TH77612A - The process was optimized for the N - ([1, 2, 4] triazolopirimidin-2-il) preparations, arylsulfonamides. - Google Patents
The process was optimized for the N - ([1, 2, 4] triazolopirimidin-2-il) preparations, arylsulfonamides.Info
- Publication number
- TH77612A TH77612A TH501001361A TH0501001361A TH77612A TH 77612 A TH77612 A TH 77612A TH 501001361 A TH501001361 A TH 501001361A TH 0501001361 A TH0501001361 A TH 0501001361A TH 77612 A TH77612 A TH 77612A
- Authority
- TH
- Thailand
- Prior art keywords
- triazolopirimidin
- modified
- arylsulfilamine
- lutidine
- picoline
- Prior art date
Links
- 125000004421 aryl sulphonamide group Chemical group 0.000 title claims abstract 6
- 238000000034 method Methods 0.000 title claims 2
- 238000002360 preparation method Methods 0.000 title claims 2
- HWWYDZCSSYKIAD-UHFFFAOYSA-N 3,5-dimethylpyridine Chemical compound CC1=CN=CC(C)=C1 HWWYDZCSSYKIAD-UHFFFAOYSA-N 0.000 claims abstract 4
- ITQTTZVARXURQS-UHFFFAOYSA-N 3-Methylpyridine Chemical compound CC1=CC=CN=C1 ITQTTZVARXURQS-UHFFFAOYSA-N 0.000 claims abstract 4
- YBBRCQOCSYXUOC-UHFFFAOYSA-N Sulfuryl chloride Chemical compound ClS(Cl)(=O)=O YBBRCQOCSYXUOC-UHFFFAOYSA-N 0.000 claims abstract 4
- 150000001412 amines Chemical class 0.000 claims abstract 4
- 125000003118 aryl group Chemical group 0.000 claims abstract 4
- 239000003054 catalyst Substances 0.000 claims abstract 4
- 239000003814 drug Substances 0.000 claims abstract 2
- 229940079593 drugs Drugs 0.000 claims abstract 2
- 239000000126 substance Substances 0.000 claims 1
Abstract
DC60 การประดิษฐ์นี้เกี่ยวข้องกับ N-แอริลซัลฟิลิมีน-เป็นตัวเร่งปฏิกิริยาอะโรเมติกซัลโฟนิล คลอไรด์ด้วย N-([1, 2, 4]- ไตรอะโซโลพิริมิดิน-2-อิล) แอมีน เพื่อก่อตัว N-([1,2,4] ไตรอะโซโล พิริมิดิน-2-อิล) แอริลซัลโฟนาไมด์ถูกปรับปรุงโดยการเลือก 3-พิโคไลน์หรือ 3, 5-ลูทิดีน เป็นเบส การประดิษฐ์นี้เกี่ยวข้องกับ N-แอริลซัลฟิลิมีน-เป็นตัวเร่งปฏิกิริยาอะโรแมติกซัลโฟนิล คลอไรด์ด้วย N-([1,2,4]- ไตรอะโซโลพิริมิดิน-2-อิล) แอมีน เพื่อก่อตัว N-([1,2,4] ไตรอะโซโล พิริมิดิน-2-อิล) แอริลซัลโฟนาไมด์ถูกปรับปรุงโดยการเลือก 3-พิโคไลน์หรือ 3, 5-ลูทิดีน เป็นเบส สิทธิบัตรยา DC60.This invention relates to N-arylsulfilamine - is an aromatic sulfonyl chloride catalyst with N - ([1, 2, 4) - triazolopirimidin-2-. Il) amines to form N - ([1,2,4] triazolopirimidin-2-il) aryl sulfonamides were modified by selection. 3-picoline or 3, 5- lutidine is the base. This invention involves N-arylsulfilamine - is an aromatic sulfonyl chloride catalyst with N - ([1,2,4] - triazolopirimidin-2-. Il) amines to form N - ([1,2,4] triazolopirimidin-2-il) aryl sulfonamides were modified by selection. 3-picoline or 3, 5- lutidine is the base drug patent.
Claims (1)
Publications (2)
| Publication Number | Publication Date |
|---|---|
| TH77612B TH77612B (en) | 2006-05-25 |
| TH77612A true TH77612A (en) | 2006-05-25 |
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