TW200603782A - (1,10b-dihydro-2-(aminocarbonyl-phenyl)-5h-pyrazolo[1,5-c][1,3]benzoxazin-5-yl)phenyl methanone derivatives as hiv viral replication inhibitors - Google Patents

(1,10b-dihydro-2-(aminocarbonyl-phenyl)-5h-pyrazolo[1,5-c][1,3]benzoxazin-5-yl)phenyl methanone derivatives as hiv viral replication inhibitors

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Publication number
TW200603782A
TW200603782A TW094114158A TW94114158A TW200603782A TW 200603782 A TW200603782 A TW 200603782A TW 094114158 A TW094114158 A TW 094114158A TW 94114158 A TW94114158 A TW 94114158A TW 200603782 A TW200603782 A TW 200603782A
Authority
TW
Taiwan
Prior art keywords
phenyl
benzoxazin
pyrazolo
viral replication
present
Prior art date
Application number
TW094114158A
Other languages
Chinese (zh)
Inventor
Abdellah Tahri
Lieve Emma Jan Michiels
Acker Koenraad Lodewijk August Van
Dominique Louis Nestor Surleraux
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Publication of TW200603782A publication Critical patent/TW200603782A/en

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Abstract

The present invention relates to 5H-pyrazolo[1,5-c][1,3]benzoxazin-5-y1) phenyl methanone derivatives as inhibitors of the viral replication of the HIV virus, processes for their preparation as well as pharmaceutical compositions, their use as medicines, and diagnostic kits comprising them. The present invention also concerns combinations of the present HIV inhibitors with other anti-retroviral agents. It further relates to their use in assays as reference compounds or as reagents. The compounds of the present invention are useful for preventing or treating infection by HIV and for treating AIDS.
TW094114158A 2004-05-04 2005-05-03 (1,10b-dihydro-2-(aminocarbonyl-phenyl)-5h-pyrazolo[1,5-c][1,3]benzoxazin-5-yl)phenyl methanone derivatives as hiv viral replication inhibitors TW200603782A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04101913 2004-05-04
US60427504P 2004-08-25 2004-08-25

Publications (1)

Publication Number Publication Date
TW200603782A true TW200603782A (en) 2006-02-01

Family

ID=57807079

Family Applications (1)

Application Number Title Priority Date Filing Date
TW094114158A TW200603782A (en) 2004-05-04 2005-05-03 (1,10b-dihydro-2-(aminocarbonyl-phenyl)-5h-pyrazolo[1,5-c][1,3]benzoxazin-5-yl)phenyl methanone derivatives as hiv viral replication inhibitors

Country Status (1)

Country Link
TW (1) TW200603782A (en)

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