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Application filed by Hoffmann La RochefiledCriticalHoffmann La Roche
Priority to UY27303ApriorityCriticalpatent/UY27303A1/en
Publication of UY27303A1publicationCriticalpatent/UY27303A1/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
Esta invención se refiere a derivados de 4-aminopirimidina de fórmula general I en donde R1 R2 R3 y R4 tienen los significados definidos en la especificación y sus sales farmacéuticamente aceptables. La invención además se refiere a la preparación de tales compuestos, a medicamentos que contengan tales compuestos y a su uso para la prevención o tratamiento de trastornos mediados por el receptor MGLUR5.This invention relates to 4-aminopyrimidine derivatives of general formula I wherein R1 R2 R3 and R4 have the meanings defined in the specification and their pharmaceutically acceptable salts. The invention further relates to the preparation of such compounds, to medicaments containing such compounds and to their use for the prevention or treatment of disorders mediated by the MGLUR5 receptor.
DERIVATIVES OF BENZOCONDENSED HETEROARILAMIDE OF USEFUL TIENOPIRIDINS AS THERAPEUTIC AGENTS, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THE SAME AND METHODS FOR USE
SUBSTITUTED DERIVATIVES OF N4- (5-METHYL-1H-PIRAZOL-3-IL) - 1,3,5-TRIAZINA-2,4-DIAMINE, THEIR ENANTIOMERS, PHARMACEUTICALLY ACCEPTABLE SALTS OF THE SAME, COMPOSITIONS, PREPARATION PROCESSES AND APPLICATIONS
DERIVATIVES OF 5, 6, 7, 8 - TETRAHYDROIMIDAZO [1,5A] PIRIDINE WITH INHIBITORY ACTIVITY OF ALDOSTERONE SYNTHEASE, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THE PREPARATION OF MEDICINES FOR THE TREATMENT OF HYPERALDOSINDISM.
COMPOSITE OF HETEROARIL SULFONAMIDE REPLACED, PROCEDURE FOR THE PREPARATION OF THE SAME, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND ITS USE TO PREPARE A MEDICINAL PRODUCT
DERIVATIVES OF ARILPIPERAZINIL-CICLOHEXIL INDOL, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM AND THE USE OF THE SAME FOR THE MANUFACTURE OF MEDICINES FOR THE TREATMENT OF DEPRESSION