SI1732931T1 - METHODS FOR THE PREPARATION OF (3R,3aS,6aR) HEXAHYDRO-FURO(2,3-b)FURAN-3-OL - Google Patents

METHODS FOR THE PREPARATION OF (3R,3aS,6aR) HEXAHYDRO-FURO(2,3-b)FURAN-3-OL

Info

Publication number
SI1732931T1
SI1732931T1 SI200532087A SI200532087A SI1732931T1 SI 1732931 T1 SI1732931 T1 SI 1732931T1 SI 200532087 A SI200532087 A SI 200532087A SI 200532087 A SI200532087 A SI 200532087A SI 1732931 T1 SI1732931 T1 SI 1732931T1
Authority
SI
Slovenia
Prior art keywords
furo
hexahydro
furan
preparation
methods
Prior art date
Application number
SI200532087A
Other languages
Slovenian (sl)
Inventor
Peter Jan Leonard Mario Quaedflieg
Bart Rudolf Romanie Kesteleyn
Robert Jan Vijn
Constantinus Simon Maria Liebregts
Jacob Hermanus Matheus Hero Kooistra
Franciscus Alphons Marie Lommen
Original Assignee
Janssen Sciences Ireland Uc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34928933&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI1732931(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Sciences Ireland Uc filed Critical Janssen Sciences Ireland Uc
Publication of SI1732931T1 publication Critical patent/SI1732931T1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D307/18—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/20—Oxygen atoms
SI200532087A 2004-03-31 2005-03-31 METHODS FOR THE PREPARATION OF (3R,3aS,6aR) HEXAHYDRO-FURO(2,3-b)FURAN-3-OL SI1732931T1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP04101336 2004-03-31
PCT/EP2005/051452 WO2005095410A1 (en) 2004-03-31 2005-03-31 METHODS FOR THE PREPARATION OF (3R,3aS,6aR) HEXAHYDRO-FURO[2,3-b]FURAN-3-OL
EP05729507.3A EP1732931B1 (en) 2004-03-31 2005-03-31 METHODS FOR THE PREPARATION OF (3R,3aS,6aR) HEXAHYDRO-FURO[2,3-b]FURAN-3-OL

Publications (1)

Publication Number Publication Date
SI1732931T1 true SI1732931T1 (en) 2016-10-28

Family

ID=34928933

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200532087A SI1732931T1 (en) 2004-03-31 2005-03-31 METHODS FOR THE PREPARATION OF (3R,3aS,6aR) HEXAHYDRO-FURO(2,3-b)FURAN-3-OL

Country Status (28)

Country Link
US (1) US7595408B2 (en)
EP (1) EP1732931B1 (en)
JP (1) JP4778955B2 (en)
KR (1) KR101135156B1 (en)
CN (1) CN1938316B (en)
AP (1) AP2528A (en)
AU (1) AU2005229435B2 (en)
BR (1) BRPI0509514B1 (en)
CA (1) CA2559959C (en)
CY (1) CY1119150T1 (en)
DK (1) DK1732931T3 (en)
ES (1) ES2587571T3 (en)
HR (1) HRP20161031T1 (en)
HU (1) HUE029886T2 (en)
IL (1) IL178019A (en)
LT (1) LT1732931T (en)
ME (1) ME02525B (en)
NO (1) NO338175B1 (en)
NZ (1) NZ549971A (en)
PL (1) PL1732931T3 (en)
PT (1) PT1732931T (en)
RS (1) RS55011B1 (en)
RU (1) RU2421458C2 (en)
SI (1) SI1732931T1 (en)
TW (1) TWI383975B (en)
UA (1) UA100835C2 (en)
WO (1) WO2005095410A1 (en)
ZA (1) ZA200609008B (en)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE602007012365D1 (en) 2006-11-09 2011-03-17 Little Island Co Cork PROCESS FOR PREPARING HEXAHYDROFUROA2,3-BÜFURAN-3-OL
CN101024646B (en) * 2007-02-06 2010-07-14 启东东岳药业有限公司 Method for purifying methoxyfuran-furan-2-one
DE602008005012D1 (en) 2007-04-27 2011-03-31 Little Island Co Cork PREPARATION FOR N-ISOBUTYL-N- (2-HYDROXY-RIVATE
WO2009030733A1 (en) * 2007-09-04 2009-03-12 Dsm Ip Assets B.V. Method for the synthesis of 4-alkoxy-, 4-hydroxy- and 4-aryloxy-substituted tetrahydro-furo[3,4-b]furan-2(3h)-one compounds
JP2012510426A (en) 2008-12-03 2012-05-10 マサチューセッツ インスティテュート オブ テクノロジー Multifunctional composite based on coated nanostructure base
US8921415B2 (en) 2009-01-29 2014-12-30 Mapi Pharma Ltd. Polymorphs of darunavir
EP2493891A2 (en) 2009-10-30 2012-09-05 Lupin Limited A novel process for preparation of darunavir and darunavir ethanolate of fine particle size
WO2011092687A1 (en) 2010-01-28 2011-08-04 Mapi Pharma Hk Limited Process for the preparation of darunavir and darunavir intermediates
WO2014016660A2 (en) 2012-07-24 2014-01-30 Laurus Labs Private Limited A process for preparation of darunavir
CN103864813B (en) * 2012-12-18 2017-02-22 上海迪赛诺化学制药有限公司 Synthetic methods of hexahydrofuro[2,3-b]furan-3-ol and enantiomer thereof
CN104628552A (en) * 2015-02-09 2015-05-20 许昌豪丰化学科技有限公司 New quenching system and application thereof
WO2017041228A1 (en) * 2015-09-08 2017-03-16 浙江九洲药业股份有限公司 Method for preparing hexahydrofurofuranol derivative, intermediate thereof and preparation method thereof
US10407438B2 (en) 2016-10-27 2019-09-10 Gilead Sciences, Inc. Crystalline forms of darunavir
CN110272398B (en) 2018-03-16 2022-11-29 江苏瑞科医药科技有限公司 Process for producing hexahydrofurofuranol derivative, intermediate therefor, and process for producing the intermediate
KR20210138609A (en) 2019-02-15 2021-11-19 디지렌즈 인코포레이티드. Method and apparatus for providing a holographic waveguide display using an integral grating
CN115557964A (en) * 2022-10-18 2023-01-03 启东东岳药业有限公司 Preparation method of pharmaceutical compound

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0427693A1 (en) * 1989-10-11 1991-05-15 Monsanto Company Method for azide displacement of alpha-triflates of 1,5-lactones
ES2127938T3 (en) 1993-08-24 1999-05-01 Searle & Co HYDROXYETHYLAMINE SULPHONAMIDES USEFUL AS RETROVIRAL PROTEASE INHIBITORS.
AU699483B2 (en) * 1994-03-07 1998-12-03 Vertex Pharmaceuticals Incorporated Sulphonamide derivatives as aspartyl protease inhibitors
WO1999065870A2 (en) 1998-06-19 1999-12-23 Vertex Pharmaceuticals Incorporated Sulfonamide inhibitors of aspartyl protease
AU771780B2 (en) 1998-06-23 2004-04-01 Board Of Trustees Of The University Of Illinois, The Fitness assay and associated methods
AU3485800A (en) 1999-02-12 2000-08-29 Vertex Pharmaceuticals Incorporated Inhibitors of aspartyl protease
AR031520A1 (en) 1999-06-11 2003-09-24 Vertex Pharma AN INHIBITOR COMPOSITE OF ASPARTILO PROTEASA, A COMPOSITION THAT INCLUDES IT AND A METHOD TO TREAT A PATIENT WITH SUCH COMPOSITION
CZ300031B6 (en) 1999-10-06 2009-01-14 Tibotec Pharmaceuticals Ltd. Hexahydrofur[2,3-b]furan-3-yl-N-{3-[(1,3-benzodioxol-5-ylsulfonyl) (isobutyl)amino]-1-benzyl-2-hydroxypropyl}carbamate and pharmaceutical composition in which the carbamate is comprised
HU229505B1 (en) * 2001-09-10 2014-01-28 Tibotec Pharm Ltd Method for the preparation of hexahydro-furo[2,3-b]furan-3-ol

Also Published As

Publication number Publication date
CN1938316B (en) 2012-12-12
EP1732931A1 (en) 2006-12-20
DK1732931T3 (en) 2016-08-29
ES2587571T3 (en) 2016-10-25
AU2005229435A1 (en) 2005-10-13
NO20064977L (en) 2006-10-31
RU2421458C2 (en) 2011-06-20
AU2005229435B2 (en) 2011-07-07
TWI383975B (en) 2013-02-01
JP4778955B2 (en) 2011-09-21
NO338175B1 (en) 2016-08-01
ZA200609008B (en) 2008-07-30
RU2006138228A (en) 2008-05-10
CY1119150T1 (en) 2018-01-10
ME02525B (en) 2017-02-20
LT1732931T (en) 2016-09-12
HRP20161031T1 (en) 2016-10-21
WO2005095410A1 (en) 2005-10-13
CN1938316A (en) 2007-03-28
AP2528A (en) 2012-12-10
IL178019A0 (en) 2006-12-31
BRPI0509514B1 (en) 2022-09-27
CA2559959A1 (en) 2005-10-13
BRPI0509514A (en) 2007-09-11
NZ549971A (en) 2010-12-24
HUE029886T2 (en) 2017-04-28
BRPI0509514A8 (en) 2016-02-10
KR20070026479A (en) 2007-03-08
JP2007530638A (en) 2007-11-01
US7595408B2 (en) 2009-09-29
PL1732931T3 (en) 2016-11-30
PT1732931T (en) 2016-07-14
EP1732931B1 (en) 2016-05-18
RS55011B1 (en) 2016-11-30
UA100835C2 (en) 2013-02-11
AP2006003748A0 (en) 2006-10-31
IL178019A (en) 2014-02-27
TW200602346A (en) 2006-01-16
US20070208184A1 (en) 2007-09-06
CA2559959C (en) 2013-11-19
KR101135156B1 (en) 2012-04-23

Similar Documents

Publication Publication Date Title
AP2528A (en) Methods for the preparation of (3R,3aS,6aR) hexahydro- furo [2,3-b] furan-3-ol
IL194122A (en) Process for the preparation of (3r,3as,6ar)-hexahydrofuro[2,3-b]furan-3-ol
WO2008055970A3 (en) Methods for the preparation of hexahydrofuro[2,3-b]furan-3-ol
IL211191A (en) Oxalate salt of (3as,4r,6s,6ar)-6-(2-hydroxyethoxy)-2,2-dimethyltetrahydro-3ah-cyclopenta[d][1,3]dioxol-4-amine
HUP0402140A3 (en) Method for the preparation of hexahydro-furo[2,3-b]furan-3-ol
ZA201202025B (en) INTERMEDIATES USEFUL IN THE PREPARATION OF PYRROLO[2,3-b] PYRIDINE DERIVATIVES
ME01059B (en) Process for the preparation of (3r,3as,6ar)-hexahydrofuro [2,3-b] furan-3-yl (1s,2r)-3-[[(4-aminophenyl) sulfonyl] (isobutyl) amino]-1-benzyl-2-hydroxypropylcarbamate
ZA200708490B (en) Intermediate compounds for the preparation of trans-5-chloro-2-methyl-2,3,3a, 12b-tetrahydro-1H-dibenz[2,3:6,7] oxepino[4,5-c]pyrrole
AU2003287038A8 (en) Method of preparing (3r, 3as, 6ar) -3- hydroxyhexahydrofuro (2, 3-b) furan and related compounds
PL1678182T3 (en) Process for preparing substituted 5-amino-pyrazolo- [4,3-e]-1,2,4-triazolo [1,5-c]pyrimidines
DK1784403T3 (en) Pyrrolo [3,2-b] pyridine derivatives as well as processes for their preparation
SMT201500309B (en) PROCEDURE FOR THE PREPARATION OF BENZYL [(3AS, 4R, 6S, 6AR) -6-HYDROXY-2,2-DIMETHYLTETRAIDRO-3AHCYCLOPENTA [D] [1,3] DIOSSOL] -4-THE] CARBAMMATE AND INTERMEDIATE IN THE PROCEDURE
LT2643326T (en) Process for the preparation of (3R, 3aS, 6aR)-hexahydrofuro[2,3-b]furan-3-ol