UA92047C2 - Carbonylamino pyrrolopyrazoles, potent kinase inhibitors - Google Patents

Carbonylamino pyrrolopyrazoles, potent kinase inhibitors

Info

Publication number
UA92047C2
UA92047C2 UAA200807387A UAA200807387A UA92047C2 UA 92047 C2 UA92047 C2 UA 92047C2 UA A200807387 A UAA200807387 A UA A200807387A UA A200807387 A UAA200807387 A UA A200807387A UA 92047 C2 UA92047 C2 UA 92047C2
Authority
UA
Ukraine
Prior art keywords
kinase inhibitors
pyrrolopyrazoles
carbonylamino
potent kinase
compounds
Prior art date
Application number
UAA200807387A
Other languages
Russian (ru)
Ukrainian (uk)
Inventor
Лімін Дун
Чансін Ґо
Юйфен Хун
Мари Кетрін Джонсон
Сюзан Елізабет Кефарт
Хайтао Лі
Індроун Джеймс Макалпін
Джаяшрі Ґіріш Тікге
Аньле Ян
Цеюньху Чжан
Original Assignee
Пфайзер Продактс Інк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Пфайзер Продактс Інк. filed Critical Пфайзер Продактс Інк.
Priority claimed from PCT/IB2006/003646 external-priority patent/WO2007072153A2/en
Publication of UA92047C2 publication Critical patent/UA92047C2/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Carbonyiamino Pyirolopyrazole compounds of formula (I), compositions including these compounds and methods of their use are provided. Preferred compounds of formula (I) have activity as protein kinase inhibitors, including as inhibitors of PAK4. EMBED ISISServer I
UAA200807387A 2005-12-21 2006-12-12 Carbonylamino pyrrolopyrazoles, potent kinase inhibitors UA92047C2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US75334905P 2005-12-21 2005-12-21
US86493206P 2006-11-08 2006-11-08
PCT/IB2006/003646 WO2007072153A2 (en) 2005-12-21 2006-12-12 Carbonylamino pyrrolopyrazoles, potent kinase inhibitors

Publications (1)

Publication Number Publication Date
UA92047C2 true UA92047C2 (en) 2010-09-27

Family

ID=40247953

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200807387A UA92047C2 (en) 2005-12-21 2006-12-12 Carbonylamino pyrrolopyrazoles, potent kinase inhibitors

Country Status (5)

Country Link
CN (1) CN101346382B (en)
SI (1) SI1979356T1 (en)
TN (1) TNSN08274A1 (en)
UA (1) UA92047C2 (en)
ZA (1) ZA200804667B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113234081A (en) * 2021-05-27 2021-08-10 东南大学 Preparation method of pyrrolopyrazole derivative and DMDPEDA as urea

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA81790C2 (en) * 2002-12-19 2008-02-11 Фармация Италия С.П.А. Substituted derivatives of pyrolopyrazol as kinaze inhibitors

Also Published As

Publication number Publication date
SI1979356T1 (en) 2013-11-29
ZA200804667B (en) 2010-05-26
CN101346382B (en) 2011-07-06
CN101346382A (en) 2009-01-14
TNSN08274A1 (en) 2009-10-30

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