UA105675C2 - Benzodiazepine bromodomain inhibitor - Google Patents

Benzodiazepine bromodomain inhibitor

Info

Publication number
UA105675C2
UA105675C2 UAA201205470A UAA201205470A UA105675C2 UA 105675 C2 UA105675 C2 UA 105675C2 UA A201205470 A UAA201205470 A UA A201205470A UA A201205470 A UAA201205470 A UA A201205470A UA 105675 C2 UA105675 C2 UA 105675C2
Authority
UA
Ukraine
Prior art keywords
bromodomain inhibitor
benzodiazepine
benzodiazepine bromodomain
compound
inhibitor
Prior art date
Application number
UAA201205470A
Other languages
Russian (ru)
Ukrainian (uk)
Inventor
Ромейн Люк Марі Ґосміні
Олівер Мірґует
Original Assignee
Ґлаксосмітклайн Ллк
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ґлаксосмітклайн Ллк filed Critical Ґлаксосмітклайн Ллк
Priority claimed from PCT/EP2010/061518 external-priority patent/WO2011054553A1/en
Publication of UA105675C2 publication Critical patent/UA105675C2/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The present invention relates to a benzodiazepine compound of formula (I), processes for its preparation, pharmaceutical compositions containing such a compound and to its use in therapy.
UAA201205470A 2009-11-05 2010-08-06 Benzodiazepine bromodomain inhibitor UA105675C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0919433A GB0919433D0 (en) 2009-11-05 2009-11-05 Novel compounds
PCT/EP2010/061518 WO2011054553A1 (en) 2009-11-05 2010-08-06 Benzodiazepine bromodomain inhibitor

Publications (1)

Publication Number Publication Date
UA105675C2 true UA105675C2 (en) 2014-06-10

Family

ID=41501976

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201205470A UA105675C2 (en) 2009-11-05 2010-08-06 Benzodiazepine bromodomain inhibitor

Country Status (2)

Country Link
GB (1) GB0919433D0 (en)
UA (1) UA105675C2 (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2742035C2 (en) * 2015-11-25 2021-02-01 Дана-Фарбер Кэнсер Инститьют, Инк. Bivalent bromodomain inhibitors and routes of use thereof
US11406645B2 (en) 2015-09-11 2022-08-09 Dana-Farber Cancer Institute, Inc. Acetamide thienotriazolodiazepines and uses thereof

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11406645B2 (en) 2015-09-11 2022-08-09 Dana-Farber Cancer Institute, Inc. Acetamide thienotriazolodiazepines and uses thereof
RU2742035C2 (en) * 2015-11-25 2021-02-01 Дана-Фарбер Кэнсер Инститьют, Инк. Bivalent bromodomain inhibitors and routes of use thereof

Also Published As

Publication number Publication date
GB0919433D0 (en) 2009-12-23

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