SV2002000474A - HYGROMYCIN DERIVATIVES TO REF.PC11O32ABCZ / BB - Google Patents

HYGROMYCIN DERIVATIVES TO REF.PC11O32ABCZ / BB

Info

Publication number
SV2002000474A
SV2002000474A SV2001000474A SV2001000474A SV2002000474A SV 2002000474 A SV2002000474 A SV 2002000474A SV 2001000474 A SV2001000474 A SV 2001000474A SV 2001000474 A SV2001000474 A SV 2001000474A SV 2002000474 A SV2002000474 A SV 2002000474A
Authority
SV
El Salvador
Prior art keywords
compounds
formula
infections
ref
refers
Prior art date
Application number
SV2001000474A
Other languages
Spanish (es)
Inventor
Hayward Mathew Merrill
Ii Robert Gerald Linde
Takushi Kaneko
Michael Scott Visser
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of SV2002000474A publication Critical patent/SV2002000474A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/12Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/14Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

ESTA INVENCION SE REFIERE A COMPUESTOS DE FORMULA, Y A SALES, PROFARMACOS Y SOLVATOS FARMACEUTICAMENTE ACEPTABLES DE LOS MISMOS, EN LA QUE R1, R2, R3 Y R10 SON COMO SE HAN DEFINIDO EN ESTE DOCUMENTO. LOS COMPUESTOS DE FORMULA 1 SON AGENTES ANTIBACTERIANOS Y ANTIPROTOZOARIOS QUE PUEDEN USARSE PARA TRATAR DIVERSAS INFECCIONES BACTERIANAS Y PROTOZOARIAS Y TRASTORNOS RELACIONADOS CON TALES INFECCIONES. LA INVENCION TAMBIEN SE REFIERE A COMPOSICIONES FARMACEUTICAS QUE CONTIENEN LOS COMPUESTOS DE FORMULA 1 Y A PROCEDIMIENTOS DE TRATAMIENTO DE INFECCIONES BACTERIANAS Y PROTOZOARIAS MEDIANTE LA ADMINISTRACION DE LOS COMPUESTOS DE FORMULA 1.THIS INVENTION REFERS TO FORMULA COMPOUNDS, AND PHARMACEUTICALLY ACCEPTABLE SALTS, PROFARMACOS AND SOLVATES OF THE SAME, IN WHICH R1, R2, R3 AND R10 ARE AS DEFINED IN THIS DOCUMENT. FORMULA 1 COMPOUNDS ARE ANTIBACTERIAL AND ANTIPROTOZOAR AGENTS THAT CAN BE USED TO TREAT DIFFERENT BACTERIAL AND PROTOZOARY INFECTIONS AND DISORDERS RELATED TO SUCH INFECTIONS. THE INVENTION ALSO REFERS TO PHARMACEUTICAL COMPOSITIONS CONTAINING THE FORMULA 1 COMPOUNDS AND PROCEDURES FOR TREATMENT OF BACTERIAL INFECTIONS AND PROTOZOES THROUGH THE ADMINISTRATION OF FORMULA 1 COMPOUNDS.

SV2001000474A 2000-06-02 2001-06-01 HYGROMYCIN DERIVATIVES TO REF.PC11O32ABCZ / BB SV2002000474A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US20902300P 2000-06-02 2000-06-02

Publications (1)

Publication Number Publication Date
SV2002000474A true SV2002000474A (en) 2002-07-03

Family

ID=22777009

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2001000474A SV2002000474A (en) 2000-06-02 2001-06-01 HYGROMYCIN DERIVATIVES TO REF.PC11O32ABCZ / BB

Country Status (31)

Country Link
US (1) US6867230B2 (en)
EP (1) EP1287011A1 (en)
JP (1) JP2003535100A (en)
KR (1) KR20030010655A (en)
CN (1) CN1432019A (en)
AP (1) AP2002002669A0 (en)
AR (1) AR028667A1 (en)
AU (1) AU2001260528A1 (en)
BG (1) BG107265A (en)
BR (1) BR0111242A (en)
CA (1) CA2410643A1 (en)
CZ (1) CZ20023859A3 (en)
EA (1) EA200201167A1 (en)
EC (1) ECSP014093A (en)
EE (1) EE200200671A (en)
GT (1) GT200100099A (en)
HU (1) HUP0302263A2 (en)
IL (1) IL152984A0 (en)
IS (1) IS6618A (en)
MA (1) MA26909A1 (en)
MX (1) MXPA02011966A (en)
NO (1) NO20025704L (en)
OA (1) OA12277A (en)
PA (1) PA8518101A1 (en)
PE (1) PE20020334A1 (en)
PL (1) PL359179A1 (en)
SK (1) SK16612002A3 (en)
SV (1) SV2002000474A (en)
TN (1) TNSN01080A1 (en)
UY (1) UY26741A1 (en)
WO (1) WO2001092280A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2486055C (en) * 2002-05-16 2012-03-06 Sepracor, Inc. Amines that inhibit a mammalian anandamide transporter, and methods of use thereof
US20210275559A1 (en) * 2018-08-20 2021-09-09 Kim Lewis Hygromycin a compounds and methods of treating spirochete diseases
CU20180159A7 (en) * 2018-12-28 2020-10-20 Chengdu Olisynn Biotechnology Co Ltd DERIVATIVES OF SYNTHETIC OLIGOSACCHARIDS AS VACCINE AGAINST BORDETELLA PERTUSSIS

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1234567A (en) * 1915-09-14 1917-07-24 Edward J Quigley Soft collar.
US2004123A (en) * 1934-02-15 1935-06-11 Jr Robert B Loibl Pest exterminator
CA2331261C (en) * 1998-05-04 2004-07-27 Pfizer Products Inc. 2"-deoxy hygromycin derivatives
IL139165A0 (en) * 1998-05-04 2001-11-25 Pfizer Prod Inc Hygromycin a derivatives
CA2352332C (en) * 1998-12-02 2004-12-07 Pfizer Products Inc. Hygromycin a derivatives
KR20020063885A (en) * 1999-10-29 2002-08-05 화이자 프로덕츠 인코포레이티드 Hygromycin derivatives
US7654321B2 (en) * 2006-12-27 2010-02-02 Schlumberger Technology Corporation Formation fluid sampling apparatus and methods

Also Published As

Publication number Publication date
NO20025704D0 (en) 2002-11-27
BR0111242A (en) 2003-06-03
SK16612002A3 (en) 2004-04-06
EA200201167A1 (en) 2003-06-26
CZ20023859A3 (en) 2004-02-18
GT200100099A (en) 2002-01-31
PE20020334A1 (en) 2002-04-30
OA12277A (en) 2006-05-11
HUP0302263A2 (en) 2003-10-28
BG107265A (en) 2003-07-31
IL152984A0 (en) 2003-06-24
US6867230B2 (en) 2005-03-15
CN1432019A (en) 2003-07-23
NO20025704L (en) 2002-11-27
PA8518101A1 (en) 2002-09-17
AR028667A1 (en) 2003-05-21
AP2002002669A0 (en) 2002-12-31
UY26741A1 (en) 2001-12-28
PL359179A1 (en) 2004-08-23
CA2410643A1 (en) 2001-12-06
EE200200671A (en) 2004-08-16
KR20030010655A (en) 2003-02-05
US20030045528A1 (en) 2003-03-06
AU2001260528A1 (en) 2001-12-11
EP1287011A1 (en) 2003-03-05
TNSN01080A1 (en) 2005-11-10
IS6618A (en) 2002-11-14
WO2001092280A1 (en) 2001-12-06
ECSP014093A (en) 2002-01-25
JP2003535100A (en) 2003-11-25
MA26909A1 (en) 2004-12-20
MXPA02011966A (en) 2003-04-22

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