SV2002000337A - NEW FORM OF SALT AND POLYMORPHES REF. PCS10385AAJR / BB - Google Patents

NEW FORM OF SALT AND POLYMORPHES REF. PCS10385AAJR / BB

Info

Publication number
SV2002000337A
SV2002000337A SV2001000337A SV2001000337A SV2002000337A SV 2002000337 A SV2002000337 A SV 2002000337A SV 2001000337 A SV2001000337 A SV 2001000337A SV 2001000337 A SV2001000337 A SV 2001000337A SV 2002000337 A SV2002000337 A SV 2002000337A
Authority
SV
El Salvador
Prior art keywords
polymorphes
ref
salt
new form
formula
Prior art date
Application number
SV2001000337A
Other languages
Spanish (es)
Inventor
Patricia Ann Basford
Hodgson Paul Blaise
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of SV2002000337A publication Critical patent/SV2002000337A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

LA PRESENTE INVENCION PROPORCIONA MESILATO DE 4-AMINO-6,7-DIMETOXI-2-(5-METANOSULFONAMIDO-1,2,3,4-TETRAHIDROISOQUINOL-2-IL)-5-(2-PIRIDIL)QUINAZOLINA DE LA FORMULA, VER FORMULA, JUNTO CON PROCEDIMIENTOS PARA SU PREPARACION Y COMPOSICIONES QUE LO CONTIENEN.LA INVENCION TAMBIEN SE REFIERE A FORMAS POLIMORFICAS CRISTALINAS ANHIDRAS SUSTANCIALMENTE PURAS DE LA BASE LIBRE.LOS COMPUESTOS SON PARTICULARMENTE UTILES EN EL TRATAMIENTO DE LA HIPERPLASIA PROSTATICA BENIGNA.THIS INVENTION PROVIDES MESILATE OF 4-AMINO-6,7-DIMETOXI-2- (5-METHANOSULPHONAMIDE-1,2,3,4-TETRAHYDROISOQUINOL-2-IL) -5- (2-PIRIDIL) QUINAZOLINE OF THE FORMULA, SEE FORMULA, TOGETHER WITH PROCEDURES FOR THE PREPARATION AND COMPOSITIONS THAT CONTAIN IT. THE INVENTION ALSO REFERS TO SUBSTANTIALLY PURE ANCHORISTED CRYSTALLY POLYMORTIC FORMS OF THE FREE BASE. THE COMPOUNDS ARE PARTICULARLY USEFUL IN THE TREATMENT OF THE BENEFIT.

SV2001000337A 2000-03-03 2001-03-02 NEW FORM OF SALT AND POLYMORPHES REF. PCS10385AAJR / BB SV2002000337A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5200100A 2000-03-03 2000-03-03
US15900400A 2000-06-28 2000-06-28

Publications (1)

Publication Number Publication Date
SV2002000337A true SV2002000337A (en) 2002-07-03

Family

ID=40091694

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2001000337A SV2002000337A (en) 2000-03-03 2001-03-02 NEW FORM OF SALT AND POLYMORPHES REF. PCS10385AAJR / BB

Country Status (1)

Country Link
SV (1) SV2002000337A (en)

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SV2002000337A (en) NEW FORM OF SALT AND POLYMORPHES REF. PCS10385AAJR / BB
AR029482A1 (en) 4-AMINO-6,7-DIMETOXI-2- (5-METHANOSULPHONAMIDE-1,2,3,4-TETRAHYDROISOQUINOL-2-IL) -5- (2-PIRIDYL) QUINAZOLINE MASSILATE SALT, ANHYDRA CRYSTAL BASE FORM, PHARMACEUTICAL FORMULATION, USE IN THE MANUFACTURE OF MEDICINES AND PREPARATION METHOD

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