UY29487A1 - "FLUORATED PIRIDINE N-OXIDES THROMBIN MODULATORS AND PROCESSES FOR N-OXIDATION OF NITROGEN HETEROARILES - Google Patents

"FLUORATED PIRIDINE N-OXIDES THROMBIN MODULATORS AND PROCESSES FOR N-OXIDATION OF NITROGEN HETEROARILES

Info

Publication number
UY29487A1
UY29487A1 UY29487A UY29487A UY29487A1 UY 29487 A1 UY29487 A1 UY 29487A1 UY 29487 A UY29487 A UY 29487A UY 29487 A UY29487 A UY 29487A UY 29487 A1 UY29487 A1 UY 29487A1
Authority
UY
Uruguay
Prior art keywords
oxidation
heteroariles
piridine
fluorated
oxides
Prior art date
Application number
UY29487A
Other languages
Spanish (es)
Inventor
Kevin Kreutter
Tianbao Lu
Yu Kai Lee
Christopher Teleha
Mark Player
Xizhen Zhu
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US11/385,056 external-priority patent/US7262210B2/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of UY29487A1 publication Critical patent/UY29487A1/en

Links

Abstract

La presente invención describe compuestos de Fórmula I donde X es: Y es: o una de sus sales aceptables para uso farmacéutico, para la profilaxis o el tratamiento de enfermedades y afecciones relacionadas con la actividad de trombina en un mamífero. La presente invención también se relaciona con un método novedoso de N-oxidación de heteroarilos nitrogenados.The present invention describes compounds of Formula I where X is: Y is: or one of its salts acceptable for pharmaceutical use, for the prophylaxis or treatment of diseases and conditions related to thrombin activity in a mammal. The present invention also relates to a novel method of N-oxidation of nitrogenous heteroaryls.

UY29487A 2005-04-20 2006-04-20 "FLUORATED PIRIDINE N-OXIDES THROMBIN MODULATORS AND PROCESSES FOR N-OXIDATION OF NITROGEN HETEROARILES UY29487A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US67313105P 2005-04-20 2005-04-20
US11/385,056 US7262210B2 (en) 2005-04-20 2006-03-21 Fluorinated pyridine N-oxide thrombin modulators and process for N-oxidation of nitrogen containing heteroaryls

Publications (1)

Publication Number Publication Date
UY29487A1 true UY29487A1 (en) 2006-06-30

Family

ID=38048149

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29487A UY29487A1 (en) 2005-04-20 2006-04-20 "FLUORATED PIRIDINE N-OXIDES THROMBIN MODULATORS AND PROCESSES FOR N-OXIDATION OF NITROGEN HETEROARILES

Country Status (2)

Country Link
AR (1) AR053590A1 (en)
UY (1) UY29487A1 (en)

Also Published As

Publication number Publication date
AR053590A1 (en) 2007-05-09

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