UA112586C2 - BENZIMIDAZOLPROLINE DERIVATIVES - Google Patents
BENZIMIDAZOLPROLINE DERIVATIVESInfo
- Publication number
- UA112586C2 UA112586C2 UAA201413919A UAA201413919A UA112586C2 UA 112586 C2 UA112586 C2 UA 112586C2 UA A201413919 A UAA201413919 A UA A201413919A UA A201413919 A UAA201413919 A UA A201413919A UA 112586 C2 UA112586 C2 UA 112586C2
- Authority
- UA
- Ukraine
- Prior art keywords
- benzimidazolproline
- derivatives
- formula
- compounds
- pharmaceuticals
- Prior art date
Links
Abstract
Даний винахід належить до сполук формули (І), Формула (I)де Аr, R, R, R, R, Rта (R)приймають значення, як описано у описі, до їх одержання, до їх фармацевтично прийнятних солей та до їх застосування як фармацевтичних засобів, до фармацевтичних композицій, що містять одну або більше сполук формули (І), та особливо до їх застосування як антагоністів рецептора орексину.The present invention relates to compounds of formula (I), Formula (I) where Ar, R, R, R, R, R and (R) take the values as described in the description, to obtain them, to their pharmaceutically acceptable salts and to their use as pharmaceuticals, to pharmaceutical compositions containing one or more compounds of formula (I), and in particular to their use as orexin receptor antagonists.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP12170748 | 2012-06-04 | ||
PCT/IB2013/054567 WO2013182972A1 (en) | 2012-06-04 | 2013-06-03 | Benzimidazole-proline derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
UA112586C2 true UA112586C2 (en) | 2016-09-26 |
Family
ID=54338069
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA201413919A UA112586C2 (en) | 2012-06-04 | 2013-03-06 | BENZIMIDAZOLPROLINE DERIVATIVES |
Country Status (2)
Country | Link |
---|---|
MA (1) | MA37741B1 (en) |
UA (1) | UA112586C2 (en) |
-
2013
- 2013-03-06 UA UAA201413919A patent/UA112586C2/en unknown
-
2015
- 2015-01-02 MA MA37741A patent/MA37741B1/en unknown
Also Published As
Publication number | Publication date |
---|---|
MA20150282A2 (en) | 2015-08-31 |
MA37741B1 (en) | 2017-01-31 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA201401351A1 (en) | DERIVATIVES OF BENZIMIDAZOL-PROLINE | |
CY1123365T1 (en) | COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENORECTOR AGENT ACTIVITY | |
EA201591195A1 (en) | NEW QUINOLON DERIVATIVES | |
UA109010C2 (en) | Morpholino pyrividines and their use in therapy | |
IN2014CN04127A (en) | ||
PH12014502363A1 (en) | N-aryltriazole compounds as lpar antagonists | |
PH12014502789A1 (en) | N-alkyltriazole compounds as lpar antagonists | |
UA111640C2 (en) | DERIVATIVES [1,2,3] TRIAZOLO [4,5-d] PYRIMIDINE AS A cannabinoid receptor agonist 2 | |
PH12014501514A1 (en) | New azetidine derivatives, pharmaceutical compositions and uses thereof | |
IN2014CN04530A (en) | ||
EA201201050A1 (en) | PYRAZOLES AS AN ANTAGONISTS CRTH2 | |
EA201291217A1 (en) | PHARMACEUTICAL COMPOSITIONS CONTAINING DERIVATIVES 1- (β-D-GLUKOPIRANOSIL) -2-THIENYLMETYLBENZENE AS NZGT INHIBITORS | |
JO3154B1 (en) | Trpv4 antagonists | |
EA202091262A1 (en) | Piperidine Receptor Modulators CXCR7 | |
EA201501163A1 (en) | CXCR7 RECEPTOR MODULATORS | |
EA201400822A1 (en) | DERIVATIVES OF HETEROCYCLIC AMIDES AS AN ANTAGONISTS OF P2HRECEPTOR | |
PH12014502364A1 (en) | Substituted pyrazole compounds as lpar antagonists | |
EA201600434A1 (en) | APPLICATION OF DERIVATIVES OF BENZIMIDAZOLPROLINE | |
NZ734542A (en) | Hydroxyalkyl-piperazine derivatives as cxcr3 receptor modulators | |
MX2017009292A (en) | (r)-2-methyl-piperazine derivatives as cxcr3 receptor modulators. | |
EA201600394A1 (en) | TRICYCLIC COMPOUNDS OF PIPERIDINE | |
EA201300857A1 (en) | PYRAZOLES AS AN ANTAGONISTS CRTH2 | |
EA201600123A1 (en) | DERIVATIVES 1- (PIPERAZIN-1-IL) -2 - ([1,2,4] TRIAZOL-1-IL) ETHANON | |
UA112586C2 (en) | BENZIMIDAZOLPROLINE DERIVATIVES | |
EA201590886A1 (en) | SUBSTITUTED INDOLA DERIVATIVES |