TH85798B - Acetylene derivatives - Google Patents
Acetylene derivativesInfo
- Publication number
- TH85798B TH85798B TH601001759A TH0601001759A TH85798B TH 85798 B TH85798 B TH 85798B TH 601001759 A TH601001759 A TH 601001759A TH 0601001759 A TH0601001759 A TH 0601001759A TH 85798 B TH85798 B TH 85798B
- Authority
- TH
- Thailand
- Prior art keywords
- substitute
- group
- aryl
- unresponsive
- intercepted
- Prior art date
Links
- 150000000475 acetylene derivatives Chemical class 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 claims abstract 2
- 125000003118 aryl group Chemical group 0.000 claims abstract 2
- 150000001875 compounds Chemical class 0.000 claims abstract 2
- 229910052736 halogen Inorganic materials 0.000 claims abstract 2
- 150000002367 halogens Chemical class 0.000 claims abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 claims abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 claims abstract 2
- 239000001257 hydrogen Substances 0.000 claims abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims abstract 2
- 125000004430 oxygen atom Chemical group O* 0.000 claims abstract 2
- 239000000126 substance Substances 0.000 claims abstract 2
- 125000003107 substituted aryl group Chemical group 0.000 claims abstract 2
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 claims 1
- 239000002253 acid Substances 0.000 abstract 1
- 125000005708 carbonyloxy group Chemical group [*:2]OC([*:1])=O 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 150000003839 salts Chemical group 0.000 abstract 1
Abstract
การประดิษฐ์ในที่นี้จัดหาสารประกอบสูตร (I) (สูตรเคมี) (I) ในที่ซึ่ง R1 แทนไฮโดรเจนหรืออาริล; R2 แทนเฮ็ตเทโรไซเคิลที่ไม่ถูกแทนแทนหรือที่ถูกแทนที่ หรือ R2 แทนอาริลที่ไม่ถูกแทนแทนหรือที่ถูกแทนที่ R3 แทนอัลคิลหรือฮาโลเจน; X แทนพันธะเดี่ยวหรือกลุ่มอัลแคนไดอิล ถูกขัดขวางโดยให้เลือกได้โดยอะตอมอ็อกซิเจนหนึ่ง อะตอมหรือมากกว่า หรือกลุ่มหนึ่งคาร์บอกนิลหนึ่งกลุ่มหรือมากกว่า หรือกลุ่มคาร์บอนิลออกซีหนึ่ง กลุ่มหรือมากกว่า ในรูปแบบของด่างอิสระหรือรูปแบบของเกลือเพิ่มเติมของกรด กระบวนการสำหรับ การเตรียมของพวกมัน และการใช้ของพวกมันเป็นเภสัชภัณฑ์ The invention here provides a compound formula (I) (chemical formula) (I) where R1 represents hydrogen or aryl; R2 is a substitute for a non-substitute or a substitute heterocycle, or a substitute for an unresponsive or substituted aryl, R3 in place of an alkyl or a halogen; X represents a single bond or alkandyl group. Intercepted selectable by an oxygen atom Atom or more Or a group of one or more carboxyels Or one carbonyl oxy group Group or more In free alkaline form or additional salt form of acid. Process for Their preparation And their use as pharmaceuticals
Claims (1)
Publications (2)
| Publication Number | Publication Date |
|---|---|
| TH85798B true TH85798B (en) | 2007-08-10 |
| TH85798A TH85798A (en) | 2007-08-10 |
Family
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