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Application filed by Національна Фармацевтична Академія УкраїниfiledCriticalНаціональна Фармацевтична Академія України
Priority to UA4422129ApriorityCriticalpatent/UA46179A1/en
Publication of UA46179A1publicationCriticalpatent/UA46179A1/en
Organic Low-Molecular-Weight Compounds And Preparation Thereof
(AREA)
Abstract
The invention relates to the amides of carbonic acids, in particular N-methylamide of 4-acetyl oxanilic acid. The substance possesses the hemostatic activity. The aim consists in searching for less toxic and more effective compound. The substance mentioned above is synthesized in the reaction of ethyl ester of 4-acetyl oxanilic acid with methylamine in the medium of dioxan. The yield is 95%. The melting point is 247 - 249°С; LD50 285 mg/kg.
UA4422129A1988-05-061988-05-06
N-METHYLAMIDE OF 4-ACETYLOXANYLIC ACID, WHICH SHOWS HEMOSTATIC ACTIVITY
UA46179A1
(en)
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