SG10201707432SA - Syk inhibitors - Google Patents

Syk inhibitors

Info

Publication number
SG10201707432SA
SG10201707432SA SG10201707432SA SG10201707432SA SG10201707432SA SG 10201707432S A SG10201707432S A SG 10201707432SA SG 10201707432S A SG10201707432S A SG 10201707432SA SG 10201707432S A SG10201707432S A SG 10201707432SA SG 10201707432S A SG10201707432S A SG 10201707432SA
Authority
SG
Singapore
Prior art keywords
syk inhibitors
syk
inhibitors
Prior art date
Application number
SG10201707432SA
Inventor
Peter A Blomgren
Kevin S Currie
Jeffrey E Kropf
Seung H Lee
Jennifer R Lo
Scott A Mitchell
Aaron C Schmitt
Jin-Ming Xiong
Jianjun Xu
Zhongdong Zhao
Sundaramoorthi Swaminathan
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52350364&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG10201707432S(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of SG10201707432SA publication Critical patent/SG10201707432SA/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
SG10201707432SA 2013-12-23 2014-12-22 Syk inhibitors SG10201707432SA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201361920407P 2013-12-23 2013-12-23

Publications (1)

Publication Number Publication Date
SG10201707432SA true SG10201707432SA (en) 2017-10-30

Family

ID=52350364

Family Applications (3)

Application Number Title Priority Date Filing Date
SG10201707432SA SG10201707432SA (en) 2013-12-23 2014-12-22 Syk inhibitors
SG10201912586UA SG10201912586UA (en) 2013-12-23 2014-12-22 Syk inhibitors
SG11201604491VA SG11201604491VA (en) 2013-12-23 2014-12-22 Syk inhibitors

Family Applications After (2)

Application Number Title Priority Date Filing Date
SG10201912586UA SG10201912586UA (en) 2013-12-23 2014-12-22 Syk inhibitors
SG11201604491VA SG11201604491VA (en) 2013-12-23 2014-12-22 Syk inhibitors

Country Status (42)

Country Link
US (5) US9968601B2 (en)
EP (2) EP3342773B9 (en)
JP (3) JP6243062B2 (en)
KR (3) KR101925859B1 (en)
CN (2) CN107746405B (en)
AP (1) AP2016009274A0 (en)
AR (1) AR098912A1 (en)
AU (3) AU2014370010B2 (en)
BR (1) BR112016014643B1 (en)
CA (1) CA2875877C (en)
CL (1) CL2016001537A1 (en)
CR (1) CR20160287A (en)
CU (1) CU20160097A7 (en)
CY (1) CY1120104T1 (en)
DK (2) DK3087075T3 (en)
DO (1) DOP2016000140A (en)
EA (2) EA201891553A1 (en)
ES (2) ES2851335T3 (en)
GT (1) GT201600123A (en)
HK (2) HK1251563A1 (en)
HR (2) HRP20180460T1 (en)
HU (2) HUE037662T2 (en)
IL (1) IL245846B (en)
LT (1) LT3087075T (en)
MD (1) MD4666C1 (en)
ME (1) ME03001B (en)
MX (2) MX371024B (en)
NO (1) NO3183247T3 (en)
NZ (1) NZ721175A (en)
PE (1) PE20160995A1 (en)
PH (1) PH12016501204A1 (en)
PL (2) PL3087075T3 (en)
PT (2) PT3087075T (en)
RS (1) RS57182B1 (en)
SG (3) SG10201707432SA (en)
SI (2) SI3087075T1 (en)
SV (1) SV2016005229A (en)
TW (2) TWI662037B (en)
UA (1) UA118463C2 (en)
UY (1) UY35898A (en)
WO (1) WO2015100217A1 (en)
ZA (1) ZA201800913B (en)

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UY35898A (en) 2013-12-23 2015-07-31 Gilead Sciences Inc ? SYK INHIBITING COMPOUNDS AND COMPOSITIONS THAT UNDERSTAND THEM ?.
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TW201617074A (en) * 2014-07-14 2016-05-16 吉李德科學股份有限公司 Syk inhibitors
JP2018513173A (en) * 2015-04-21 2018-05-24 ギリアード サイエンシーズ， インコーポレイテッド Treatment of chronic graft-versus-host disease with SYK inhibitors
US20170173034A1 (en) * 2015-12-17 2017-06-22 Gilead Sciences, Inc. Combination of a jak inhibitor and a syk inhibitor for treating cancers and inflammatory disorders
TW201822764A (en) * 2016-09-14 2018-07-01 美商基利科學股份有限公司 Syk inhibitors
AU2017325844A1 (en) * 2016-09-14 2019-03-07 Gilead Sciences, Inc. SYK inhibitors
JOP20180040A1 (en) 2017-04-20 2019-01-30 Gilead Sciences Inc Pd-1/pd-l1 inhibitors
KR102399996B1 (en) 2017-08-25 2022-05-20 길리애드 사이언시즈, 인코포레이티드 Polymorphs of SYK Inhibitors
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