SI2024372T1 - Tieno(3,2-d)pirimidinski derivat, uporaben kot inhibitor PI3K - Google Patents

Tieno(3,2-d)pirimidinski derivat, uporaben kot inhibitor PI3K

Info

Publication number
SI2024372T1
SI2024372T1 SI200730339T SI200730339T SI2024372T1 SI 2024372 T1 SI2024372 T1 SI 2024372T1 SI 200730339 T SI200730339 T SI 200730339T SI 200730339 T SI200730339 T SI 200730339T SI 2024372 T1 SI2024372 T1 SI 2024372T1
Authority
SI
Slovenia
Prior art keywords
åpyrimidine
thieno
pi3k inhibitor
derivative useful
derivative
Prior art date
Application number
SI200730339T
Other languages
English (en)
Inventor
Irina Chuckowree
Adrian FOLKES
Tim Hancox
Stephen Shuttleworth
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Priority claimed from PCT/IB2007/001058 external-priority patent/WO2007129161A2/en
Publication of SI2024372T1 publication Critical patent/SI2024372T1/sl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5355—Non-condensed oxazines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
SI200730339T 2006-04-26 2007-04-24 Tieno(3,2-d)pirimidinski derivat, uporaben kot inhibitor PI3K SI2024372T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US79496606P 2006-04-26 2006-04-26
EP07734376A EP2024372B1 (en) 2006-04-26 2007-04-24 Thieno[3,2-d]pyrimidine derivative useful as pi3k inhibitor
PCT/IB2007/001058 WO2007129161A2 (en) 2006-04-26 2007-04-24 Thieno [3, 2-d] pyrimidine derivative useful as pi3k inhibitor

Publications (1)

Publication Number Publication Date
SI2024372T1 true SI2024372T1 (sl) 2010-10-29

Family

ID=43034244

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200730339T SI2024372T1 (sl) 2006-04-26 2007-04-24 Tieno(3,2-d)pirimidinski derivat, uporaben kot inhibitor PI3K

Country Status (3)

Country Link
EP (2) EP2246354A1 (sl)
PL (1) PL2024372T3 (sl)
SI (1) SI2024372T1 (sl)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3773919A (en) 1969-10-23 1973-11-20 Du Pont Polylactide-drug mixtures
AU5261001A (en) 2000-04-27 2001-11-12 Imperial Cancer Research Technology Ltd Condensed heteroaryl derivatives
US6608053B2 (en) * 2000-04-27 2003-08-19 Yamanouchi Pharmaceutical Co., Ltd. Fused heteroaryl derivatives
US6894055B2 (en) * 2001-10-24 2005-05-17 Iconix Pharmaceuticals Inc. Thieno-2′,3′ -5,6pyrimido[3,4-A]-1,2,4-triazole derivatives as modulators of phoshoinositide 3-kinase
WO2005007083A2 (en) * 2003-06-18 2005-01-27 Smithkline Beecham Corporation Chemical compounds
EP1682123A1 (en) * 2003-11-07 2006-07-26 SmithKline Beecham (Cork) Limited Cancer treatment method
GB0423653D0 (en) * 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds

Also Published As

Publication number Publication date
EP2246354A1 (en) 2010-11-03
EP2024372A2 (en) 2009-02-18
EP2024372B1 (en) 2010-06-23
PL2024372T3 (pl) 2010-11-30

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