TH124651A - A new type of N- (arylsulfonyl) beta-amino acid derivative consisting of an aminomethyl group. Which was replaced, the process of preparing such substances And pharmaceutical components containing such substances - Google Patents
A new type of N- (arylsulfonyl) beta-amino acid derivative consisting of an aminomethyl group. Which was replaced, the process of preparing such substances And pharmaceutical components containing such substancesInfo
- Publication number
- TH124651A TH124651A TH201001052A TH0201001052A TH124651A TH 124651 A TH124651 A TH 124651A TH 201001052 A TH201001052 A TH 201001052A TH 0201001052 A TH0201001052 A TH 0201001052A TH 124651 A TH124651 A TH 124651A
- Authority
- TH
- Thailand
- Prior art keywords
- substances
- replaced
- receptors
- arylsulfonyl
- beta
- Prior art date
Links
- 239000000126 substance Substances 0.000 title claims abstract 5
- 125000004202 aminomethyl group Chemical group [H]N([H])C([H])([H])* 0.000 title 1
- 125000004391 aryl sulfonyl group Chemical group 0.000 title 1
- 150000001576 beta-amino acids Chemical class 0.000 title 1
- 239000005426 pharmaceutical component Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 claims abstract 6
- 229940079593 drug Drugs 0.000 claims abstract 2
- 239000003814 drug Substances 0.000 claims abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 claims 1
- 125000001624 naphthyl group Chemical group 0.000 claims 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 1
- -1 phenyl vinyl group Chemical group 0.000 claims 1
- 125000001712 tetrahydronaphthyl group Chemical group C1(CCCC2=CC=CC=C12)* 0.000 claims 1
- 208000017667 Chronic Disease Diseases 0.000 abstract 2
- 208000037976 chronic inflammation Diseases 0.000 abstract 2
- 230000001684 chronic effect Effects 0.000 abstract 1
- 230000006020 chronic inflammation Effects 0.000 abstract 1
- 208000037893 chronic inflammatory disorder Diseases 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 230000002757 inflammatory effect Effects 0.000 abstract 1
- 230000005923 long-lasting effect Effects 0.000 abstract 1
- 229940126601 medicinal product Drugs 0.000 abstract 1
- 230000001575 pathological effect Effects 0.000 abstract 1
- 230000007170 pathology Effects 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- 229940127557 pharmaceutical product Drugs 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Abstract
DC60 (19/05/53) สารประกอบตามสูตร (สูตรเคมี) (I) สารประกอบเหล่านี้แสดงสัมพรรคภาพสำหรับตัวรับแบรดีไคนินโดยเลือกออกฤทธิ์ที่ตัวรับ B1 มากกว่า สารเหล่านี้อาจนำไปใช้เพื่อเตรียมผลิตภัณฑ์ยาซึ่งมุ่งหมายสำหรับรักษาหรือป้องกัน พยาธิสภาพที่มีการอักเสบหรือโรคที่มีการอักเสบยาวนานหรือเรื้อรัง สารประกอบตามสูตร: (สูตรเคมี) (I) สารประกอบเหล่านี้แสดงสัมพรรคภาพสำหรับตัวรับแบรดีไคนินโดยเลือกออกฤทธิ์ที่ตัวรับ B1 มากกว่า สารเหล่านี้อาจนำไปใช้เพื่อเตรียมผลิตภัณฑ์ยาซึ่งมุ่งหมายสำหรับรักษาหรือป้องกัน พยาธิสภาพที่มีการอักเสบหรือโรคที่มีการอักเสบยาวนานหรือเรื้อรัง: สิทธิบัตรยา DC60 (19/05/53) Compounds according to the formula (Chemical formula) (I) These compounds exhibit affinity for bradyinine receptors, more selective on B1 receptors. These compounds may be used to Prepare a medicinal product intended for treatment or prevention. Pathological conditions with long-lasting or chronic inflammation or disease Formulated Compounds: (Chemical Formula) (I) These compounds exhibit affinity for bradyinine receptors, selecting greater activity on B1 receptors.These may be used to prepare pharmaceutical products intended for therapeutic purposes. Or protect Inflammatory pathology or chronic or chronic inflammatory disease: Drug patent.
Claims (1)
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TH124651A true TH124651A (en) | 2013-06-21 |
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