SG10201909796PA - Chemosensory receptor ligand-based therapies - Google Patents

Chemosensory receptor ligand-based therapies

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Publication number
SG10201909796PA
SG10201909796PA SG10201909796PA SG10201909796PA SG 10201909796P A SG10201909796P A SG 10201909796PA SG 10201909796P A SG10201909796P A SG 10201909796PA SG 10201909796P A SG10201909796P A SG 10201909796PA
Authority
SG
Singapore
Prior art keywords
chemosensory receptor
receptor ligand
based therapies
methods
chemosensory
Prior art date
Application number
Inventor
Alain Baron
Martin R Brown
Christopher R G Jones
Original Assignee
Elcelyx Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Elcelyx Therapeutics Inc filed Critical Elcelyx Therapeutics Inc
Publication of SG10201909796PA publication Critical patent/SG10201909796PA/en

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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
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    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
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    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
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    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

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  • Health & Medical Sciences (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Zoology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Emergency Medicine (AREA)
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  • Nutrition Science (AREA)
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  • Gynecology & Obstetrics (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Physiology (AREA)

Abstract

Chemosensory Receptor Ligand-Based Therapies Provided herein are methods for treating diabetes, obesity, and other metabolic diseases, disorders or conditions comprising chemosensory receptor ligands. Also provided herein are chemosensory receptor ligand compositions and the preparation thereof for the methods of the present invention. No fig.
SG10201909796P 2010-04-20 2010-10-19 Chemosensory receptor ligand-based therapies SG10201909796PA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12/763,926 US9901551B2 (en) 2009-04-20 2010-04-20 Chemosensory receptor ligand-based therapies

Publications (1)

Publication Number Publication Date
SG10201909796PA true SG10201909796PA (en) 2019-11-28

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ID=44834962

Family Applications (3)

Application Number Title Priority Date Filing Date
SG10201909796P SG10201909796PA (en) 2010-04-20 2010-10-19 Chemosensory receptor ligand-based therapies
SG10201503098PA SG10201503098PA (en) 2010-04-20 2010-10-19 Chemosensory receptor ligand-based therapies
SG2012077558A SG184935A1 (en) 2010-04-20 2010-10-19 Chemosensory receptor ligand-based therapies

Family Applications After (2)

Application Number Title Priority Date Filing Date
SG10201503098PA SG10201503098PA (en) 2010-04-20 2010-10-19 Chemosensory receptor ligand-based therapies
SG2012077558A SG184935A1 (en) 2010-04-20 2010-10-19 Chemosensory receptor ligand-based therapies

Country Status (14)

Country Link
US (1) US9901551B2 (en)
EP (1) EP2560660A4 (en)
JP (1) JP5907952B2 (en)
KR (1) KR101881608B1 (en)
CN (2) CN106039313A (en)
AR (1) AR078678A1 (en)
BR (1) BR112012026838A2 (en)
CA (1) CA2800470A1 (en)
EA (1) EA201270767A1 (en)
IL (1) IL222586A0 (en)
MX (1) MX2012012157A (en)
SG (3) SG10201909796PA (en)
WO (1) WO2011133180A1 (en)
ZA (1) ZA201208277B (en)

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