SG11201702632QA - Pharmaceutical composition of fused aminodihydrothiazine derivative - Google Patents

Pharmaceutical composition of fused aminodihydrothiazine derivative

Info

Publication number
SG11201702632QA
SG11201702632QA SG11201702632QA SG11201702632QA SG11201702632QA SG 11201702632Q A SG11201702632Q A SG 11201702632QA SG 11201702632Q A SG11201702632Q A SG 11201702632QA SG 11201702632Q A SG11201702632Q A SG 11201702632QA SG 11201702632Q A SG11201702632Q A SG 11201702632QA
Authority
SG
Singapore
Prior art keywords
pharmaceutical composition
fused aminodihydrothiazine
aminodihydrothiazine derivative
derivative
fused
Prior art date
Application number
SG11201702632QA
Inventor
Yasuhiro Zaima
Kazuo Kazama
Shuntaro Arase
Kentaro Nagane
Kanta Horie
Yosuke Ueki
Original Assignee
Eisai R&D Man Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai R&D Man Co Ltd filed Critical Eisai R&D Man Co Ltd
Publication of SG11201702632QA publication Critical patent/SG11201702632QA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/20Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SG11201702632QA 2014-10-10 2015-10-08 Pharmaceutical composition of fused aminodihydrothiazine derivative SG11201702632QA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2014209289 2014-10-10
PCT/JP2015/078688 WO2016056638A1 (en) 2014-10-10 2015-10-08 Pharmaceutical composition of fused aminodihydrothiazine derivative

Publications (1)

Publication Number Publication Date
SG11201702632QA true SG11201702632QA (en) 2017-05-30

Family

ID=55653242

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201702632QA SG11201702632QA (en) 2014-10-10 2015-10-08 Pharmaceutical composition of fused aminodihydrothiazine derivative

Country Status (14)

Country Link
US (1) US10117876B2 (en)
EP (1) EP3205343B1 (en)
JP (3) JP6590822B2 (en)
KR (1) KR102524217B1 (en)
CN (1) CN107106568B (en)
AU (1) AU2015329027B2 (en)
BR (1) BR112017007293B1 (en)
CA (1) CA2963761C (en)
ES (1) ES2909797T3 (en)
IL (1) IL251559B (en)
MX (1) MX370338B (en)
RU (1) RU2710227C2 (en)
SG (1) SG11201702632QA (en)
WO (1) WO2016056638A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG11201702632QA (en) * 2014-10-10 2017-05-30 Eisai R&D Man Co Ltd Pharmaceutical composition of fused aminodihydrothiazine derivative
CN117244056A (en) 2016-10-27 2023-12-19 卫材研究发展管理有限公司 Compositions comprising anti-Abeta-protofibril antibodies and beta-secretase BACE1 inhibitors for the treatment of Alzheimer's disease
JP6326114B2 (en) * 2016-11-01 2018-05-16 エルメッド エーザイ株式会社 Levetiracetam-containing pharmaceutical composition and method for producing the same, method for preventing delay of dissolution and / or dissolution of levetiracetam-containing pharmaceutical composition, and agent for preventing delay and / or dissolution of levetiracetam-containing pharmaceutical composition

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20010042536A (en) * 1998-04-08 2001-05-25 히라타 다다시 Tablet manufacturing method and tablet
EP1813274B1 (en) * 2004-10-06 2009-12-16 Eisai R&D Management Co., Ltd. Medicinal composition, process for producing the same, and method of stabilizing dihydropyridine compound in medicinal composition
JP5158922B2 (en) * 2006-02-24 2013-03-06 塩野義製薬株式会社 Composition containing vitamin B12
AU2009205072C1 (en) * 2008-01-18 2016-10-13 Eisai R & D Management Co., Ltd. Condensed aminodihydrothiazine derivative
KR20100121483A (en) * 2008-02-11 2010-11-17 다이닛본 스미토모 세이야꾸 가부시끼가이샤 Tablet having improved elution properties
EP2665716B1 (en) * 2011-01-21 2017-03-08 Eisai R&D Management Co., Ltd. Methods and compounds useful in the synthesis of fused aminodihydrothiazine derivatives
JP2014037356A (en) * 2012-08-13 2014-02-27 Takada Seiyaku Kk Candesartan cilexetil oral formulation
US20140271911A1 (en) * 2014-03-26 2014-09-18 James Wallace Lithium and a beta-secretase inhibitor for the treatment of alzheimer's disease
SG11201702632QA (en) * 2014-10-10 2017-05-30 Eisai R&D Man Co Ltd Pharmaceutical composition of fused aminodihydrothiazine derivative

Also Published As

Publication number Publication date
RU2017111801A (en) 2018-11-13
CA2963761A1 (en) 2016-04-14
BR112017007293B1 (en) 2022-12-13
IL251559A0 (en) 2017-05-29
EP3205343A4 (en) 2018-06-06
MX370338B (en) 2019-12-10
AU2015329027A1 (en) 2017-04-27
CN107106568B (en) 2023-09-26
KR20170066397A (en) 2017-06-14
JP2020125330A (en) 2020-08-20
EP3205343A1 (en) 2017-08-16
AU2015329027B2 (en) 2020-04-30
JPWO2016056638A1 (en) 2017-07-20
KR102524217B1 (en) 2023-04-21
BR112017007293A2 (en) 2017-12-26
IL251559B (en) 2021-02-28
JP2019196395A (en) 2019-11-14
CA2963761C (en) 2023-10-17
EP3205343B1 (en) 2022-01-26
JP6590822B2 (en) 2019-10-16
US20180263998A1 (en) 2018-09-20
RU2710227C2 (en) 2019-12-25
US10117876B2 (en) 2018-11-06
WO2016056638A1 (en) 2016-04-14
MX2017004418A (en) 2017-06-26
RU2017111801A3 (en) 2019-02-12
CN107106568A (en) 2017-08-29
ES2909797T3 (en) 2022-05-10

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