TR200806302A2 - Solubility and stability enhancing pharmaceutical formulation. - Google Patents

Solubility and stability enhancing pharmaceutical formulation.

Info

Publication number
TR200806302A2
TR200806302A2 TR2008/06302A TR200806302A TR200806302A2 TR 200806302 A2 TR200806302 A2 TR 200806302A2 TR 2008/06302 A TR2008/06302 A TR 2008/06302A TR 200806302 A TR200806302 A TR 200806302A TR 200806302 A2 TR200806302 A2 TR 200806302A2
Authority
TR
Turkey
Prior art keywords
solubility
pharmaceutical formulation
stability enhancing
enhancing pharmaceutical
stability
Prior art date
Application number
TR2008/06302A
Other languages
Turkish (tr)
Inventor
Bi̇lgi̇ç Mahmut
Original Assignee
Bi̇lgi̇ç Mahmut
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bi̇lgi̇ç Mahmut filed Critical Bi̇lgi̇ç Mahmut
Priority to TR2008/06302A priority Critical patent/TR200806302A2/en
Priority to PCT/TR2009/000109 priority patent/WO2010021609A1/en
Publication of TR200806302A2 publication Critical patent/TR200806302A2/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • A61K31/366Lactones having six-membered rings, e.g. delta-lactones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin

Abstract

Mevcut buluş, çözünürlük sorunu olan bir aktif maddeyi stabilite sorunu olan bir terapötik ajanla kombinasyon halinde içeren farmasötik formülasyonlara, bunların hazırlanma yöntemlerine ve tıbbi kullanımlarına ilişkindir.The present invention relates to pharmaceutical formulations, methods of preparation and medical uses comprising an active substance having a solubility problem in combination with a therapeutic agent having a stability problem.

TR2008/06302A 2008-08-22 2008-08-22 Solubility and stability enhancing pharmaceutical formulation. TR200806302A2 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
TR2008/06302A TR200806302A2 (en) 2008-08-22 2008-08-22 Solubility and stability enhancing pharmaceutical formulation.
PCT/TR2009/000109 WO2010021609A1 (en) 2008-08-22 2009-08-24 Solubility and stability enhancing pharmaceutical formulation

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
TR2008/06302A TR200806302A2 (en) 2008-08-22 2008-08-22 Solubility and stability enhancing pharmaceutical formulation.

Publications (1)

Publication Number Publication Date
TR200806302A2 true TR200806302A2 (en) 2010-03-22

Family

ID=41396995

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2008/06302A TR200806302A2 (en) 2008-08-22 2008-08-22 Solubility and stability enhancing pharmaceutical formulation.

Country Status (2)

Country Link
TR (1) TR200806302A2 (en)
WO (1) WO2010021609A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011002424A2 (en) * 2009-07-02 2011-01-06 Bilgic Mahmut Solubility and stability enchancing pharmaceutical formulation

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR040588A1 (en) * 2002-07-26 2005-04-13 Schering Corp PHARMACEUTICAL FORMULATION INCLUDING AN INHIBITOR OF CHOLESTEROL ABSORPTION AND AN INHIBITOR OF A HMGCO TO REDUCTASE
WO2006134604A1 (en) * 2005-06-15 2006-12-21 Hetero Drugs Limited Combination composition of cholesterol absorption inhibitor and 3-hydroxy-3-methylglutaryl-coenzyme a (hmg-coa) reductase inhibitor
EP1741427A1 (en) * 2005-07-06 2007-01-10 KRKA, D.D., Novo Mesto Pharmaceutical composition comprising simvastatin and ezetimibe
EP1905424A3 (en) * 2006-02-02 2008-04-30 Ranbaxy Laboratories Limited Process for the preparation of a pharmaceutical composition comprising stabilized statin particles
EP2120882A2 (en) * 2007-02-23 2009-11-25 Krka Pharmaceutical composition containing a cholesterol absorption inhibitor

Also Published As

Publication number Publication date
WO2010021609A1 (en) 2010-02-25

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