TNSN05161A1 - 1-n-phenylamino-1h-imidazole derivatives as aromatase inhibitors - Google Patents

1-n-phenylamino-1h-imidazole derivatives as aromatase inhibitors

Info

Publication number
TNSN05161A1
TNSN05161A1 TNP2005000161A TNSN05161A TNSN05161A1 TN SN05161 A1 TNSN05161 A1 TN SN05161A1 TN P2005000161 A TNP2005000161 A TN P2005000161A TN SN05161 A TNSN05161 A TN SN05161A TN SN05161 A1 TNSN05161 A1 TN SN05161A1
Authority
TN
Tunisia
Prior art keywords
phenylamino
imidazole derivatives
aromatase inhibitors
derivatives
relates
Prior art date
Application number
TNP2005000161A
Inventor
Nathalie Adje
Paule Bonnet
Denis Carniato
Jean Lafay
Rémi Delansorne
Jean-Claude Pascal
Original Assignee
Laboratoire Theramex
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP02293107A external-priority patent/EP1431292A1/en
Application filed by Laboratoire Theramex filed Critical Laboratoire Theramex
Publication of TNSN05161A1 publication Critical patent/TNSN05161A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The present invention relates to imidazole derivatives of the formula (I) in which R1, R2,R3, R4, R5, R6 and n are as defined in the specification. The invention also relates to pharmaceutical compositions containing these derivatives, and to the uses thereof.
TNP2005000161A 2002-12-16 2005-06-15 1-n-phenylamino-1h-imidazole derivatives as aromatase inhibitors TNSN05161A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP02293107A EP1431292A1 (en) 2002-12-16 2002-12-16 1-N-phenylamino-1H-imidazole derivatives as aromatase inhibitors
PCT/EP2003/015027 WO2004054983A2 (en) 2002-12-16 2003-12-15 1-n-phenylamino-1h-imidazole derivatives as aromatase inhibitors

Publications (1)

Publication Number Publication Date
TNSN05161A1 true TNSN05161A1 (en) 2007-05-14

Family

ID=42333598

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2005000161A TNSN05161A1 (en) 2002-12-16 2005-06-15 1-n-phenylamino-1h-imidazole derivatives as aromatase inhibitors

Country Status (5)

Country Link
AR (1) AR042478A1 (en)
IL (1) IL169094A0 (en)
OA (1) OA12973A (en)
TN (1) TNSN05161A1 (en)
TW (1) TWI311556B (en)

Also Published As

Publication number Publication date
TW200500345A (en) 2005-01-01
OA12973A (en) 2006-10-13
AR042478A1 (en) 2005-06-22
IL169094A0 (en) 2007-07-04
TWI311556B (en) 2009-07-01

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