UY29295A1 - SULFONAMIDO-MACRICÍCLOS AND ITS SALTS, A PHARMACEUTICAL COMPOSITION THAT INCLUDES THESE COMPOUNDS, A METHOD OF PREPARATION AND THE USE OF THEM. - Google Patents
SULFONAMIDO-MACRICÍCLOS AND ITS SALTS, A PHARMACEUTICAL COMPOSITION THAT INCLUDES THESE COMPOUNDS, A METHOD OF PREPARATION AND THE USE OF THEM.Info
- Publication number
- UY29295A1 UY29295A1 UY29295A UY29295A UY29295A1 UY 29295 A1 UY29295 A1 UY 29295A1 UY 29295 A UY29295 A UY 29295A UY 29295 A UY29295 A UY 29295A UY 29295 A1 UY29295 A1 UY 29295A1
- Authority
- UY
- Uruguay
- Prior art keywords
- sulfonamido
- salts
- pharmaceutical composition
- compounds
- macricíclos
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 230000002074 deregulated effect Effects 0.000 abstract 2
- 230000006444 vascular growth Effects 0.000 abstract 2
- 102000009840 Angiopoietins Human genes 0.000 abstract 1
- 108010009906 Angiopoietins Proteins 0.000 abstract 1
- 101100481408 Danio rerio tie2 gene Proteins 0.000 abstract 1
- 101100481410 Mus musculus Tek gene Proteins 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000037824 growth disorder Diseases 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 230000011664 signaling Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Sulfonamido-macrocíclos de acuerdo con la Fórmula general I y sus sales, composiciones farmacéuticas que comprenden los sulfonamido-macrocíclos y un método para preparar los sulfonamido-macrocíclos así como su uso para fabricar una composición farmacéutica para el tratamiento de enfermedades de crecimiento vascular desregulado o de enfermedades acompanadas por un crecimiento vascular desregulado, donde los compuestos interfieren en forma efectiva con la angiopoyetina y por lo tanto afectan la senalización de Tie2. donde R1, R2, y R3 tienen los valores que se les asigna en la memoria descriptiva y en las reivindicaciones.Sulfonamido-macrocycles according to General Formula I and its salts, pharmaceutical compositions comprising sulfonamido-macrocycles and a method for preparing sulfonamido-macrocycles as well as their use to manufacture a pharmaceutical composition for the treatment of deregulated vascular growth diseases or of diseases accompanied by deregulated vascular growth, where the compounds effectively interfere with angiopoietin and therefore affect the signaling of Tie2. where R1, R2, and R3 have the values assigned to them in the specification and in the claims.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
UY29295A UY29295A1 (en) | 2005-12-21 | 2005-12-21 | SULFONAMIDO-MACRICÍCLOS AND ITS SALTS, A PHARMACEUTICAL COMPOSITION THAT INCLUDES THESE COMPOUNDS, A METHOD OF PREPARATION AND THE USE OF THEM. |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
UY29295A UY29295A1 (en) | 2005-12-21 | 2005-12-21 | SULFONAMIDO-MACRICÍCLOS AND ITS SALTS, A PHARMACEUTICAL COMPOSITION THAT INCLUDES THESE COMPOUNDS, A METHOD OF PREPARATION AND THE USE OF THEM. |
Publications (1)
Publication Number | Publication Date |
---|---|
UY29295A1 true UY29295A1 (en) | 2006-07-31 |
Family
ID=38813128
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY29295A UY29295A1 (en) | 2005-12-21 | 2005-12-21 | SULFONAMIDO-MACRICÍCLOS AND ITS SALTS, A PHARMACEUTICAL COMPOSITION THAT INCLUDES THESE COMPOUNDS, A METHOD OF PREPARATION AND THE USE OF THEM. |
Country Status (1)
Country | Link |
---|---|
UY (1) | UY29295A1 (en) |
-
2005
- 2005-12-21 UY UY29295A patent/UY29295A1/en not_active Application Discontinuation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20160606 |