UA85554U - PROCESS FOR THE PREPARATION OF 1-CYCLOPROPYL-6-FLUORO-1,4-DIHYDRO-8-METHOXY-7-[(4AS,7AS)-OCTAHYDRO-6H-PYRROLO[3,4-b]PYRIDINE-6-YL]-4-OXO-3-QUINOLINECARBOXYLIC ACID) - Google Patents
PROCESS FOR THE PREPARATION OF 1-CYCLOPROPYL-6-FLUORO-1,4-DIHYDRO-8-METHOXY-7-[(4AS,7AS)-OCTAHYDRO-6H-PYRROLO[3,4-b]PYRIDINE-6-YL]-4-OXO-3-QUINOLINECARBOXYLIC ACID)Info
- Publication number
- UA85554U UA85554U UAU201305963U UAU201305963U UA85554U UA 85554 U UA85554 U UA 85554U UA U201305963 U UAU201305963 U UA U201305963U UA U201305963 U UAU201305963 U UA U201305963U UA 85554 U UA85554 U UA 85554U
- Authority
- UA
- Ukraine
- Prior art keywords
- oxo
- preparation
- octahydro
- pyrrolo
- cyclopropyl
- Prior art date
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
A process for the preparation of 1-cyclopropyl-6-fluoro-1,4-dihydro-8-methoxy-7-[(4AS,7AS)-octahydro-6H-pyrrolo[3,4-b]pyridine-6-yl]-4-oxo-3-quinolinecarboxylic acid consists in addition of heterocyclic amine comprising protective group to ethyl-3-oxo-3-(2,4,5-trifluoro-3-methoxyphenyl)propanoate followed by interaction with triethylorthoformiate, addition of cyclic amine, further cyclization and preparation of desired product.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
UAU201305963U UA85554U (en) | 2013-05-13 | 2013-05-13 | PROCESS FOR THE PREPARATION OF 1-CYCLOPROPYL-6-FLUORO-1,4-DIHYDRO-8-METHOXY-7-[(4AS,7AS)-OCTAHYDRO-6H-PYRROLO[3,4-b]PYRIDINE-6-YL]-4-OXO-3-QUINOLINECARBOXYLIC ACID) |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
UAU201305963U UA85554U (en) | 2013-05-13 | 2013-05-13 | PROCESS FOR THE PREPARATION OF 1-CYCLOPROPYL-6-FLUORO-1,4-DIHYDRO-8-METHOXY-7-[(4AS,7AS)-OCTAHYDRO-6H-PYRROLO[3,4-b]PYRIDINE-6-YL]-4-OXO-3-QUINOLINECARBOXYLIC ACID) |
Publications (1)
Publication Number | Publication Date |
---|---|
UA85554U true UA85554U (en) | 2013-11-25 |
Family
ID=52285072
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAU201305963U UA85554U (en) | 2013-05-13 | 2013-05-13 | PROCESS FOR THE PREPARATION OF 1-CYCLOPROPYL-6-FLUORO-1,4-DIHYDRO-8-METHOXY-7-[(4AS,7AS)-OCTAHYDRO-6H-PYRROLO[3,4-b]PYRIDINE-6-YL]-4-OXO-3-QUINOLINECARBOXYLIC ACID) |
Country Status (1)
Country | Link |
---|---|
UA (1) | UA85554U (en) |
-
2013
- 2013-05-13 UA UAU201305963U patent/UA85554U/en unknown
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