UY30386A1 - AMIDA COMPOUNDS OF ACID 3-AMINO-TIENO (2,3B (BETA) PIRIDINA-2- REPLACED CARBOXYLIC, PROCESSES FOR THEIR PREPARATION AND USES OF THE SAME - Google Patents

AMIDA COMPOUNDS OF ACID 3-AMINO-TIENO (2,3B (BETA) PIRIDINA-2- REPLACED CARBOXYLIC, PROCESSES FOR THEIR PREPARATION AND USES OF THE SAME

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Publication number
UY30386A1
UY30386A1 UY30386A UY30386A UY30386A1 UY 30386 A1 UY30386 A1 UY 30386A1 UY 30386 A UY30386 A UY 30386A UY 30386 A UY30386 A UY 30386A UY 30386 A1 UY30386 A1 UY 30386A1
Authority
UY
Uruguay
Prior art keywords
compounds
processes
piridina
tieno
beta
Prior art date
Application number
UY30386A
Other languages
Spanish (es)
Inventor
Erick Richard Roush Young
Michael Robert Turner
Ronald J Sorcek
John David Ginn
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Priority to UY30386A priority Critical patent/UY30386A1/en
Publication of UY30386A1 publication Critical patent/UY30386A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Se describen compuestos de formula (I): en la que R1 y R4 se definen en este documento, que son utiles como inhibidores de la actividad de quisana del complejo de quisana Ikb (IKK). Por lo tanto, los compuestos son utiles en el tratamiento de enfermedades mediadas por IKK incluyendo enfermedades autoinmunes, enfermedades inflamatorias, enfermedades cardiovasculares y cáncer. También se describen composiciones farmacéuticas que comprenden estos compuestos y procesos para preparar estos compuestosCompounds of formula (I) are described: in which R1 and R4 are defined herein, which are useful as inhibitors of the kenyan activity of the Ikb (IKK) kiwana complex. Therefore, the compounds are useful in the treatment of IKK-mediated diseases including autoimmune diseases, inflammatory diseases, cardiovascular diseases and cancer. Pharmaceutical compositions comprising these compounds and processes for preparing these compounds are also described.

UY30386A 2007-06-04 2007-06-04 AMIDA COMPOUNDS OF ACID 3-AMINO-TIENO (2,3B (BETA) PIRIDINA-2- REPLACED CARBOXYLIC, PROCESSES FOR THEIR PREPARATION AND USES OF THE SAME UY30386A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
UY30386A UY30386A1 (en) 2007-06-04 2007-06-04 AMIDA COMPOUNDS OF ACID 3-AMINO-TIENO (2,3B (BETA) PIRIDINA-2- REPLACED CARBOXYLIC, PROCESSES FOR THEIR PREPARATION AND USES OF THE SAME

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
UY30386A UY30386A1 (en) 2007-06-04 2007-06-04 AMIDA COMPOUNDS OF ACID 3-AMINO-TIENO (2,3B (BETA) PIRIDINA-2- REPLACED CARBOXYLIC, PROCESSES FOR THEIR PREPARATION AND USES OF THE SAME

Publications (1)

Publication Number Publication Date
UY30386A1 true UY30386A1 (en) 2008-01-31

Family

ID=39015803

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30386A UY30386A1 (en) 2007-06-04 2007-06-04 AMIDA COMPOUNDS OF ACID 3-AMINO-TIENO (2,3B (BETA) PIRIDINA-2- REPLACED CARBOXYLIC, PROCESSES FOR THEIR PREPARATION AND USES OF THE SAME

Country Status (1)

Country Link
UY (1) UY30386A1 (en)

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20170627