TN2011000262A1 - Hemifumarate salt of 1-[4-(cyclohexyl-3-trifluoromethyl-benzyloxymino)-ethyl]-2-ethyl-benzyl]-a zetidine-3-carboxylic acid
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Hemifumarate salt of 1-[4-(cyclohexyl-3-trifluoromethyl-benzyloxymino)-ethyl]-2-ethyl-benzyl]-a zetidine-3-carboxylic acid
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Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
This invention relates to a hemifumarate salt of 1-(4-{1-[(E)-4-cyclohexyl-3-trifluoromethyl-benzyloxyimino]-ethyl}-2-ethyl-benzyl)-azetidine-3-carboxylic acid (Compound I), to pharmaceutical compositions comprising this salt, to processes for forming this salt and to its use in medical treatment. In addition, the present invention also relates to new polymorphic forms of the hemifumarate salt form of Compound I, as well as to pharmaceutical compositions comprising these polymorphic forms, to processes for obtaining them, and their use in medical treatment.
TN2011000262A2011-05-232011-05-23Hemifumarate salt of 1-[4-(cyclohexyl-3-trifluoromethyl-benzyloxymino)-ethyl]-2-ethyl-benzyl]-a zetidine-3-carboxylic acid
TN2011000262A1
(en)
METHOD OF PREPARATION OF CRYSTAL FORMS OF 4-(CYCLOPROPYLMETHOXY)- N-(3,5-DICHLORO-1-OXIDOPYRIDYN-4-yl)-5-METHOXYPYRIDINE-2-CARBOXA MIDE AND CRISTAL FORMS THEREOF.