SG11201609483YA - Novel crystalline polymorphs of pyridine derivative and method for producing the same - Google Patents

Novel crystalline polymorphs of pyridine derivative and method for producing the same

Info

Publication number
SG11201609483YA
SG11201609483YA SG11201609483YA SG11201609483YA SG11201609483YA SG 11201609483Y A SG11201609483Y A SG 11201609483YA SG 11201609483Y A SG11201609483Y A SG 11201609483YA SG 11201609483Y A SG11201609483Y A SG 11201609483YA SG 11201609483Y A SG11201609483Y A SG 11201609483YA
Authority
SG
Singapore
Prior art keywords
producing
same
pyridine derivative
novel crystalline
crystalline polymorphs
Prior art date
Application number
SG11201609483YA
Inventor
Hidetoshi Miyamoto
Hisae Nozato
Akinobu Maruyama
Original Assignee
Teijin Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teijin Pharma Ltd filed Critical Teijin Pharma Ltd
Publication of SG11201609483YA publication Critical patent/SG11201609483YA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/06Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs
SG11201609483YA 2014-05-13 2015-05-12 Novel crystalline polymorphs of pyridine derivative and method for producing the same SG11201609483YA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2014099678 2014-05-13
PCT/JP2015/063632 WO2015174411A1 (en) 2014-05-13 2015-05-12 Novel crystalline polymorph of pyridine derivative, and method for producing same

Publications (1)

Publication Number Publication Date
SG11201609483YA true SG11201609483YA (en) 2016-12-29

Family

ID=54479948

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201609483YA SG11201609483YA (en) 2014-05-13 2015-05-12 Novel crystalline polymorphs of pyridine derivative and method for producing the same

Country Status (15)

Country Link
US (1) US20170144987A1 (en)
EP (1) EP3144304A4 (en)
JP (1) JP6289619B2 (en)
KR (1) KR20170003569A (en)
CN (1) CN106458970B (en)
AR (1) AR100404A1 (en)
AU (1) AU2015260294A1 (en)
CA (1) CA2948792A1 (en)
IL (1) IL248901A0 (en)
MX (1) MX2016014692A (en)
PH (1) PH12016502222A1 (en)
RU (1) RU2016148736A (en)
SG (1) SG11201609483YA (en)
TW (1) TW201625580A (en)
WO (1) WO2015174411A1 (en)

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE122008000051I1 (en) * 1990-11-30 2009-02-05 Teijin Ltd 2-ARYLTHIAZOL DERIVATIVE AND MEDICAMENT CONTAINING THEREOF
US8148542B2 (en) * 2006-06-23 2012-04-03 Teijin Pharma Limited Method for producing crystal polymorphs of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazolecarboxylic acid
TWI613203B (en) * 2008-03-31 2018-02-01 C&C新藥研究所 Heterocyclic derivatives
CN102333765B (en) * 2009-02-27 2015-01-14 帝人制药株式会社 Process for producing phenyl-substituted heterocyclic derivative through coupling using transition metal catalyst
JP5519201B2 (en) * 2009-07-15 2014-06-11 光孝 北村 Process for producing crystalline polymorph of 2- (3-cyano-4-isobutyloxyphenyl) -4-methyl-5-thiazolecarboxylic acid
BRPI1011671A2 (en) * 2009-07-15 2016-03-22 Teijin Pharma Ltd process for producing 2- (3-cyano-4-isobutyloxyphenyl) -4-methyl-5-thiazolacarbocyclic acid form crystals
PL2610248T3 (en) * 2010-08-27 2016-12-30 Method for producing phenyl-substituted heterocyclic derivative by means of coupling method using a palladium compound
UA117359C2 (en) * 2012-11-14 2018-07-25 Тейдзін Фарма Лімітед Pyridine derivative

Also Published As

Publication number Publication date
RU2016148736A3 (en) 2018-06-14
US20170144987A1 (en) 2017-05-25
KR20170003569A (en) 2017-01-09
EP3144304A4 (en) 2017-10-25
JPWO2015174411A1 (en) 2017-04-20
PH12016502222A1 (en) 2017-02-06
MX2016014692A (en) 2017-02-23
RU2016148736A (en) 2018-06-14
AR100404A1 (en) 2016-10-05
WO2015174411A1 (en) 2015-11-19
AU2015260294A1 (en) 2017-01-05
CA2948792A1 (en) 2015-11-19
TW201625580A (en) 2016-07-16
EP3144304A1 (en) 2017-03-22
JP6289619B2 (en) 2018-03-07
CN106458970A (en) 2017-02-22
CN106458970B (en) 2019-09-13
IL248901A0 (en) 2017-01-31

Similar Documents

Publication Publication Date Title
EP3159339A4 (en) Method for producing pyridine compound
IL249988A0 (en) Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine
PL3174891T3 (en) Crystalline form of nicotinamide riboside
IL250628A0 (en) Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine
ZA201700243B (en) Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine
IL289910B1 (en) Method for producing allulose crystals
IL250984A0 (en) Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine
ZA201700168B (en) Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine
PT3323628T (en) Method for producing decorative panels
PT3152177T (en) Method for expanding sand-grain-shaped raw material
HK1256031A1 (en) Method for producing novel 4-benzazonine derivative
EP3190087A4 (en) Method for producing crystalline silicotitanate
EP3118194A4 (en) Method for producing 2-acyliminopyridine derivative
PL3190115T3 (en) Salt of cephalosporin derivative, crystalline solid form of same and method for producing same
HK1249518A1 (en) Process of synthesizing substituted pyridine and pyrimidine compound
EP3181545A4 (en) Method for producing triphenylbutene derivative
SG11201609483YA (en) Novel crystalline polymorphs of pyridine derivative and method for producing the same
GB201619463D0 (en) Method for producing allulose crystals
IL246920A0 (en) Method for producing purified compound
HK1208220A1 (en) Synthesis method of 9-allylcamptothecin derivatives 9-
EP3190105A4 (en) Crystalline anti-trichophyton drug and method for producing same
EP3130581A4 (en) Method for producing heterocyclic compound
EP3144305A4 (en) Method for producing 2-pyridone compound