SI1611144T1 - Derivatives of 2-(8,9-dioxo-2,6-diazabicyclo(5.2.0)non-1(7)-en-2-yl)alkyl phosphonic acid and their use as n-methyl-d-aspartate (nmda) recetor antagonists - Google Patents

Derivatives of 2-(8,9-dioxo-2,6-diazabicyclo(5.2.0)non-1(7)-en-2-yl)alkyl phosphonic acid and their use as n-methyl-d-aspartate (nmda) recetor antagonists

Info

Publication number
SI1611144T1
SI1611144T1 SI200431536T SI200431536T SI1611144T1 SI 1611144 T1 SI1611144 T1 SI 1611144T1 SI 200431536 T SI200431536 T SI 200431536T SI 200431536 T SI200431536 T SI 200431536T SI 1611144 T1 SI1611144 T1 SI 1611144T1
Authority
SI
Slovenia
Prior art keywords
recetor
nmda
dioxo
diazabicyclo
aspartate
Prior art date
Application number
SI200431536T
Other languages
Slovenian (sl)
Inventor
Reinhardt Bernhard Baudy
John Anthony Butera
Original Assignee
Wyeth Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Llc filed Critical Wyeth Llc
Priority claimed from PCT/US2004/010596 external-priority patent/WO2004092189A1/en
Publication of SI1611144T1 publication Critical patent/SI1611144T1/en

Links

SI200431536T 2003-04-09 2004-04-07 Derivatives of 2-(8,9-dioxo-2,6-diazabicyclo(5.2.0)non-1(7)-en-2-yl)alkyl phosphonic acid and their use as n-methyl-d-aspartate (nmda) recetor antagonists SI1611144T1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US46149003P 2003-04-09 2003-04-09
PCT/US2004/010596 WO2004092189A1 (en) 2003-04-09 2004-04-07 Derivatives of 2-(8,9-dioxo-2,6-diazabicyclo(5.2.0)non-1(7)-en-2-yl)alkyl phosphonic acid and their use as n-methyl-d-aspartate (nmda) recetor antagonists
EP04759168A EP1611144B1 (en) 2003-04-09 2004-04-07 Derivatives of 2-(8,9-dioxo-2,6-diazabicyclo(5.2.0)non-1(7)-en-2-yl)alkyl phosphonic acid and their use as n-methyl-d-aspartate (nmda) recetor antagonists

Publications (1)

Publication Number Publication Date
SI1611144T1 true SI1611144T1 (en) 2010-12-31

Family

ID=43416258

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200431536T SI1611144T1 (en) 2003-04-09 2004-04-07 Derivatives of 2-(8,9-dioxo-2,6-diazabicyclo(5.2.0)non-1(7)-en-2-yl)alkyl phosphonic acid and their use as n-methyl-d-aspartate (nmda) recetor antagonists

Country Status (1)

Country Link
SI (1) SI1611144T1 (en)

Similar Documents

Publication Publication Date Title
PL1611144T3 (en) Derivatives of 2-(8,9-dioxo-2,6-diazabicyclo(5.2.0)non-1(7)-en-2-yl)alkyl phosphonic acid and their use as n-methyl-d-aspartate (nmda) recetor antagonists
HRP20090281T1 (en) 1,2,3,4-tetrasubstituted indole for the treatment of respiratory diseases
AP1614A (en) New heterocyclic compounds, their preparation and their use as medicaments, in particular as anti-bacterial agents.
PT911333E (en) PYRAZOLINE-4,3-D | PYRIMIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
WO2002098856A3 (en) Piperazine oxyquinoline (naphthaline) platelet adenosine diphosphate receptor antagonists
IL161074A0 (en) Lactam derivatives as antagonists for human 11cby receptors
MXPA05009508A (en) 6-substituted nicotinamide derivatives as opioid receptor antagonists.
DE502004011328D1 (en) SUBSTITUTED HEXAHYDRO-PYRAZINO (1,2-A) PYRIMIDINE-4,7-DION DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, AND THEIR USE AS A MEDICAMENT
HK1155146A1 (en) Indene derivatives as pharmaceutical agents
GB0415365D0 (en) Pyrimidine derivatives
UA95223C2 (en) Pyrido-pyrido pyrimidine derivatives, preparation thereof, therapeutic use thereof
CY1105028T1 (en) SUBSTITUTED C-IMIDAZO-[1,2-A]PYRIDIN-3-YL-METHYLAMINES
WO2004100865A3 (en) New benzimidazole derivatives
WO2002048148A3 (en) Pyrazolopyridine derivatives
IL169184A0 (en) Aromatic compounds as anti-inflammatory, immunomdulatory and anti-proliferatory agents
WO2003051274A3 (en) Benzodiazepine derivatives, preparation thereof and use thereof
CY1105019T1 (en) SUBSTITUTED C-IMIDAZO-[1,2-A]PYRIDIN-3-YL-METHYLAMINES
IL164555A0 (en) 4-'7-Halo-2-quino (xa-)linyloxy! phenoxy-propionicacid derivatives as antineoplastic agents
IL195837A0 (en) 4-amino-3-arylamino-6-arylpyrazolo[3,4-d]
WO2004067703A3 (en) 5ht7 antagonists and inverse agonists
AU2001246999A1 (en) New neurokinin antagonists for use as medicaments
EP1610795A4 (en) Heterocyclic substituted 1,4-dihydro-4-oxo-1,8-naphthpyridine analogs
ZA200603236B (en) Methods for the preparation of {2-[8,9-dioxo-2,6-diaza-bicyclo[5.2.0]-non-1(7)-en-2-yl]ethyl} phosphonic acid and esters thereof
DK0896822T3 (en) 4-Aminopyrrole (3,2-d) pyrimidines as neuropeptide Y receptor antagonists
MXPA02012400A (en) Hetaryl-substituted heterocycles.