UY29629A1 - OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAME - Google Patents

OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAME

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Publication number
UY29629A1
UY29629A1 UY29629A UY29629A UY29629A1 UY 29629 A1 UY29629 A1 UY 29629A1 UY 29629 A UY29629 A UY 29629A UY 29629 A UY29629 A UY 29629A UY 29629 A1 UY29629 A1 UY 29629A1
Authority
UY
Uruguay
Prior art keywords
oxazolidinone compounds
compounds
compositions
same
formula
Prior art date
Application number
UY29629A
Other languages
Spanish (es)
Inventor
Monserrat Cano
Albert Palomer
Antonio Guglietta
Original Assignee
Ferrer Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferrer Int filed Critical Ferrer Int
Priority to UY29629A priority Critical patent/UY29629A1/en
Publication of UY29629A1 publication Critical patent/UY29629A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención proporciona nuevos compuestos de oxazolidinona de fórmula (I), en la que A representa determinados heterociclos opcionalmente sustiutido; R1, R2, R3 y R4 se seleccionan independientemente de -H y halógeno; X se selecciona entre O,S, NR9 y CR9R10; teniendo R9 y R10 diferentes significados; Y se selecciona entre O, S, SO, SO2, NO, NR12 y CR12R13, teniendo R12 y R13 diferentes significados.También se proporcionan diferentes procedimientos para la preparación de dichos compuestos. Los compuestos de oxazolidinona de fórmula (I) son activos contra patógenos humanos y veterinarios Gram-positivos y algunos Gram-negativos con una débil actividad inhibidora de la monoaminooxidas (MAO). Son útiles para el tratamiento de infecciones bacterianas.The invention provides novel oxazolidinone compounds of formula (I), in which A represents certain optionally substituted heterocycles; R1, R2, R3 and R4 are independently selected from -H and halogen; X is selected from O, S, NR9 and CR9R10; having R9 and R10 different meanings; Y is selected from O, S, SO, SO2, NO, NR12 and CR12R13, with R12 and R13 having different meanings. Different procedures are also provided for the preparation of said compounds. The oxazolidinone compounds of formula (I) are active against human and veterinary Gram-positive and some Gram-negative pathogens with a weak monoamine oxides (MAO) inhibitory activity. They are useful for the treatment of bacterial infections.

UY29629A 2006-06-27 2006-06-27 OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAME UY29629A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
UY29629A UY29629A1 (en) 2006-06-27 2006-06-27 OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAME

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
UY29629A UY29629A1 (en) 2006-06-27 2006-06-27 OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAME

Publications (1)

Publication Number Publication Date
UY29629A1 true UY29629A1 (en) 2006-10-31

Family

ID=38813193

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29629A UY29629A1 (en) 2006-06-27 2006-06-27 OXAZOLIDINONE COMPOUNDS AND COMPOSITIONS AND PROCEDURES RELATED TO THE SAME

Country Status (1)

Country Link
UY (1) UY29629A1 (en)

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