SV2002000776A - NEW SUBSTITUTED IMIDAZOTRIAZINONES REF.LEA 34 985-SV - Google Patents
NEW SUBSTITUTED IMIDAZOTRIAZINONES REF.LEA 34 985-SVInfo
- Publication number
- SV2002000776A SV2002000776A SV2001000776A SV2001000776A SV2002000776A SV 2002000776 A SV2002000776 A SV 2002000776A SV 2001000776 A SV2001000776 A SV 2001000776A SV 2001000776 A SV2001000776 A SV 2001000776A SV 2002000776 A SV2002000776 A SV 2002000776A
- Authority
- SV
- El Salvador
- Prior art keywords
- lea
- ref
- new substituted
- substituted imidazotriazinones
- imidazotriazinones
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A NUEVAS IMIDAZOTRIAZINONAS SUSTITUIDAS, A PROCEDIMIENTOS PARA SU PREPARACION Y A SU USO PARA LA PREPARACION DE MEDICAMENTOS, ESPECIALMENTE PARA LA MEJORA E LA PERCEPCION, LA CAPACIDAD DE CONCENTRACION, LA CAPACIDAD DE APRENDIZAJE Y/O LA CAPACIDAD DE MEMORIA.THE PRESENT INVENTION REFERS TO NEW REPLACED IMIDAZOTRIAZINONES, PROCEDURES FOR THEIR PREPARATION AND THEIR USE FOR THE PREPARATION OF MEDICINES, ESPECIALLY FOR THE IMPROVEMENT AND PERCEPTION, THE CAPACITY OF CONCENTRATION, THE CAPACITY OF LEARNING AND LEARNING / CAPACITY.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10064105A DE10064105A1 (en) | 2000-12-21 | 2000-12-21 | New substituted imidazotriazinones |
Publications (1)
Publication Number | Publication Date |
---|---|
SV2002000776A true SV2002000776A (en) | 2002-12-02 |
Family
ID=7668333
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SV2001000776A SV2002000776A (en) | 2000-12-21 | 2001-12-20 | NEW SUBSTITUTED IMIDAZOTRIAZINONES REF.LEA 34 985-SV |
Country Status (15)
Country | Link |
---|---|
US (1) | US6573263B2 (en) |
EP (1) | EP1347978B1 (en) |
JP (1) | JP2004525098A (en) |
AR (1) | AR034423A1 (en) |
AU (1) | AU2002216087A1 (en) |
CA (1) | CA2431965A1 (en) |
DE (2) | DE10064105A1 (en) |
DO (1) | DOP2001000297A (en) |
ES (1) | ES2248228T3 (en) |
GT (1) | GT200100254A (en) |
HN (1) | HN2001000281A (en) |
PE (1) | PE20020756A1 (en) |
SV (1) | SV2002000776A (en) |
UY (1) | UY27080A1 (en) |
WO (1) | WO2002050078A1 (en) |
Families Citing this family (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7087605B2 (en) | 2001-06-01 | 2006-08-08 | Bayer Aktiengesellschaft | 5-Ethyl-imidazotriazinones |
GB0113342D0 (en) * | 2001-06-01 | 2001-07-25 | Bayer Ag | Novel Heterocycles 1 |
DE60320529T2 (en) * | 2002-02-04 | 2009-06-10 | F. Hoffmann-La Roche Ag | CHINOLINE DERIVATIVES AS NPY ANTAGONISTS |
CA2489251A1 (en) * | 2002-07-05 | 2004-01-15 | F. Hoffmann-La Roche Ag | Quinazoline derivatives |
CA2493712A1 (en) * | 2002-08-07 | 2004-02-19 | F. Hoffmann-La Roche Ag | Aminothiazole derivatives as npy5 receptor inhibitors |
JP2006219374A (en) | 2003-06-13 | 2006-08-24 | Daiichi Asubio Pharma Co Ltd | Imidazotriazinone derivative having pde 7 inhibition |
UA115057C2 (en) | 2012-04-25 | 2017-09-11 | Такеда Фармасьютікал Компані Лімітед | Nitrogenated heterocyclic compound |
EP2873669A4 (en) * | 2012-07-13 | 2015-11-25 | Takeda Pharmaceutical | Heterocyclic compound |
WO2014142255A1 (en) | 2013-03-14 | 2014-09-18 | 武田薬品工業株式会社 | Heterocyclic compound |
JP6411342B2 (en) | 2013-07-03 | 2018-10-24 | 武田薬品工業株式会社 | Amide compounds |
JP6427491B2 (en) | 2013-07-03 | 2018-11-21 | 武田薬品工業株式会社 | Heterocyclic compounds |
EP3087060B1 (en) | 2013-12-23 | 2020-05-13 | Merck Sharp & Dohme Corp. | Pyrimidone carboxamide compounds as pde2 inhibitors |
US9849132B2 (en) | 2014-01-08 | 2017-12-26 | Intra-Cellular Therapies, Inc. | Products and pharmaceutical compositions |
MA50375A (en) | 2014-04-23 | 2021-05-26 | Dart Neuroscience Cayman Ltd | COMPOSITIONS CONTAINING [1,2,4] TRIAZOLO [1,5-A] PYRIMIDINE-7-YL SUBSTITUTE COMPOUNDS USED AS PDE2 INHIBITORS |
TWI568737B (en) | 2014-11-05 | 2017-02-01 | 達特神經科學(開曼)有限責任公司 | Substituted 5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-amine compounds as pde2 inhibitors |
US10105349B2 (en) | 2014-12-06 | 2018-10-23 | Intra-Cellular Therapies, Inc. | Organic compounds |
KR102557603B1 (en) | 2014-12-06 | 2023-07-19 | 인트라-셀룰라 써래피스, 인코퍼레이티드. | Organic compounds |
WO2016145614A1 (en) | 2015-03-17 | 2016-09-22 | Merck Sharp & Dohme Corp. | Triazolyl pyrimidinone compounds as pde2 inhibitors |
EP3285581B1 (en) | 2015-03-26 | 2021-08-11 | Merck Sharp & Dohme Corp. | Pyrazolyl pyrimidinone compounds as pde2 inhibitors |
US10195201B2 (en) | 2015-05-05 | 2019-02-05 | Merck Sharp & Dohme Corp. | Heteroaryl-pyrimidinone compounds as PDE2 inhibitors |
WO2016183741A1 (en) | 2015-05-15 | 2016-11-24 | Merck Sharp & Dohme Corp. | Pyrimidinone amide compounds as pde2 inhibitors |
WO2016191935A1 (en) | 2015-05-29 | 2016-12-08 | Merck Sharp & Dohme Corp. | 6-alkyl dihydropyrazolopyrimidinone compounds as pde2 inhibitors |
WO2016192083A1 (en) | 2015-06-04 | 2016-12-08 | Merck Sharp & Dohme Corp. | Dihydropyrazolopyrimidinone compounds as pde2 inhibitors |
EP3313852B1 (en) | 2015-06-25 | 2021-01-20 | Merck Sharp & Dohme Corp. | Substituted pyrazolo/imidazolo bicyclic compounds as pde2 inhibitors |
WO2017000276A1 (en) | 2015-07-01 | 2017-01-05 | Merck Sharp & Dohme Corp. | Bicyclic heterocyclic compounds as pde2 inhibitors |
WO2017000277A1 (en) | 2015-07-01 | 2017-01-05 | Merck Sharp & Dohme Corp. | Substituted triazolo bicycliccompounds as pde2 inhibitors |
WO2019101970A1 (en) | 2017-11-23 | 2019-05-31 | Oslo University Hospital Hf | Treatment of tachycardia |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK109578A (en) | 1977-03-25 | 1978-09-26 | Allen & Hanburys Ltd | PROCEDURE FOR MAKING HETEROCYCLIC COMPOUNDS |
DE19541264A1 (en) | 1995-11-06 | 1997-05-07 | Bayer Ag | Purin-6-one derivatives |
DE19709877A1 (en) | 1997-03-11 | 1998-09-17 | Bayer Ag | 1,5-dihydro-pyrazolo [3,4-d] pyrimidinone derivatives |
HU230154B1 (en) * | 1997-11-12 | 2015-09-28 | Bayer Intellectual Property Gmbh | Process for the preparation of 2-phenyl substituted imidazotriazinones |
DE19827640A1 (en) | 1998-06-20 | 1999-12-23 | Bayer Ag | New imidazotriazine derivatives useful as smooth muscle relaxants for treating e.g. cardiovascular disorders, cerebrovascular disorders, or erectile dysfunction |
DE19838705A1 (en) | 1998-08-26 | 2000-03-02 | Bayer Ag | New dihydro- (1,2,3) -triazolo- [4,5-d] pyrimidin-7-ones |
-
2000
- 2000-12-21 DE DE10064105A patent/DE10064105A1/en not_active Withdrawn
-
2001
- 2001-11-30 DO DO2001000297A patent/DOP2001000297A/en unknown
- 2001-12-07 AR ARP010105704A patent/AR034423A1/en unknown
- 2001-12-10 EP EP01271375A patent/EP1347978B1/en not_active Expired - Lifetime
- 2001-12-10 ES ES01271375T patent/ES2248228T3/en not_active Expired - Lifetime
- 2001-12-10 CA CA002431965A patent/CA2431965A1/en not_active Abandoned
- 2001-12-10 WO PCT/EP2001/014450 patent/WO2002050078A1/en active IP Right Grant
- 2001-12-10 AU AU2002216087A patent/AU2002216087A1/en not_active Abandoned
- 2001-12-10 JP JP2002551971A patent/JP2004525098A/en active Pending
- 2001-12-10 DE DE50107316T patent/DE50107316D1/en not_active Expired - Fee Related
- 2001-12-18 UY UY27080A patent/UY27080A1/en not_active Application Discontinuation
- 2001-12-19 GT GT200100254A patent/GT200100254A/en unknown
- 2001-12-19 HN HN2001000281A patent/HN2001000281A/en unknown
- 2001-12-20 SV SV2001000776A patent/SV2002000776A/en unknown
- 2001-12-20 PE PE2001001277A patent/PE20020756A1/en not_active Application Discontinuation
- 2001-12-21 US US10/026,310 patent/US6573263B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
CA2431965A1 (en) | 2002-06-27 |
WO2002050078A1 (en) | 2002-06-27 |
PE20020756A1 (en) | 2002-10-02 |
EP1347978B1 (en) | 2005-08-31 |
DOP2001000297A (en) | 2003-08-15 |
JP2004525098A (en) | 2004-08-19 |
AU2002216087A1 (en) | 2002-07-01 |
UY27080A1 (en) | 2002-07-31 |
EP1347978A1 (en) | 2003-10-01 |
AR034423A1 (en) | 2004-02-25 |
HN2001000281A (en) | 2003-02-04 |
US6573263B2 (en) | 2003-06-03 |
GT200100254A (en) | 2002-08-19 |
DE10064105A1 (en) | 2002-06-27 |
US20020198377A1 (en) | 2002-12-26 |
ES2248228T3 (en) | 2006-03-16 |
DE50107316D1 (en) | 2005-10-06 |
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