TH64286A - New pyrolidinium derivatives - Google Patents
New pyrolidinium derivativesInfo
- Publication number
- TH64286A TH64286A TH301001396A TH0301001396A TH64286A TH 64286 A TH64286 A TH 64286A TH 301001396 A TH301001396 A TH 301001396A TH 0301001396 A TH0301001396 A TH 0301001396A TH 64286 A TH64286 A TH 64286A
- Authority
- TH
- Thailand
- Prior art keywords
- derivatives
- pyrolidinium
- new
- formula
- muscarin
- Prior art date
Links
- 239000000126 substance Substances 0.000 claims abstract 5
- -1 naphthalinyl Chemical group 0.000 claims 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 2
- 235000010290 biphenyl Nutrition 0.000 claims 1
- 150000004074 biphenyls Chemical class 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 239000003814 drug Substances 0.000 claims 1
- 229940079593 drug Drugs 0.000 claims 1
- 229910052736 halogen Inorganic materials 0.000 claims 1
- 150000002367 halogens Chemical class 0.000 claims 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 1
- 229910052760 oxygen Inorganic materials 0.000 claims 1
- 229910052717 sulfur Inorganic materials 0.000 claims 1
- UQOFGTXDASPNLL-XHNCKOQMSA-N Muscarine Chemical compound C[C@@H]1O[C@H](C[N+](C)(C)C)C[C@H]1O UQOFGTXDASPNLL-XHNCKOQMSA-N 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 239000005557 antagonist Substances 0.000 abstract 1
- 239000005426 pharmaceutical component Substances 0.000 abstract 1
- 239000002464 receptor antagonist Substances 0.000 abstract 1
- 229940044551 receptor antagonist Drugs 0.000 abstract 1
Abstract
DC60 (21/10/46) อนุพันธ์พันธ์ไพร์โรลิดิเนียมชนิดใหม่ ซึ่งมีโครงสร้างทางเคมีที่มีสูตร (I) (สูตรเคมี) (I) เปิดเผยไว้ในการประดิษฐ์นี้เช่นเดียวกับกรรมวิธีสำหรับการ เตรียมของอนุพันธ์ดังกล่าวเหล่านี้, องค์ประกอบทางเภสัชกรรม ซึ่งประกอบรวมด้วยอนุพันธ์ดังกล่าวเหล่านี้และการใช้องค์ประกอบ ดังกล่าวเหล่านี้เป็นตัวต้านฤทธิ์ของตัวรับซึ่งเกี่ยว กับมัสคาริน M3 อนุพันธ์พันธ์ไพร์โรลิดิเนียมชนิดใหม่ ซึ่งมีโครงสร้างทางเคมีที่มีสูตร (I) (สูตรเคมี) (I) เปิดเผยไว้ในการประดิษฐ์นี้เช่นเดียวกับกรรมวิธีสำหรับการ เตรียมของอนุพันธ์ดังกล่าวเหล่านี้, สาร ผสมทางเภสัชกรรม ซึ่งประกอบรวมด้วยอนุพันธ์ดังกล่าวเหล่านี้และการใช้สารผสม ดังกล่าวเหล่านี้ เป็นตัวต้านฤทธิ์ของตัวรับซึ่งเกี่ยว กับมัสคาริน M3 สิทธิบัตรยา DC60 (21/10/46), a new type of pyrolidinium derivative There is a chemical structure with the formula (I) (chemical formula) (I) disclosed in this invention, as well as a process for the Preparation of these derivatives, pharmaceutical components Which includes these derivatives and their use These are receptor antagonists related to muscarin M3, a new pyrolidinium derivative. There is a chemical structure with the formula (I) (chemical formula) (I) disclosed in this invention, as well as a process for the Preparation of these derivatives, pharmaceutical mixtures This includes these derivatives and their use of mixtures. Such these It is an antagonist of the receptor M3 muscarin.
Claims (1)
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TH64286A true TH64286A (en) | 2004-09-24 |
Family
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