SV2004001577A - HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS - Google Patents

HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS

Info

Publication number
SV2004001577A
SV2004001577A SV2003001577A SV2003001577A SV2004001577A SV 2004001577 A SV2004001577 A SV 2004001577A SV 2003001577 A SV2003001577 A SV 2003001577A SV 2003001577 A SV2003001577 A SV 2003001577A SV 2004001577 A SV2004001577 A SV 2004001577A
Authority
SV
El Salvador
Prior art keywords
compounds
hiv protease
synthesis
pharmaceutical
compositions
Prior art date
Application number
SV2003001577A
Other languages
Spanish (es)
Inventor
Stacie S Canon-Koch
Therese N Alexander
Mark Barvian
Gary Bolton
Frederick E Boyer
Benjamin J Burke
Tod Holler
Tanya M Jewell
Josyula Vara Prasad
David J Kucera
Maria A Linton
Jeff Machak
Lennert J Mitchell
Sean T Murphy
Siegfried H Reich
Donald J Skalitzky
John H Tatlock
Michael D Varney
Scott C Virgil
Stephen E Webber
Stephen T Worland
Original Assignee
Agouron Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Agouron Pharma filed Critical Agouron Pharma
Priority to SV2003001577A priority Critical patent/SV2004001577A/en
Publication of SV2004001577A publication Critical patent/SV2004001577A/en

Links

Landscapes

  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

SE REVELAN COMPUESTOS DE LA FORMULA (VER FORMULA), DONDE LAS VARIABLES DE FORMULA SON TALES COMO LAS ANTES DEFINIDAS AQUI, QUE INHIBEN O BLOQUEAN VENTAJOSAMENTE LA ACTIVIDAD BIOLOGICA DE LA PROTEASA DEL VIH. ESTOS COMPUESTOS, ASI COMO LAS COMPOSICIONES FARMACEUTICAS QUE CONTIENEN ESTOS COMPUESTOS, SON UTILES PARA EL TRATAMIENTO DE PACIENTES O HUESPEDES INFECTADOS CON EL VIRUS VIH. TAMBIEN SE DESCRIBEN PRODUCTOS INTERMEDIOS Y METODOS DE SINTESIS PARA LA PREPARACION DE TALES COMPUESTOS.FORMULA COMPOUNDS ARE DISCLOSED (SEE FORMULA), WHERE THE FORMULA VARIABLES ARE SUCH AS THE BEFORE DEFINED HERE, THAT INHIBIT OR BLOCK ADVANTAGES THE BIOLOGICAL ACTIVITY OF HIV PROTEASE. THESE COMPOUNDS, AS WELL AS THE PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, ARE USEFUL FOR THE TREATMENT OF PATIENTS OR GUESTS INFECTED WITH HIV VIRUS. INTERMEDIATE PRODUCTS AND SYNTHESIS METHODS ARE ALSO DESCRIBED FOR THE PREPARATION OF SUCH COMPOUNDS.

SV2003001577A 2003-07-09 2003-07-09 HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS SV2004001577A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
SV2003001577A SV2004001577A (en) 2003-07-09 2003-07-09 HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SV2003001577A SV2004001577A (en) 2003-07-09 2003-07-09 HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS

Publications (1)

Publication Number Publication Date
SV2004001577A true SV2004001577A (en) 2004-03-05

Family

ID=40091721

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2003001577A SV2004001577A (en) 2003-07-09 2003-07-09 HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS

Country Status (1)

Country Link
SV (1) SV2004001577A (en)

Similar Documents

Publication Publication Date Title
PA8547501A1 (en) HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS
CO2022018811A2 (en) Kras g12c protein inhibitors and their uses
PE20181045A1 (en) USEFUL COMPOUNDS AS IMMUNOMODULATORS
CR7716A (en) USE OF IKB-KINASE INHIBITORS FOR PAIN TREATMENT
UY29458A1 (en) REPLACED HETEROCICLES AND USES OF THE SAME
BR112021025928A2 (en) Bempedoic acid preparation methods and compositions thereof
UY27882A1 (en) CHEMICAL COMPOUNDS
SV2004001690A (en) NEW DERIVATIVES OF HETEROCICLIC FLUOROGLYCOSIDS, MEDICINES CONTAINING THESE COMPOUNDS, AND THE USE OF THE SAME
ECSP088099A (en) NEW DERIVATIVES OF 2-AZETIDINONE FOR THE TREATMENT OF HYPERLIPIDEMIC DISEASES
UY28691A1 (en) DERIVATIVES OF DIFENILAZETIDONA
ECSP078051A (en) NEW DERIVATIVES OF 2-AZETIDINONE AS INHIBITORS OF CHOLESTEROL ABSORPTION FOR THE TREATMENT OF HYPERLIPIDEMIC CONDITIONS
DOP2000000108A (en) ANTI-CORPOVIRAL COMPOUNDS AND COMPOSITIONS, THEIR PHARMACEUTICAL USES, AND MATERIALS FOR SYNTHESIS
PA8719401A1 (en) TETRAHYDROPIRIDOTIENOPIRIMIDINA COMPOUNDS AND METHODS FOR USE
UY27851A1 (en) DIFENILAZETIDINONAS REPLACED IN RING, PROCEDURE FOR PREPARATION, MEDICATIONS UNDERSTANDING THESE COMPOUNDS AND THEIR USE.
HN2003000162A (en) DERIVATIVES OF ISOINDOLONE, PREPARATION PROCESS AND INTERMEDIATE COMPOUNDS OF THIS PROCESS, ITS USE AS MEDICATIONS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
AR045159A1 (en) DERIVATIVES OF 1-SULPHONYLINDOLS, ITS PREPARATION AND ITS APPLICATION AS MEDICINES
CL2021001198A1 (en) Heteroaromatic compounds as vanine inhibitors
UY26666A1 (en) ANTIPICORNAVIRAL COMPOUNDS AND COMPOSITIONS, THEIR PHARMACEUTICAL USES AND THE MATERIALS FOR THEIR SYNTHESIS
PE20181450A1 (en) 1,3,4-THADIAZOLE COMPOUNDS AND THEIR USE IN THE TREATMENT OF CANCER
SV2004001577A (en) HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS
DOP2002000415A (en) HIV PROTEASE INHIBITORS, COMPOSOTIONS CONTAINING THE SAME, ITS PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS.
UY27394A1 (en) ORDERS WITH ANTI-ANGIOGÉNA ACTIVITY.
UY27330A1 (en) HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS.
SV2004001553A (en) HIV INHIBITORY PROTEASA, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS
ECSP034892A (en) HIV PROTEASE INHIBITORS, COMPOSITIONS THAT CONTAIN THEM, THEIR PHARMACEUTICAL AND MATERIAL USES FOR SYNTHESIS

Legal Events

Date Code Title Description
FD Lapse