SG10201605196PA - Novel Inhibitor Compounds Of Phosphodiesterase Type 10A - Google Patents
Novel Inhibitor Compounds Of Phosphodiesterase Type 10AInfo
- Publication number
- SG10201605196PA SG10201605196PA SG10201605196PA SG10201605196PA SG10201605196PA SG 10201605196P A SG10201605196P A SG 10201605196PA SG 10201605196P A SG10201605196P A SG 10201605196PA SG 10201605196P A SG10201605196P A SG 10201605196PA SG 10201605196P A SG10201605196P A SG 10201605196PA
- Authority
- SG
- Singapore
- Prior art keywords
- inhibitor compounds
- phosphodiesterase type
- novel inhibitor
- novel
- phosphodiesterase
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems
- C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161503040P | 2011-06-30 | 2011-06-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG10201605196PA true SG10201605196PA (en) | 2016-08-30 |
Family
ID=46456562
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG10201605196PA SG10201605196PA (en) | 2011-06-30 | 2012-06-28 | Novel Inhibitor Compounds Of Phosphodiesterase Type 10A |
Country Status (24)
| Country | Link |
|---|---|
| US (2) | US9938269B2 (en) |
| EP (1) | EP2726479A1 (en) |
| JP (1) | JP2014518237A (en) |
| KR (1) | KR20140050028A (en) |
| CN (1) | CN103958504B (en) |
| AR (1) | AR086817A1 (en) |
| AU (1) | AU2012277802A1 (en) |
| BR (1) | BR112013033696A2 (en) |
| CA (1) | CA2839655A1 (en) |
| CL (1) | CL2013003731A1 (en) |
| CO (1) | CO6870032A2 (en) |
| CR (1) | CR20140023A (en) |
| DO (1) | DOP2013000315A (en) |
| EC (1) | ECSP14013188A (en) |
| GT (1) | GT201300324A (en) |
| MX (1) | MX2013015390A (en) |
| NZ (1) | NZ618930A (en) |
| PE (1) | PE20141308A1 (en) |
| RU (1) | RU2014102962A (en) |
| SG (1) | SG10201605196PA (en) |
| TW (1) | TW201311662A (en) |
| UY (1) | UY34177A (en) |
| WO (1) | WO2013000994A1 (en) |
| ZA (1) | ZA201309561B (en) |
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| US9200005B2 (en) | 2013-03-13 | 2015-12-01 | AbbVie Deutschland GmbH & Co. KG | Inhibitor compounds of phosphodiesterase type 10A |
| MX2015012008A (en) | 2013-03-14 | 2016-04-15 | Abbvie Deutschland | Novel inhibitor compounds of phosphodiesterase type 10a. |
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| MX2016009448A (en) | 2014-01-31 | 2016-10-13 | Hoffmann La Roche | (hetero)aryl imidazoles/pyrazoles for treatment of neurological disorders. |
| WO2015116904A1 (en) | 2014-02-03 | 2015-08-06 | Vitae Pharmaceuticals, Inc. | Dihydropyrrolopyridine inhibitors of ror-gamma |
| CA2943882A1 (en) * | 2014-05-22 | 2015-11-26 | F. Hoffmann-La Roche Ag | Indolin-2-one and 1,3-dihydro-pyrrolo[3,2-c]pyridin-2-one derivatives |
| TWI713455B (en) | 2014-06-25 | 2020-12-21 | 美商伊凡克特治療公司 | Mnk inhibitors and methods related thereto |
| WO2016061160A1 (en) | 2014-10-14 | 2016-04-21 | Vitae Pharmaceuticals, Inc. | Dihydropyrrolopyridine inhibitors of ror-gamma |
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-
2012
- 2012-06-27 US US13/534,127 patent/US9938269B2/en active Active
- 2012-06-28 BR BR112013033696A patent/BR112013033696A2/en not_active IP Right Cessation
- 2012-06-28 KR KR1020147002761A patent/KR20140050028A/en not_active Application Discontinuation
- 2012-06-28 CN CN201280042318.5A patent/CN103958504B/en not_active Expired - Fee Related
- 2012-06-28 JP JP2014517695A patent/JP2014518237A/en active Pending
- 2012-06-28 WO PCT/EP2012/062544 patent/WO2013000994A1/en active Application Filing
- 2012-06-28 PE PE2013002907A patent/PE20141308A1/en not_active Application Discontinuation
- 2012-06-28 EP EP12731416.9A patent/EP2726479A1/en active Pending
- 2012-06-28 SG SG10201605196PA patent/SG10201605196PA/en unknown
- 2012-06-28 CA CA2839655A patent/CA2839655A1/en not_active Abandoned
- 2012-06-28 NZ NZ618930A patent/NZ618930A/en not_active IP Right Cessation
- 2012-06-28 RU RU2014102962/04A patent/RU2014102962A/en not_active Application Discontinuation
- 2012-06-28 AU AU2012277802A patent/AU2012277802A1/en not_active Abandoned
- 2012-06-28 MX MX2013015390A patent/MX2013015390A/en unknown
- 2012-06-29 AR ARP120102358A patent/AR086817A1/en unknown
- 2012-06-29 UY UY0001034177A patent/UY34177A/en not_active Application Discontinuation
- 2012-06-29 TW TW101123611A patent/TW201311662A/en unknown
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2013
- 2013-12-18 ZA ZA2013/09561A patent/ZA201309561B/en unknown
- 2013-12-26 CL CL2013003731A patent/CL2013003731A1/en unknown
- 2013-12-26 GT GT201300324A patent/GT201300324A/en unknown
- 2013-12-27 DO DO2013000315A patent/DOP2013000315A/en unknown
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2014
- 2014-01-16 CR CR20140023A patent/CR20140023A/en unknown
- 2014-01-27 CO CO14015863A patent/CO6870032A2/en unknown
- 2014-01-30 EC ECSP14013188 patent/ECSP14013188A/en unknown
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2018
- 2018-04-09 US US15/948,299 patent/US20180222905A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20130005705A1 (en) | 2013-01-03 |
| CA2839655A1 (en) | 2013-01-03 |
| AU2012277802A1 (en) | 2014-01-09 |
| EP2726479A1 (en) | 2014-05-07 |
| UY34177A (en) | 2013-01-31 |
| CR20140023A (en) | 2014-08-21 |
| KR20140050028A (en) | 2014-04-28 |
| RU2014102962A (en) | 2015-08-10 |
| WO2013000994A1 (en) | 2013-01-03 |
| ECSP14013188A (en) | 2014-12-30 |
| CL2013003731A1 (en) | 2014-10-10 |
| CO6870032A2 (en) | 2014-02-20 |
| US20180222905A1 (en) | 2018-08-09 |
| CN103958504A (en) | 2014-07-30 |
| CN103958504B (en) | 2016-10-12 |
| BR112013033696A2 (en) | 2016-08-30 |
| DOP2013000315A (en) | 2014-04-15 |
| GT201300324A (en) | 2014-09-26 |
| MX2013015390A (en) | 2014-07-14 |
| US9938269B2 (en) | 2018-04-10 |
| ZA201309561B (en) | 2014-08-27 |
| NZ618930A (en) | 2015-05-29 |
| TW201311662A (en) | 2013-03-16 |
| AR086817A1 (en) | 2014-01-22 |
| JP2014518237A (en) | 2014-07-28 |
| AU2012277802A8 (en) | 2014-03-06 |
| PE20141308A1 (en) | 2014-10-26 |
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