TW202430507A - 新穎atp-敏感性鉀通道增效劑、其製備及用途 - Google Patents

新穎atp-敏感性鉀通道增效劑、其製備及用途 Download PDF

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Publication number
TW202430507A
TW202430507A TW112139862A TW112139862A TW202430507A TW 202430507 A TW202430507 A TW 202430507A TW 112139862 A TW112139862 A TW 112139862A TW 112139862 A TW112139862 A TW 112139862A TW 202430507 A TW202430507 A TW 202430507A
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TW
Taiwan
Prior art keywords
preparation
potentiators
potassium channel
sensitive potassium
hyperinsulinism
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TW112139862A
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English (en)
Inventor
皮耶特 維傑尼克
德 桑迪 克勞汀 凡
博特蘭 維偉特
羅倫斯 安 梅維勒
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美商律森製藥股份有限公司
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Application filed by 美商律森製藥股份有限公司 filed Critical 美商律森製藥股份有限公司
Publication of TW202430507A publication Critical patent/TW202430507A/zh

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Abstract

本發明係關於通式(I)化合物或其醫藥上可接受之鹽、溶劑合物及/或水合物、其製備方法、該等化合物用作藥劑之用途及其等於治療及/或預防疾病或疾患之用途。在一實施例中,該疾病或疾患係高胰島素血症,特定言之先天性高胰島素血症。本發明亦係關於包含通式(I)化合物及醫藥上可接受之載劑之醫藥組合物及其用作藥劑之用途,特定言之其於治療疾病或疾患(諸如高胰島素血症或先天性高胰島素血症)之用途。
TW112139862A 2022-10-18 2023-10-18 新穎atp-敏感性鉀通道增效劑、其製備及用途 TW202430507A (zh)

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NL2033343 2022-10-18

Publications (1)

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TW202430507A true TW202430507A (zh) 2024-08-01

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