UA103208C2 - 2-[(5-chloro-2-{[3-methyl-1-(1-methylethyl)-1h-pyrazol-5-yl]amino}-4-pyridinyl)amino]-n-methylbenzamide as focal adhesion kinase (fak) inhibitor - Google Patents

2-[(5-chloro-2-{[3-methyl-1-(1-methylethyl)-1h-pyrazol-5-yl]amino}-4-pyridinyl)amino]-n-methylbenzamide as focal adhesion kinase (fak) inhibitor

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Publication number
UA103208C2
UA103208C2 UAA201106674A UAA201106674A UA103208C2 UA 103208 C2 UA103208 C2 UA 103208C2 UA A201106674 A UAA201106674 A UA A201106674A UA A201106674 A UAA201106674 A UA A201106674A UA 103208 C2 UA103208 C2 UA 103208C2
Authority
UA
Ukraine
Prior art keywords
amino
fak
methylbenzamide
pyrazol
methylethyl
Prior art date
Application number
UAA201106674A
Other languages
Russian (ru)
Ukrainian (uk)
Inventor
Джерри Лерой Адамс
Томас Х. Фейтг
Нейл В. Джонсон
Хонг Лин
Иржи Каспарец
Марк Меллинджер
Синь Пенг
Рен Се
Original Assignee
Глаксосмитклайн Ллс
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Глаксосмитклайн Ллс filed Critical Глаксосмитклайн Ллс
Priority claimed from PCT/US2009/062163 external-priority patent/WO2010062578A1/en
Publication of UA103208C2 publication Critical patent/UA103208C2/en

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Abstract

The present invention relates to a compound of formula (I) or a pharmaceutically acceptable salt thereof, wherein R, R, R, R, R, R, Q, Z, and p are as described herein. Compounds of the present invention are useful for the treatment of cancers., (I)
UAA201106674A 2008-10-27 2009-10-27 2-[(5-chloro-2-{[3-methyl-1-(1-methylethyl)-1h-pyrazol-5-yl]amino}-4-pyridinyl)amino]-n-methylbenzamide as focal adhesion kinase (fak) inhibitor UA103208C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10856808P 2008-10-27 2008-10-27
PCT/US2009/062163 WO2010062578A1 (en) 2008-10-27 2009-10-27 Pyrazolylaminopyridines as inhibitors of fak

Publications (1)

Publication Number Publication Date
UA103208C2 true UA103208C2 (en) 2013-09-25

Family

ID=52278871

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201106674A UA103208C2 (en) 2008-10-27 2009-10-27 2-[(5-chloro-2-{[3-methyl-1-(1-methylethyl)-1h-pyrazol-5-yl]amino}-4-pyridinyl)amino]-n-methylbenzamide as focal adhesion kinase (fak) inhibitor

Country Status (1)

Country Link
UA (1) UA103208C2 (en)

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