SE7908629L - A NEW PROCEDURE FOR THE PREPARATION OF 6-PIPERIDINO-2,4-DIAMINOPYRIMIDIN-3-OXIDE - Google Patents

A NEW PROCEDURE FOR THE PREPARATION OF 6-PIPERIDINO-2,4-DIAMINOPYRIMIDIN-3-OXIDE

Info

Publication number
SE7908629L
SE7908629L SE7908629A SE7908629A SE7908629L SE 7908629 L SE7908629 L SE 7908629L SE 7908629 A SE7908629 A SE 7908629A SE 7908629 A SE7908629 A SE 7908629A SE 7908629 L SE7908629 L SE 7908629L
Authority
SE
Sweden
Prior art keywords
diaminopyrimidin
piperidino
oxide
preparation
new procedure
Prior art date
Application number
SE7908629A
Other languages
Swedish (sv)
Other versions
SE432596B (en
Inventor
A Vedres
C Szantay
G Balogh
J Horvath
T Mester
Original Assignee
Egyt Gyogyszervegyeszeti Gyar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar
Publication of SE7908629L publication Critical patent/SE7908629L/en
Publication of SE432596B publication Critical patent/SE432596B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50Three nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52Two oxygen atoms
SE7908629A 1978-10-27 1979-10-17 PROCEDURE FOR PREPARING 6-PIPERIDINO-2,4-DIAMINOPYRIMIDINE-3-OXIDE SE432596B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU78EE2594A HU177601B (en) 1978-10-27 1978-10-27 New process for preparing 6-piperidino-2,4-diamino-pyrimidine-3-oxide

Publications (2)

Publication Number Publication Date
SE7908629L true SE7908629L (en) 1980-04-28
SE432596B SE432596B (en) 1984-04-09

Family

ID=10995794

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7908629A SE432596B (en) 1978-10-27 1979-10-17 PROCEDURE FOR PREPARING 6-PIPERIDINO-2,4-DIAMINOPYRIMIDINE-3-OXIDE

Country Status (14)

Country Link
JP (1) JPS5559172A (en)
AT (1) AT373246B (en)
CH (1) CH642365A5 (en)
CS (1) CS213398B2 (en)
DE (1) DE2943161A1 (en)
DK (1) DK454579A (en)
ES (1) ES485457A1 (en)
FI (1) FI793307A (en)
GB (1) GB2032434B (en)
HU (1) HU177601B (en)
PL (1) PL119712B1 (en)
SE (1) SE432596B (en)
SU (1) SU913942A3 (en)
YU (1) YU262579A (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1179344A (en) * 1981-07-15 1984-12-11 Jean-Claude Muller Process for the preparation of 6-¬3,6-dihydro-1(2h)- pyridyl| pyrimidine-3-oxides
CH649291A5 (en) * 1982-03-16 1985-05-15 Hoffmann La Roche DICARBAMATE.
HU196061B (en) * 1986-07-10 1988-09-28 Richter Gedeon Vegyeszet Process for production of pirimidine-derivatives
HU196067B (en) * 1986-07-10 1988-09-28 Richter Gedeon Vegyeszet Process for production of 6-amin-1,2-dihydro-1-hydroxi-2-imino-4-piperidin-piramidin
FI864046A (en) * 1986-10-07 1988-04-08 Farmos Oy FOERFARANDE FOER FRAMSTAELLNING AV EN TERAPEUTISKT AKTIV FOERENING.
LU86958A1 (en) * 1987-07-31 1989-03-08 Oreal SALTS OF THIAMORPHOLINONE CARBOXYLIC ACID AND 2,4-DIAMINO PYRIMIDINE DERIVATIVES, THEIR USE IN COSMETICS AND PHARMACY
LU86960A1 (en) * 1987-07-31 1989-03-08 Oreal PROCESS FOR THE PREPARATION OF PIPERIDINO-6 DIAMINO-2,4 PYRIMIDINE OXIDE-3 AND NEW COMPOUNDS
JPH02225474A (en) * 1989-01-04 1990-09-07 Lonza Ag Preparation of 2,4-diamino-6-piperidinyl-pyrimidine- 3-n-oxide

Also Published As

Publication number Publication date
YU262579A (en) 1983-01-21
CH642365A5 (en) 1984-04-13
HU177601B (en) 1981-11-28
JPS5559172A (en) 1980-05-02
GB2032434A (en) 1980-05-08
SU913942A3 (en) 1982-03-15
DE2943161A1 (en) 1980-05-08
DK454579A (en) 1980-04-28
PL219242A1 (en) 1980-06-16
CS213398B2 (en) 1982-04-09
AT373246B (en) 1983-12-27
PL119712B1 (en) 1982-01-30
ATA689879A (en) 1983-05-15
FI793307A (en) 1980-04-28
ES485457A1 (en) 1980-10-01
SE432596B (en) 1984-04-09
GB2032434B (en) 1982-11-17

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