UA87845C2 - Thienopyridinone compounds and methods of treatment of nervous system disorders - Google Patents

Thienopyridinone compounds and methods of treatment of nervous system disorders

Info

Publication number
UA87845C2
UA87845C2 UAA200613298A UAA200613298A UA87845C2 UA 87845 C2 UA87845 C2 UA 87845C2 UA A200613298 A UAA200613298 A UA A200613298A UA A200613298 A UAA200613298 A UA A200613298A UA 87845 C2 UA87845 C2 UA 87845C2
Authority
UA
Ukraine
Prior art keywords
disorders
methods
treatment
nervous system
system disorders
Prior art date
Application number
UAA200613298A
Other languages
Russian (ru)
Ukrainian (uk)
Inventor
Шай Бар-Хаим
Орен Бекер
Донли Чень
Дейл С. Даноа
Александр Хейфетц
Мерседес Лобера
Яел Марантц
Прадиумна Моханти
Сильвия Нойман
Шарон Шачем
Лоуренс Ву
Original Assignee
Эпикс Делавер, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Эпикс Делавер, Инк. filed Critical Эпикс Делавер, Инк.
Publication of UA87845C2 publication Critical patent/UA87845C2/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

The invention relates to 5-HT receptor agonists and partial agonists. Novel thienopyridinone compounds represented by Formula I, and synthesis and uses thereof for treating diseases mediated directly or indirectly by 5-HT receptors, are disclosed. Such conditions include Alzheimer's disease, cognition disorders, irritable bowel syndrome, nausea, emesis, vomiting, prokinesia, gastroesophageal reflux disease, nonulcer dyspepsia, depression, anxiety, urinary incontinence, migraine, arrhythmia, atrial fibrillation, ischemic stroke, gastritis, gastric emptying disorders, feeding disorders, gastrointestinal disorders, constipation, erectile dysfunction, and respiratory depression. Methods of preparation and novel intermediates and pharmaceutical salts thereof are also included.
UAA200613298A 2004-05-17 2005-05-16 Thienopyridinone compounds and methods of treatment of nervous system disorders UA87845C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57185204P 2004-05-17 2004-05-17

Publications (1)

Publication Number Publication Date
UA87845C2 true UA87845C2 (en) 2009-08-25

Family

ID=38716194

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200613298A UA87845C2 (en) 2004-05-17 2005-05-16 Thienopyridinone compounds and methods of treatment of nervous system disorders

Country Status (3)

Country Link
CN (1) CN101031299A (en)
UA (1) UA87845C2 (en)
ZA (1) ZA200609213B (en)

Also Published As

Publication number Publication date
CN101031299A (en) 2007-09-05
ZA200609213B (en) 2007-10-31

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