SG11201700741WA - Azole benzene derivative and crystalline form thereof - Google Patents
Azole benzene derivative and crystalline form thereofInfo
- Publication number
- SG11201700741WA SG11201700741WA SG11201700741WA SG11201700741WA SG11201700741WA SG 11201700741W A SG11201700741W A SG 11201700741WA SG 11201700741W A SG11201700741W A SG 11201700741WA SG 11201700741W A SG11201700741W A SG 11201700741WA SG 11201700741W A SG11201700741W A SG 11201700741WA
- Authority
- SG
- Singapore
- Prior art keywords
- crystalline form
- benzene derivative
- azole benzene
- azole
- derivative
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/04—Drugs for disorders of the urinary system for urolithiasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Immunology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2014155032 | 2014-07-30 | ||
JP2014155030 | 2014-07-30 | ||
PCT/JP2015/071530 WO2016017708A1 (en) | 2014-07-30 | 2015-07-29 | Azole benzene derivative and crystal thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
SG11201700741WA true SG11201700741WA (en) | 2017-02-27 |
Family
ID=55217605
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11201700741WA SG11201700741WA (en) | 2014-07-30 | 2015-07-29 | Azole benzene derivative and crystalline form thereof |
Country Status (31)
Country | Link |
---|---|
US (1) | US10179780B2 (en) |
EP (1) | EP3176166B1 (en) |
JP (1) | JP6279085B2 (en) |
KR (1) | KR102474325B1 (en) |
CN (1) | CN106661014B (en) |
AU (1) | AU2015297501B2 (en) |
BR (1) | BR112017001657B1 (en) |
CA (1) | CA2956553C (en) |
CY (1) | CY1121189T1 (en) |
DK (1) | DK3176166T3 (en) |
ES (1) | ES2712850T3 (en) |
HR (1) | HRP20182084T1 (en) |
HU (1) | HUE042576T2 (en) |
IL (1) | IL250143B (en) |
LT (1) | LT3176166T (en) |
ME (1) | ME03319B (en) |
MX (1) | MX370524B (en) |
MY (1) | MY180730A (en) |
NZ (1) | NZ729068A (en) |
PH (1) | PH12017500124A1 (en) |
PL (1) | PL3176166T3 (en) |
PT (1) | PT3176166T (en) |
RS (1) | RS58315B1 (en) |
RU (1) | RU2701515C2 (en) |
SA (1) | SA517380787B1 (en) |
SG (1) | SG11201700741WA (en) |
SI (1) | SI3176166T1 (en) |
TR (1) | TR201902314T4 (en) |
TW (1) | TWI688563B (en) |
WO (1) | WO2016017708A1 (en) |
ZA (1) | ZA201700664B (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR102259713B1 (en) * | 2014-07-30 | 2021-06-01 | 데이진 화-마 가부시키가이샤 | Xanthine oxidase inhibitor |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK0513379T3 (en) | 1990-11-30 | 1996-09-30 | Teijin Ltd | 2-Arylthiazole derivatives and pharmaceutical compositions containing them |
WO1996031211A1 (en) * | 1995-04-07 | 1996-10-10 | Teijin Limited | Protective agent for organ or tissue |
SK287928B6 (en) | 1998-06-19 | 2012-04-03 | Teijin Pharma Limited | Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4- methyl-5-thiazole-carboxylic acid and processes for the preparation thereof |
JP2002105067A (en) | 2000-09-28 | 2002-04-10 | Teijin Ltd | 2-phenylthiazone derivative and medicine composition comprising the same as active ingredient |
WO2007043400A1 (en) | 2005-10-07 | 2007-04-19 | Kissei Pharmaceutical Co., Ltd. | Nitrogenated aromatic heterocyclic compound and pharmaceutical composition comprising the same |
WO2008126770A1 (en) * | 2007-04-05 | 2008-10-23 | Astellas Pharma Inc. | Method for producing triarylcarboxylic acid derivative |
EP2133331A4 (en) | 2007-04-11 | 2011-06-22 | Kissei Pharmaceutical | 5-membered heterocyclic derivative and use thereof for medical purposes |
WO2010018458A2 (en) | 2008-08-12 | 2010-02-18 | Crystalgenomics, Inc. | Phenol derivatives and methods of use thereof |
WO2010128163A2 (en) | 2009-05-08 | 2010-11-11 | Pike Pharma Gmbh | Small molecule inhibitors of influenza a and b virus and respiratory syncytial virus replication |
WO2011101867A2 (en) | 2010-02-19 | 2011-08-25 | Cadila Healthcare Limited | Substantially pure salts of febuxostat and processes for preparation thereof |
EP2563768A4 (en) | 2010-04-29 | 2013-07-31 | Reddys Lab Ltd Dr | Preparation of febuxostat |
TWI606048B (en) * | 2013-01-31 | 2017-11-21 | 帝人製藥股份有限公司 | Azolebenzene derivatives |
-
2015
- 2015-07-29 CA CA2956553A patent/CA2956553C/en active Active
- 2015-07-29 HU HUE15827218A patent/HUE042576T2/en unknown
- 2015-07-29 JP JP2016538406A patent/JP6279085B2/en active Active
- 2015-07-29 AU AU2015297501A patent/AU2015297501B2/en active Active
- 2015-07-29 ES ES15827218T patent/ES2712850T3/en active Active
- 2015-07-29 US US15/329,813 patent/US10179780B2/en active Active
- 2015-07-29 LT LTEP15827218.7T patent/LT3176166T/en unknown
- 2015-07-29 TW TW104124554A patent/TWI688563B/en active
- 2015-07-29 PL PL15827218T patent/PL3176166T3/en unknown
- 2015-07-29 RS RS20190109A patent/RS58315B1/en unknown
- 2015-07-29 EP EP15827218.7A patent/EP3176166B1/en active Active
- 2015-07-29 RU RU2017106052A patent/RU2701515C2/en active
- 2015-07-29 SI SI201530528T patent/SI3176166T1/en unknown
- 2015-07-29 MY MYPI2017700278A patent/MY180730A/en unknown
- 2015-07-29 DK DK15827218.7T patent/DK3176166T3/en active
- 2015-07-29 SG SG11201700741WA patent/SG11201700741WA/en unknown
- 2015-07-29 ME MEP-2019-22A patent/ME03319B/en unknown
- 2015-07-29 NZ NZ729068A patent/NZ729068A/en unknown
- 2015-07-29 WO PCT/JP2015/071530 patent/WO2016017708A1/en active Application Filing
- 2015-07-29 KR KR1020177002443A patent/KR102474325B1/en active IP Right Grant
- 2015-07-29 PT PT15827218T patent/PT3176166T/en unknown
- 2015-07-29 MX MX2017000412A patent/MX370524B/en active IP Right Grant
- 2015-07-29 BR BR112017001657-5A patent/BR112017001657B1/en active IP Right Grant
- 2015-07-29 CN CN201580040080.6A patent/CN106661014B/en active Active
- 2015-07-29 TR TR2019/02314T patent/TR201902314T4/en unknown
-
2017
- 2017-01-16 IL IL25014317A patent/IL250143B/en active IP Right Grant
- 2017-01-20 PH PH12017500124A patent/PH12017500124A1/en unknown
- 2017-01-24 SA SA517380787A patent/SA517380787B1/en unknown
- 2017-01-26 ZA ZA2017/00664A patent/ZA201700664B/en unknown
-
2018
- 2018-12-10 HR HRP20182084TT patent/HRP20182084T1/en unknown
-
2019
- 2019-01-24 CY CY20191100112T patent/CY1121189T1/en unknown
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