UY29629A1 - OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAME - Google Patents
OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAMEInfo
- Publication number
- UY29629A1 UY29629A1 UY29629A UY29629A UY29629A1 UY 29629 A1 UY29629 A1 UY 29629A1 UY 29629 A UY29629 A UY 29629A UY 29629 A UY29629 A UY 29629A UY 29629 A1 UY29629 A1 UY 29629A1
- Authority
- UY
- Uruguay
- Prior art keywords
- oxazolidinone compounds
- compounds
- compositions
- same
- formula
- Prior art date
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La invención proporciona nuevos compuestos de oxazolidinona de fórmula (I), en la que A representa determinados heterociclos opcionalmente sustiutido; R1, R2, R3 y R4 se seleccionan independientemente de -H y halógeno; X se selecciona entre O,S, NR9 y CR9R10; teniendo R9 y R10 diferentes significados; Y se selecciona entre O, S, SO, SO2, NO, NR12 y CR12R13, teniendo R12 y R13 diferentes significados.También se proporcionan diferentes procedimientos para la preparación de dichos compuestos. Los compuestos de oxazolidinona de fórmula (I) son activos contra patógenos humanos y veterinarios Gram-positivos y algunos Gram-negativos con una débil actividad inhibidora de la monoaminooxidas (MAO). Son útiles para el tratamiento de infecciones bacterianas.The invention provides novel oxazolidinone compounds of formula (I), in which A represents certain optionally substituted heterocycles; R1, R2, R3 and R4 are independently selected from -H and halogen; X is selected from O, S, NR9 and CR9R10; having R9 and R10 different meanings; Y is selected from O, S, SO, SO2, NO, NR12 and CR12R13, with R12 and R13 having different meanings. Different procedures are also provided for the preparation of said compounds. The oxazolidinone compounds of formula (I) are active against human and veterinary Gram-positive and some Gram-negative pathogens with a weak monoamine oxides (MAO) inhibitory activity. They are useful for the treatment of bacterial infections.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
UY29629A UY29629A1 (en) | 2006-06-27 | 2006-06-27 | OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAME |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
UY29629A UY29629A1 (en) | 2006-06-27 | 2006-06-27 | OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAME |
Publications (1)
Publication Number | Publication Date |
---|---|
UY29629A1 true UY29629A1 (en) | 2006-10-31 |
Family
ID=38813193
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY29629A UY29629A1 (en) | 2006-06-27 | 2006-06-27 | OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAME |
Country Status (1)
Country | Link |
---|---|
UY (1) | UY29629A1 (en) |
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2006
- 2006-06-27 UY UY29629A patent/UY29629A1/en unknown
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