TH166320A - Pyrazine derivatives - Google Patents
Pyrazine derivativesInfo
- Publication number
- TH166320A TH166320A TH1601006810A TH1601006810A TH166320A TH 166320 A TH166320 A TH 166320A TH 1601006810 A TH1601006810 A TH 1601006810A TH 1601006810 A TH1601006810 A TH 1601006810A TH 166320 A TH166320 A TH 166320A
- Authority
- TH
- Thailand
- Prior art keywords
- substance
- group
- represented
- acceptable salt
- following formula
- Prior art date
Links
- 150000003216 pyrazines Chemical class 0.000 title claims abstract 4
- 239000000126 substance Substances 0.000 claims abstract 7
- 150000003839 salts Chemical class 0.000 claims abstract 3
- 206010003210 Arteriosclerosis Diseases 0.000 claims abstract 2
- 201000005569 Gout Diseases 0.000 claims abstract 2
- 101000821903 Homo sapiens Solute carrier family 22 member 12 Proteins 0.000 claims abstract 2
- 206010020772 Hypertension Diseases 0.000 claims abstract 2
- 201000001431 Hyperuricemia Diseases 0.000 claims abstract 2
- 102100021495 Solute carrier family 22 member 12 Human genes 0.000 claims abstract 2
- 208000011775 arteriosclerosis disease Diseases 0.000 claims abstract 2
- 206010012601 diabetes mellitus Diseases 0.000 claims abstract 2
- 239000003814 drug Substances 0.000 claims abstract 2
- 229940079593 drug Drugs 0.000 claims abstract 2
- 201000006334 interstitial nephritis Diseases 0.000 claims abstract 2
- 208000017169 kidney disease Diseases 0.000 claims abstract 2
- 238000011321 prophylaxis Methods 0.000 claims abstract 2
- 208000011580 syndromic disease Diseases 0.000 claims abstract 2
- 238000011282 treatment Methods 0.000 claims abstract 2
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 claims 1
- 125000005843 halogen group Chemical group 0.000 claims 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 1
- 229910052757 nitrogen Inorganic materials 0.000 claims 1
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 1
- 239000012453 solvate Substances 0.000 claims 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 claims 1
Abstract
สิ่งที่จัดไว้คือสารอนุพันธ์ไพราซีนชนิดใหม่ซึ่งถูกแทนโดยสูตรต่อไปนี้ (I) หรือ เกลือที่ สามารถยอมรับได้ทางเภสัชกรรมของสารนั้น,หรือโชลเวตของสารนั้น ซึ่งเป็นประโยชน์ส๎าหรับการ บำบัดหรือการป้องกันโรคซึ่ง URAT1 เกี่ยวข้องด้วย ที่รวมถึง โรคเกาต์, ภาวะกรดยูริกในเลือดสูง, ภาวะความดันสูง, โรคไต เช่น โรคไตอักเสบแบบอินเตอร์สติเชียล และที่คล้ายกันนั้น, เบาหวาน, โรคท่อเลือดแดงแข็ง, กลุ่มอาการเลช-นีฮาน, และที่คล้ายกันนั้น สิทธิบัตรยา What is classified is a new pyrazine derivative, represented by the following formula (I) or the pharmacologically acceptable salt of that substance, or the cholvate of that substance. Which is useful for Treatment or prophylaxis in which URAT1 is associated with gout, hyperuricemia, hypertension, kidney disease such as interstitial nephritis. And like that, diabetes, arteriosclerosis, Lech-Nihan syndrome, and the like, drug patents.
Claims (1)
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TH166320A true TH166320A (en) | 2017-08-17 |
Family
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