UY25233A1 - BIOISOSTERIC SUBSTITUTION OF CATECOL BY INDAZOL IN THERAPEUTICALLY ACTIVE COMPOUNDS - Google Patents

BIOISOSTERIC SUBSTITUTION OF CATECOL BY INDAZOL IN THERAPEUTICALLY ACTIVE COMPOUNDS

Info

Publication number
UY25233A1
UY25233A1 UY25233A UY25233A UY25233A1 UY 25233 A1 UY25233 A1 UY 25233A1 UY 25233 A UY25233 A UY 25233A UY 25233 A UY25233 A UY 25233A UY 25233 A1 UY25233 A1 UY 25233A1
Authority
UY
Uruguay
Prior art keywords
therapeutically active
catecol
indazol
active compounds
substitution
Prior art date
Application number
UY25233A
Other languages
Spanish (es)
Inventor
Anthony Marfat
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of UY25233A1 publication Critical patent/UY25233A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Composiciones terapéuticamente activas de materia y tipos de miembros de las mismas que comprenden compuestos que contienen indazol, resultando dichos compuestos y su actividad terapéutica directamente de una sustitución biosostérica de atecol por indazol de un compuesto que contienen catecol que tiene dicha actividad terapéutica, donde los substituyentes no catecol son los mismos u homólogos antes y después de dicha sustitución, en la que dichas composiciones de materia comprenden un compuesto de fórmula (I1)o (I2).Therapeutically active compositions of matter and types of members thereof comprising indazole-containing compounds, said compounds and their therapeutic activity resulting directly from a biososteric substitution of atecol for indazole of a catechol-containing compound having said therapeutic activity, where the substituents non-catechol are the same or homologous before and after said substitution, in which said compositions of matter comprise a compound of formula (I1) or (I2).

UY25233A 1997-11-04 1998-11-04 BIOISOSTERIC SUBSTITUTION OF CATECOL BY INDAZOL IN THERAPEUTICALLY ACTIVE COMPOUNDS UY25233A1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US6418797P 1997-11-04 1997-11-04
US6422997P 1997-11-04 1997-11-04
US6402497P 1997-11-04 1997-11-04
US6419897P 1997-11-04 1997-11-04

Publications (1)

Publication Number Publication Date
UY25233A1 true UY25233A1 (en) 2000-12-29

Family

ID=38812097

Family Applications (1)

Application Number Title Priority Date Filing Date
UY25233A UY25233A1 (en) 1997-11-04 1998-11-04 BIOISOSTERIC SUBSTITUTION OF CATECOL BY INDAZOL IN THERAPEUTICALLY ACTIVE COMPOUNDS

Country Status (1)

Country Link
UY (1) UY25233A1 (en)

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Legal Events

Date Code Title Description
DESI Application deemed to be withdrawn

Effective date: 20071105