
---|---|
US (1) | US20100035907A1 (en) |
EP (1) | EP2104673A2 (en) |
JP (1) | JP2010514820A (en) |
CN (1) | CN101605780A (en) |
AR (1) | AR064729A1 (en) |
CA (1) | CA2672955A1 (en) |
CL (1) | CL2008000021A1 (en) |
FR (1) | FR2911137B1 (en) |
TW (1) | TW200836740A (en) |
UY (1) | UY30856A1 (en) |
WO (1) | WO2008099072A2 (en) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2911138B1 (en) * | 2007-01-05 | 2009-02-20 | Sanofi Aventis Sa | NOVEL N, N'-2,4-DIANILINOPYRIMIDINE DERIVATIVES, THEIR PREPARATION AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND IN PARTICULAR AS INHIBITORS OF IKK |
FR2911140B1 (en) * | 2007-01-05 | 2009-02-20 | Sanofi Aventis Sa | NOVEL 2-ANILINO 4-HETEROARYL PYRIMIDES DERIVATIVES, THEIR PREPARATION AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS, AND IN PARTICULAR AS INHIBITORS OF IKK |
FR2911139A1 (en) * | 2007-01-05 | 2008-07-11 | Sanofi Aventis Sa | New 2,4-diaminopyrimidine derivatives useful for treating inflammatory diseases, diabetes or cancer |
WO2011107494A1 (en) | 2010-03-03 | 2011-09-09 | Sanofi | Novel aromatic glycoside derivatives, medicaments containing said compounds, and the use thereof |
EP2582709B1 (en) | 2010-06-18 | 2018-01-24 | Sanofi | Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
EP2760862B1 (en) | 2011-09-27 | 2015-10-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
EP3152557A4 (en) | 2014-06-09 | 2017-12-13 | Biometry Inc. | Low cost test strip and method to measure analyte |
US11175268B2 (en) | 2014-06-09 | 2021-11-16 | Biometry Inc. | Mini point of care gas chromatographic test strip and method to measure analytes |
WO2017009751A1 (en) | 2015-07-15 | 2017-01-19 | Pfizer Inc. | Pyrimidine derivatives |
CN109715067B (en) | 2016-07-19 | 2022-05-17 | 生物统计股份有限公司 | Method and system for measuring analytes using batch calibratable test strips |
CN113061117B (en) * | 2021-03-30 | 2023-02-10 | 长治学院 | 2- ((5-chloro-2- (4-morpholine methylanilino) pyrimidine-4-yl) amino) benzamide derivative |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2003231231A1 (en) * | 2002-05-06 | 2003-11-11 | Bayer Pharmaceuticals Corporation | Pyridinyl amino pyrimidine derivatives useful for treating hyper-proliferative disorders |
EP1598343A1 (en) * | 2004-05-19 | 2005-11-23 | Boehringer Ingelheim International GmbH | 2-Arylaminopyrimidine derivatives as PLK inhibitors |
EP1904479A2 (en) * | 2005-07-11 | 2008-04-02 | Sanofi-Aventis | Novel 2,4-dianilinopyrimidine derivatives, the preparation thereof, their use as medicaments, pharmaceutical compositions and, in particular, as ikk inhibitors |
-
2007
- 2007-01-05 FR FR0700063A patent/FR2911137B1/en not_active Expired - Fee Related
-
2008
- 2008-01-02 WO PCT/FR2008/000001 patent/WO2008099072A2/en active Application Filing
- 2008-01-02 CA CA002672955A patent/CA2672955A1/en not_active Abandoned
- 2008-01-02 CN CNA2008800040919A patent/CN101605780A/en active Pending
- 2008-01-02 EP EP08750460A patent/EP2104673A2/en not_active Withdrawn
- 2008-01-02 JP JP2009544425A patent/JP2010514820A/en not_active Withdrawn
- 2008-01-03 CL CL2008000021A patent/CL2008000021A1/en unknown
- 2008-01-03 AR ARP080100011A patent/AR064729A1/en unknown
- 2008-01-04 UY UY30856A patent/UY30856A1/en not_active Application Discontinuation
- 2008-01-04 TW TW097100457A patent/TW200836740A/en unknown
-
2009
- 2009-07-01 US US12/495,992 patent/US20100035907A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CL2008000021A1 (en) | 2009-03-27 |
JP2010514820A (en) | 2010-05-06 |
TW200836740A (en) | 2008-09-16 |
FR2911137A1 (en) | 2008-07-11 |
WO2008099072A2 (en) | 2008-08-21 |
CN101605780A (en) | 2009-12-16 |
CA2672955A1 (en) | 2008-08-21 |
AR064729A1 (en) | 2009-04-22 |
US20100035907A1 (en) | 2010-02-11 |
EP2104673A2 (en) | 2009-09-30 |
WO2008099072A3 (en) | 2008-11-13 |
FR2911137B1 (en) | 2009-02-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20130205 |