UA86777C2 - 6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors - Google Patents
6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitorsInfo
- Publication number
- UA86777C2 UA86777C2 UAA200603731A UAA200603731A UA86777C2 UA 86777 C2 UA86777 C2 UA 86777C2 UA A200603731 A UAA200603731 A UA A200603731A UA A200603731 A UAA200603731 A UA A200603731A UA 86777 C2 UA86777 C2 UA 86777C2
- Authority
- UA
- Ukraine
- Prior art keywords
- quinoxalinones
- quinolinones
- adp
- ribose
- alkenyl
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
The present invention provides compounds of formula (I) and compounds of formula (I), (VII-a), as well as pharmaceutical compositions comprising said compounds and their use as PARP inhibitors wherein n, RR, R, R, R, R, R, R, Rand X have defined meanings.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP0313028 | 2003-11-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
UA86777C2 true UA86777C2 (en) | 2009-05-25 |
Family
ID=34957030
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA200603731A UA86777C2 (en) | 2003-11-20 | 2004-11-18 | 6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors |
Country Status (3)
Country | Link |
---|---|
CN (1) | CN1882547B (en) |
UA (1) | UA86777C2 (en) |
ZA (1) | ZA200604075B (en) |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2002864C (en) * | 1988-11-29 | 1999-11-16 | Eddy J. E. Freyne | (1h-azol-1-ylmethyl) substituted quinoline, quinazoline or quinoxaline derivatives |
-
2004
- 2004-11-18 UA UAA200603731A patent/UA86777C2/en unknown
- 2004-11-18 CN CN2004800341763A patent/CN1882547B/en not_active Expired - Fee Related
-
2006
- 2006-05-19 ZA ZA200604075A patent/ZA200604075B/en unknown
Also Published As
Publication number | Publication date |
---|---|
ZA200604075B (en) | 2007-09-26 |
CN1882547B (en) | 2011-04-13 |
CN1882547A (en) | 2006-12-20 |
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