SV2004001577A -
HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS
- Google Patents
HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS
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Publication number
SV2004001577A
SV2004001577ASV2003001577ASV2003001577ASV2004001577ASV 2004001577 ASV2004001577 ASV 2004001577ASV 2003001577 ASV2003001577 ASV 2003001577ASV 2003001577 ASV2003001577 ASV 2003001577ASV 2004001577 ASV2004001577 ASV 2004001577A
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Application filed by Agouron PharmafiledCriticalAgouron Pharma
Priority to SV2003001577ApriorityCriticalpatent/SV2004001577A/en
Publication of SV2004001577ApublicationCriticalpatent/SV2004001577A/en
Medicines That Contain Protein Lipid Enzymes And Other Medicines
(AREA)
Abstract
SE REVELAN COMPUESTOS DE LA FORMULA (VER FORMULA), DONDE LAS VARIABLES DE FORMULA SON TALES COMO LAS ANTES DEFINIDAS AQUI, QUE INHIBEN O BLOQUEAN VENTAJOSAMENTE LA ACTIVIDAD BIOLOGICA DE LA PROTEASA DEL VIH. ESTOS COMPUESTOS, ASI COMO LAS COMPOSICIONES FARMACEUTICAS QUE CONTIENEN ESTOS COMPUESTOS, SON UTILES PARA EL TRATAMIENTO DE PACIENTES O HUESPEDES INFECTADOS CON EL VIRUS VIH. TAMBIEN SE DESCRIBEN PRODUCTOS INTERMEDIOS Y METODOS DE SINTESIS PARA LA PREPARACION DE TALES COMPUESTOS.FORMULA COMPOUNDS ARE DISCLOSED (SEE FORMULA), WHERE THE FORMULA VARIABLES ARE SUCH AS THE BEFORE DEFINED HERE, THAT INHIBIT OR BLOCK ADVANTAGES THE BIOLOGICAL ACTIVITY OF HIV PROTEASE. THESE COMPOUNDS, AS WELL AS THE PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, ARE USEFUL FOR THE TREATMENT OF PATIENTS OR GUESTS INFECTED WITH HIV VIRUS. INTERMEDIATE PRODUCTS AND SYNTHESIS METHODS ARE ALSO DESCRIBED FOR THE PREPARATION OF SUCH COMPOUNDS.
SV2003001577A2003-07-092003-07-09
HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS
SV2004001577A
(en)
DERIVATIVES OF ISOINDOLONE, PREPARATION PROCESS AND INTERMEDIATE COMPOUNDS OF THIS PROCESS, ITS USE AS MEDICATIONS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.