TH106989A - Triazolo derivatives [4,3-a] a new type of pyridine, the process for its preparation. The use of the substance as a drug, pharmaceutical component And new use Specific As an inhibitor - Google Patents
Triazolo derivatives [4,3-a] a new type of pyridine, the process for its preparation. The use of the substance as a drug, pharmaceutical component And new use Specific As an inhibitorInfo
- Publication number
- TH106989A TH106989A TH901003233A TH0901003233A TH106989A TH 106989 A TH106989 A TH 106989A TH 901003233 A TH901003233 A TH 901003233A TH 0901003233 A TH0901003233 A TH 0901003233A TH 106989 A TH106989 A TH 106989A
- Authority
- TH
- Thailand
- Prior art keywords
- new
- drug
- formula
- pyridine
- inhibitor
- Prior art date
Links
Abstract
DC60 (09/10/52) การประดิษฐ์เกี่ยวกับผลิตภัณฑ์ของสูตร (I) ชนิดใหม่ (สูตร) (I) ซึ่ง: Ra แสดงแทน H, Hal หรือแอริล หรือเฮเทอโรแอริล, ซึ่งถูกเลือกแทนที่; Rb แสดงแทน H, Rc, -COORc, -CO-Rc หรือ -CO-NRcRd; ซึ่ง Rc แสดงแทนแอลคิล, ไซโคลแอลคิล, เฮเทอโรไซโคลแอลคิล, แอริล และเฮเทอโรแอริล, ทั้งหมด ที่เลือกแทนที่; Rd แสดงแทน H, alk หรือ ไซโคลแอลคิล; ผลิตภัณฑ์เหล่านี้อยู่ในไอโซเมอร์ทั้งหมด และเกลือ, ในรูปยา, ที่เฉพาะเจาะจง เป็นสารยับยั้ง MET. การประดิษฐ์เกี่ยวกับผลิตภัณฑ์ของสูตร (I) ชนิดใหม่ (สูตร) (I) ซึ่ง: Ra แสดงแทน H, Hal หรือแอริล หรือเฮเทอโรแอริล, ซึ่งถูกเลือกแทนที่; Rb แสดงแทน H, Rc, -COORc, -CO-Rc หรือ -CO-NRcRd; ซึ่ง Rc แสดงแทนแอลคิล, ไซโคลแอลคิล, เฮเทอโรไซโคลแอลคิล, แอริล และเฮเทอโรแอริล, ทั้งหมด ที่เลือกแทนที่; Rd แสดงแทน H, alk หรือ ไซดคลแอลคิล; ผลิตภัณฑ์เหล่านี้อยู่ในไอโซเมอร์ทั้งหมด และเกลือ, ในรูปยา, ที่เฉพาะเจาะจง เป็นสารยับยั้ง MET.DC60 (09/10/09) Invention concerning a new product of formula (I) (formula) (I) in which: Ra represents H, Hal or aryl or heteroaryl, selectively substituted; Rb represents H, Rc, -COORc, -CO-Rc or -CO-NRcRd; in which Rc represents alkyl, cycloalkyl, heterocycloalkyl, aryl and heteroaryl, all selectively substituted; Rd represents H, alk or cycloalkyl; these products are all isomers and salts, in pharmaceutical form, specifically MET inhibitors. Invention concerning a new product of formula (I) (formula) (I) in which: Ra represents H, Hal or aryl or heteroaryl, selectively substituted; Rb represents H, Rc, -COORc, -CO-Rc or -CO-NRcRd; Where Rc represents alkyl, cycloalkyl, heterocycloalkyl, aryl, and heteroaryl, all selectively substituted; Rd represents H, alk, or cyclic alkyl; these products are all isomers, and salts, in pharmaceutical form, are specific MET inhibitors.
Claims (1)
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TH106989A true TH106989A (en) | 2011-03-30 |
Family
ID=
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EA201170223A1 (en) | NEW IMIDAZO DERIVATIVES [1,2-a] PYRIDINE, METHOD FOR THEIR PRODUCTION, THEIR APPLICATION AS A MEDICINE, PHARMACEUTICAL COMPOSITIONS AND A NEW APPLICATION, PARTICULAR AS INHIBITORS | |
| WO2010007316A3 (en) | Novel triazolo(4,3-a)pyridine derivatives, process for the preparation thereof, use thereof as medicaments, pharmaceutical compositions and novel use, in particular as met inhibitors | |
| EA201201663A1 (en) | DERIVATIVES 2- (ARYLAMINO) -3H-IMIDAZO [4,5-B] Pyridine-6-carboxamide and their use as MPGES-1 inhibitors | |
| CR20110031A (en) | NEW IMIDAZO DERIVATIVES [1,2-a] PYRIMIDINE, ITS PREPARATION PROCEDURE, ITS APPLICATION AS MEDICINES, PHARMACEUTICAL COMPOSITIONS AND NEW USE IN PARTICULARLY AS MET INHIBITORS | |
| EA201290260A1 (en) | BENZIMIDAZOL-IMIDAZOL DERIVATIVES | |
| EA201001683A1 (en) | Derivatives of phenyl or pyridinyl substituted indazols | |
| PH12015501585A1 (en) | Manufacturing process for pyrimidine derivatives | |
| EA201491376A1 (en) | DERIVATIVES 1H-PYRROLO [2,3-B] Pyridine and THEIR APPLICATION AS KINASE INHIBITORS | |
| MX2012004311A (en) | Spiro-condensed cyclohexane derivatives as hsl inhibitors useful for the treatment of diabetes. | |
| EA201270302A1 (en) | ANHARROUND FORMS OF PYRIDINE DERIVATIVES | |
| CO6480974A2 (en) | NEW DERIVATIVES OF (6-OXO-1,6-DIHIDRO-PIRIMIDIN-2-IL) -AMIDA, ITS PREPARATION AND ITS PHARMACEUTICAL USE AS AKT PHOSPHORILATION INHIBITORS (PKB) | |
| CU20100157A7 (en) | NEW DIHYDROINDOLONE DERIVATIVES, THEIR PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
| PL401473A1 (en) | New, highly fluorescent heterocyclic substances and their preparation | |
| HK1210162A1 (en) | Pyrimidinone derivatives as antimalarial agents | |
| MX2016001095A (en) | Salts of dasatinib in crystalline form. | |
| EA201170300A1 (en) | CRYSTAL FORMS OF PYRIDINE DERIVATIVE | |
| NO20076161L (en) | Methods for preparing 4-biphenylazetidin-2-ones | |
| UA111334C2 (en) | Delta crystalline form of the arginine salt of perindopril, a process for its preparation, and pharmaceutical compositions containing it | |
| TH106989A (en) | Triazolo derivatives [4,3-a] a new type of pyridine, the process for its preparation. The use of the substance as a drug, pharmaceutical component And new use Specific As an inhibitor | |
| WO2013024358A3 (en) | Substituted heterocyclic amine compounds as cholestryl ester-transfer protein (cetp) inhibitors | |
| TH106990A (en) | Imidazo derivative [1,2-a], a new type of piridine. Process for the preparation of the substance, the use of the substance in the form of drugs, pharmaceutical constituents And new, specific uses as a MET inhibitor. | |
| EA201170183A1 (en) | SUBSTITUTED DERIVATIVES 1-BENZYLCINNOLIN-4- (1H) -OH, THEIR RECEIVING AND THEIR USE IN THERAPY | |
| UY33927A (en) | NEW DIHIDRO-OXAZOLOBENZODIAZEPINONAS DERIVATIVES, THEIR PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
| CU20130037A7 (en) | NEW DIHYDROBENZOXATIAZEPIN DERIVATIVES, THEIR PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
| TW201612188A (en) | The L-proline complex, monohydrate and crystal of a sodium-glucose contransporter 2 inhibitor |