SI2084162T1 - Bicyclic triazoles as protein kinase modulators - Google Patents

Bicyclic triazoles as protein kinase modulators

Info

Publication number
SI2084162T1
SI2084162T1 SI200731025T SI200731025T SI2084162T1 SI 2084162 T1 SI2084162 T1 SI 2084162T1 SI 200731025 T SI200731025 T SI 200731025T SI 200731025 T SI200731025 T SI 200731025T SI 2084162 T1 SI2084162 T1 SI 2084162T1
Authority
SI
Slovenia
Prior art keywords
protein kinase
kinase modulators
bicyclic triazoles
triazoles
bicyclic
Prior art date
Application number
SI200731025T
Other languages
Slovenian (sl)
Inventor
Pierre-Yves Bounaud
Christopher Ronald Smith
Elizabeth Anne Jefferson
Original Assignee
Sgx Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sgx Pharmaceuticals Inc filed Critical Sgx Pharmaceuticals Inc
Priority claimed from PCT/US2007/081841 external-priority patent/WO2008051808A2/en
Publication of SI2084162T1 publication Critical patent/SI2084162T1/en

Links

SI200731025T 2006-10-23 2007-10-18 Bicyclic triazoles as protein kinase modulators SI2084162T1 (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US86255206P 2006-10-23 2006-10-23
US87030906P 2006-12-15 2006-12-15
US91376607P 2007-04-24 2007-04-24
US95284007P 2007-07-30 2007-07-30
PCT/US2007/081841 WO2008051808A2 (en) 2006-10-23 2007-10-18 Bicyclic triazoles as protein kinase modulators
EP07844414A EP2084162B1 (en) 2006-10-23 2007-10-18 Bicyclic triazoles as protein kinase modulators

Publications (1)

Publication Number Publication Date
SI2084162T1 true SI2084162T1 (en) 2012-11-30

Family

ID=41157042

Family Applications (2)

Application Number Title Priority Date Filing Date
SI200731024T SI2081937T1 (en) 2006-10-23 2007-10-18 Triazolopyridazine protein kinase modulators
SI200731025T SI2084162T1 (en) 2006-10-23 2007-10-18 Bicyclic triazoles as protein kinase modulators

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SI200731024T SI2081937T1 (en) 2006-10-23 2007-10-18 Triazolopyridazine protein kinase modulators

Country Status (3)

Country Link
CN (2) CN101558070A (en)
SI (2) SI2081937T1 (en)
ZA (1) ZA200902170B (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102812027B (en) * 2010-02-03 2015-01-07 因西特公司 Imidazo[1,2-b][1,2,4]triazines as c-met inhibitors
AR085183A1 (en) * 2010-07-30 2013-09-18 Lilly Co Eli COMPOUND 6- (1-METHYL-1H-PIRAZOL-4-IL) -3- (2-METHYL-2H-INDAZOL-5-ILTIO) - [1,2,4] TRIAZOL [4,3-B] PIRIDAZINE, PHARMACEUTICAL COMPOSITION THAT UNDERSTAND AND USE IT TO PREPARE A USEFUL MEDICINAL PRODUCT TO TREAT CANCER
CN103122000B (en) * 2012-09-03 2013-12-25 中美冠科生物技术(太仓)有限公司 High-selectivity c-Met kinase inhibitor used as antitumor drug
CN103664954A (en) * 2012-09-17 2014-03-26 杨育新 Compounds for treating traumatic brain injury diseases and application thereof
CN103655576A (en) * 2012-09-25 2014-03-26 杨子娇 Compounds for treating narrow chamber angle and application thereof
AU2014262326B2 (en) * 2013-05-10 2018-03-22 Jiangsu Hansoh Pharmaceutical Co., Ltd. [1,2,4] triazol [4,3-a] pyridine derivate, preparation method therefor or medical application thereof
GB201321745D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
CN103804289B (en) * 2014-01-16 2016-06-22 苏州泰利三佳纳米科技有限公司 The synthetic method of 6-methoxy quinoline
TW201607930A (en) * 2014-07-18 2016-03-01 百濟神州有限公司 5-amino-4-carbamoyl-pyrazole compounds as selective and irreversible T790M over WT EGFR kinase inhibitors and the use thereof
CN107922396B (en) 2015-07-20 2022-08-05 建新公司 Colony stimulating factor-1 receptor (CSF-1R) inhibitors
US10301325B2 (en) * 2015-09-24 2019-05-28 Shanghai Haiju Biological Technology Co., Ltd. Quinoline derivative, and pharmaceutical composition, preparation method and use thereof
BR112018006873A2 (en) * 2015-10-05 2018-11-06 The Trustees Of Columbia University In The City Of New York autophageal flow activators and phospholipase d and clearance of protein aggregates including tau and treatment of proteinopathies
CN106928233B (en) * 2015-12-31 2021-02-12 上海医药集团股份有限公司 Salt of quinoline compound, crystal form, preparation method, composition and application thereof
CN108864101B (en) * 2017-05-12 2019-12-17 中国科学院上海药物研究所 Deuterated SGX523 and application thereof
EP4267573A1 (en) 2020-12-23 2023-11-01 Genzyme Corporation Deuterated colony stimulating factor-1 receptor (csf-1r) inhibitors

Also Published As

Publication number Publication date
SI2081937T1 (en) 2012-11-30
CN101558070A (en) 2009-10-14
CN101553490A (en) 2009-10-07
ZA200902170B (en) 2010-06-30

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