TH105532A - Carbamoyl benzoethiazole derivatives are lipase inhibitors. And phospholipase - Google Patents
Carbamoyl benzoethiazole derivatives are lipase inhibitors. And phospholipaseInfo
- Publication number
- TH105532A TH105532A TH601005100A TH0601005100A TH105532A TH 105532 A TH105532 A TH 105532A TH 601005100 A TH601005100 A TH 601005100A TH 0601005100 A TH0601005100 A TH 0601005100A TH 105532 A TH105532 A TH 105532A
- Authority
- TH
- Thailand
- Prior art keywords
- benzoethiazole
- phospholipase
- carbamoyl
- derivatives
- lipase inhibitors
- Prior art date
Links
- 229940040461 Lipase Drugs 0.000 title 1
- 239000004367 Lipase Substances 0.000 title 1
- 102000015439 Phospholipases Human genes 0.000 title 1
- 108010064785 Phospholipases Proteins 0.000 title 1
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 230000002401 inhibitory effect Effects 0.000 title 1
- 102000004882 lipase Human genes 0.000 title 1
- 108090001060 lipase Proteins 0.000 title 1
- 235000019421 lipase Nutrition 0.000 title 1
- 239000000126 substance Substances 0.000 claims abstract 6
- 239000003814 drug Substances 0.000 claims abstract 4
- 229940079593 drugs Drugs 0.000 claims abstract 3
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 claims 2
- LUMNWCHHXDUKFI-UHFFFAOYSA-N 5-bicyclo[2.2.1]hept-2-enylmethanol Chemical compound C1C2C(CO)CC1C=C2 LUMNWCHHXDUKFI-UHFFFAOYSA-N 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 229910052736 halogen Inorganic materials 0.000 claims 1
- 150000002367 halogens Chemical class 0.000 claims 1
- 125000005842 heteroatoms Chemical group 0.000 claims 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims 1
- IOJUPLGTWVMSFF-UHFFFAOYSA-N Benzothiazole Chemical class C1=CC=C2SC=NC2=C1 IOJUPLGTWVMSFF-UHFFFAOYSA-N 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000011780 sodium chloride Substances 0.000 abstract 2
Abstract
DC60 (15/01/50) การประดิษฐ์นี้เกี่ยวข้องกับอนุพันธ์เบนโซไทรอะโซลที่มีสูตร I ซึ่งจะมีความหมายตามที่ได้ ระบุไว้ในรายละเอียดการประดิษฐ์, เกลือของสารนั้นที่สามารถใช้ได้ทางเภสัชกรรม และการใช้สาร นั้นเป็นสารทางยา (I) (สูตรเคมี) การประดิษฐ์นี้เกี่ยวข้องกับอนุพันธ์เบนโซไทรอะโซลที่มีสูตร I ซึ่งจะมีความหมายตามที่ได้ ระบุไว้ในรายละเอียดการประดิษฐ์, เกลือของสารนั้นที่สามารถใช้ได้ทางเภสัชกรรม และการใช้สาร นั้นเป็นสารทางยา (I) (สูตรเคมี) สิทธิบัตรยา DC60 (15/01/50) This invention relates to a benzothiazole derivative with the formula I, which takes the meaning according to the resulting Specified in the invention description, the salts of that substance are available for pharmaceutical use and their use as a medicinal substance (I) (chemical formula) .This invention involves a benzothiazole derivative with formula I, which will have Meaning as expected Specified in the invention details, the salt of that substance is usable in pharmaceuticals and its use as a drug (I) (chemical formula), drug patent.
Claims (1)
Publications (2)
Publication Number | Publication Date |
---|---|
TH105532B TH105532B (en) | 2010-12-30 |
TH105532A true TH105532A (en) | 2010-12-30 |
Family
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