SI1461338T1 - Improved process for the preparation of 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-6,7,8,9-tetrahydro-2-methyl-4h-pyrido(1,2-a)pyrimidin-4-one
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Improved process for the preparation of 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-6,7,8,9-tetrahydro-2-methyl-4h-pyrido(1,2-a)pyrimidin-4-one
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SI1461338T1
SI1461338T1SI200230569TSI200230569TSI1461338T1SI 1461338 T1SI1461338 T1SI 1461338T1SI 200230569 TSI200230569 TSI 200230569TSI 200230569 TSI200230569 TSI 200230569TSI 1461338 T1SI1461338 T1SI 1461338T1
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Priority claimed from HU0104873Aexternal-prioritypatent/HU227118B1/en
Application filed by Egis Gyogyszergyar NyrtfiledCriticalEgis Gyogyszergyar Nyrt
Publication of SI1461338T1publicationCriticalpatent/SI1461338T1/en
SI200230569T2001-11-132002-11-13Improved process for the preparation of 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-6,7,8,9-tetrahydro-2-methyl-4h-pyrido(1,2-a)pyrimidin-4-one
SI1461338T1
(en)
Process for the preparation of 3-{2-[4-(6-fluoro-1,2-benzizoxazol-3-yl)-1-piperidinyl]-ethyl}-6,7,8,9-tetrahydro-2-methyl-4h-pyrido[1,2-a]pyrimidin-4-one
Improved process for the preparation of 3-{2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl}-6,7,8,9-tetrahydro-2-methyl-4h-pyrido[1,2-a]pyrimidin-4-one
Improved process for the preparation of 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-6,7,8,9-tetrahydro-2-methyl-4h-pyrido(1,2-a)pyrimidin-4-one
Improved process for the preparation of 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-6,7,8,9-tetrahydro-2-methyl-4h-pyrido(1,2-a)pyrimidin-4-one
Process for preparation of aseptic 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3- yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4h- pyrido[1,2-a]pyrimidin-4-one palmitate ester
Refined process for the preparation of 3-{2-[4-(6-fluoro-1,2-benzizoxazol-3-yl)-1-piperidinyl]-ethyl}-6,7,8,9-tetrahydro-2-methyl-4h-pyrido[1,2-a]pyrimidin-4-one
Improved process for the preparation of 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-6,7,8,9-tetrahydro-2-methyl-4h-pyrido(1,2-a)pyrimidin-4-one
Improved process for the preparation of 3-{2-`4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl!ethyl}-6,7,8,9-tetrahydro-2-methyl-4h-pyrido`1,2-a!pyrimidin-4-one
Substituted alkylpyridazinone derivatives, process for their preparation, their use for the preparation of pharmaceutical compositions with anxiolytic activity