TN2010000388A1 -
BICYCLIC HETEROCYCLIC DERIVATIVES SPIRO-BICYCLIC PYRAZOLO [1,5-a] PYRIMIDINES HETEROCYCLIC BRIDGES OR DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND USES THEREOF
- Google Patents
BICYCLIC HETEROCYCLIC DERIVATIVES SPIRO-BICYCLIC PYRAZOLO [1,5-a] PYRIMIDINES HETEROCYCLIC BRIDGES OR DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND USES THEREOF
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Priority claimed from PCT/US2009/035422external-prioritypatent/WO2009108838A1/en
Application filed by Wyeth LlcfiledCriticalWyeth Llc
Publication of TN2010000388A1publicationCriticalpatent/TN2010000388A1/en
Il est décrit des composés de formule A Et leurs sels pharmaceutiquement acceptables, qui inhibent sélectivement l'activité des kinases Raf et sont utiles pour le traitement de troubles à médiation par les kinases Raf.Compounds of formula A and their pharmaceutically acceptable salts are described which selectively inhibit the activity of Raf kinases and are useful for the treatment of Raf kinase-mediated disorders.
TNP2010000388A2009-02-272010-08-20
BICYCLIC HETEROCYCLIC DERIVATIVES SPIRO-BICYCLIC PYRAZOLO [1,5-a] PYRIMIDINES HETEROCYCLIC BRIDGES OR DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND USES THEREOF
TN2010000388A1
(en)
BICYCLIC HETEROCYCLIC DERIVATIVES SPIRO-BICYCLIC PYRAZOLO [1,5-a] PYRIMIDINES HETEROCYCLIC BRIDGES OR DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND USES THEREOF
Bicyclic bridged heterocyclic derivatives or spiro-bicyclic heterocyclic derivatives of pyrazolo [1,5-a] pyrimidines, processes for their preparation and their uses
N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2, 3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS.