SE380806B - PROCEDURE FOR MAKING NEW ESTRAS OF ALFA-AMINOPENICILLINS - Google Patents

PROCEDURE FOR MAKING NEW ESTRAS OF ALFA-AMINOPENICILLINS

Info

Publication number
SE380806B
SE380806B SE1572070A SE1572070A SE380806B SE 380806 B SE380806 B SE 380806B SE 1572070 A SE1572070 A SE 1572070A SE 1572070 A SE1572070 A SE 1572070A SE 380806 B SE380806 B SE 380806B
Authority
SE
Sweden
Prior art keywords
estras
aminopenicillins
alfa
procedure
making new
Prior art date
Application number
SE1572070A
Other languages
Swedish (sv)
Inventor
Bertil A Ekstroem
Berndt O Sjoeberg
Original Assignee
Astra Laekemedel Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Laekemedel Ab filed Critical Astra Laekemedel Ab
Priority to SE1572070A priority Critical patent/SE380806B/en
Priority to DE19712144457 priority patent/DE2144457C3/en
Priority to US178426A priority patent/US3873521A/en
Priority to FR7133107A priority patent/FR2106578B1/fr
Priority to AT795771A priority patent/AT309681B/en
Priority to AT537872A priority patent/AT311557B/en
Priority to SU1696133A priority patent/SU553936A3/en
Priority to IE1167/71A priority patent/IE35642B1/en
Priority to GB4309071A priority patent/GB1363506A/en
Priority to CA122,881A priority patent/CA960211A/en
Priority to IT28678/71A priority patent/IT1049876B/en
Priority to FI2580/71A priority patent/FI55203C/en
Priority to DK453871A priority patent/DK132759C/en
Priority to CH1362371A priority patent/CH583239A5/xx
Priority to CS71442A priority patent/CS187316B2/cs
Priority to NO3449/71A priority patent/NO140931C/en
Priority to CH859975A priority patent/CH577513A5/xx
Priority to ES195145A priority patent/ES395145A1/en
Priority to CH860075A priority patent/CH589654A5/xx
Priority to CS716617A priority patent/CS187312B2/en
Priority to BR6116/71A priority patent/BR7106116D0/en
Priority to HUAA684A priority patent/HU165868B/hu
Priority to JP7184971A priority patent/JPS5317597B1/ja
Priority to BE772723A priority patent/BE772723A/en
Priority to NL7112789.A priority patent/NL164860C/en
Priority to DD157795A priority patent/DD94815A5/xx
Priority to NO236/72A priority patent/NO140930C/en
Priority to AR241427A priority patent/AR201730A1/en
Priority to ES401745A priority patent/ES401745A1/en
Priority to US05/339,364 priority patent/US3939270A/en
Priority to SU731899287A priority patent/SU1153830A3/en
Priority to CA184,183A priority patent/CA1008447A/en
Priority to DK509774A priority patent/DK509774A/da
Priority to DK509674A priority patent/DK150200C/en
Priority to NO74744606A priority patent/NO142670C/en
Priority to FI3814/74A priority patent/FI59600C/en
Priority to ES433637A priority patent/ES433637A1/en
Priority to AR258235A priority patent/AR210991A1/en
Priority to JP7921675A priority patent/JPS5537996B2/ja
Priority to DK375975A priority patent/DK375975A/da
Publication of SE380806B publication Critical patent/SE380806B/en
Priority to CA240,891A priority patent/CA1008446A/en
Priority to CH493776A priority patent/CH613207A5/xx
Priority to CH1155377A priority patent/CH602745A5/xx
Priority to FI773032A priority patent/FI57951C/en
Priority to NL7801086A priority patent/NL7801086A/en
Priority to NO784144A priority patent/NO142671C/en
Priority to FI791386A priority patent/FI59103C/en
Priority to NLAANVRAGE8001563,A priority patent/NL171160C/en
Priority to DK133380A priority patent/DK150201C/en
Priority to DK163482A priority patent/DK158519C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04Preparation
    • C07D499/08Modification of a carboxyl radical directly attached in position 2, e.g. esterification

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
SE1572070A 1970-09-17 1970-11-20 PROCEDURE FOR MAKING NEW ESTRAS OF ALFA-AMINOPENICILLINS SE380806B (en)

Priority Applications (50)

Application Number Priority Date Filing Date Title
SE1572070A SE380806B (en) 1970-11-20 1970-11-20 PROCEDURE FOR MAKING NEW ESTRAS OF ALFA-AMINOPENICILLINS
DE19712144457 DE2144457C3 (en) 1970-09-17 1971-09-04 α-Aminobenzylpenicillin esters, processes for their preparation and pharmaceuticals containing them
US178426A US3873521A (en) 1970-09-17 1971-09-07 Esters of {60 -amino penicillins
FR7133107A FR2106578B1 (en) 1970-09-17 1971-09-14
AT795771A AT309681B (en) 1970-09-17 1971-09-14 Process for the production of new α-aminopenicillins
AT537872A AT311557B (en) 1970-09-17 1971-09-14 Process for the production of new α-aminopenicillins
SU1696133A SU553936A3 (en) 1970-09-17 1971-09-14 Method for producing β-aminopenicillin esters
IE1167/71A IE35642B1 (en) 1970-09-17 1971-09-15 A process for the preparation of new alpha-aminopenicillins and such penicillins and intermediates and pharmaceutical preparations
GB4309071A GB1363506A (en) 1970-09-17 1971-09-15 Process for the preparation of alpha-amino-penicillins and such penicillins and intermediates and pharmaceutical preparations
CA122,881A CA960211A (en) 1970-09-17 1971-09-15 PROCESS FOR THE PREPARATION OF NEW .alpha.-AMINOPENICILLINS AND SUCH PENICILLINS, AND INTERMEDIATES AND PHARMACEUTICAL PREPARATIONS
IT28678/71A IT1049876B (en) 1970-09-17 1971-09-15 PROCEDURE FOR THE PREPARATION OF ALPHA AMINOPENICILLINS PEN ICILLINS THUS PREPARED INTERMEDIATE AND PHARMACEUTICAL PREPARATIONS
FI2580/71A FI55203C (en) 1970-09-17 1971-09-15 ANALOG FOUNDATION FRAMSTAELLNING AV ESTRAR AV ALFA-AMINOPENICILLINER
DK453871A DK132759C (en) 1970-09-17 1971-09-16 ANALOGICAL PROCEDURE FOR THE PREPARATION OF ALFA AMINOPENICILLINESTERS OR ACID ADDITIONAL SALTS THEREOF OR THE CORRESPONDING OPTICAL ANTIPODES
CH1362371A CH583239A5 (en) 1970-09-17 1971-09-16
CS71442A CS187316B2 (en) 1970-09-17 1971-09-16
NO3449/71A NO140931C (en) 1970-09-17 1971-09-16 ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE ESTERS OF ALFA-AMINOBENZYLPENICILLINES
CH859975A CH577513A5 (en) 1970-09-17 1971-09-16
ES195145A ES395145A1 (en) 1970-09-17 1971-09-16 Esters of {60 -amino penicillins
CH860075A CH589654A5 (en) 1970-09-17 1971-09-16
CS716617A CS187312B2 (en) 1970-09-17 1971-09-16 Method of producing novel esters of alpha-aminopenicillins
BR6116/71A BR7106116D0 (en) 1970-09-17 1971-09-16 ALPHA-AMINO-PENICILLIN COMPOUNDS PROCESS OF CHEMICAL INTERMEDIATE PREPARATION PHARMACEUTICAL PREPARATIONS AND PROCESS FOR THE TREATMENT OF INFECTIOUS DISEASES
HUAA684A HU165868B (en) 1970-09-17 1971-09-16
JP7184971A JPS5317597B1 (en) 1970-09-17 1971-09-17
BE772723A BE772723A (en) 1970-09-17 1971-09-17 PROCESS FOR THE PREPARATION OF NEW ALPHA-AMINOPENICILLINS, PENICILLINS THUS OBTAINED AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
NL7112789.A NL164860C (en) 1970-09-17 1971-09-17 METHOD FOR PREPARING A MEDICINAL PRODUCT WITH ANTIBIOTIC ACTION AND METHOD FOR PREPARING A SUBSTITUTED HYDROXYALKYL ESTER OF AN ALFA-AMINOARALKYLPENICILLIN
DD157795A DD94815A5 (en) 1970-09-17 1971-09-17
NO236/72A NO140930C (en) 1970-09-17 1972-01-31 6-AMINOPENICILLANIC RESIDUES FOR USE AS A STARTING MATERIAL FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE ESTERS OF ALFA-AMINOBENZYLPENICILLINS
AR241427A AR201730A1 (en) 1970-09-17 1972-04-12 PROCEDURE FOR THE PREPARATION OF NEW ALPHAAMINOPENICILLIN ESTERS
ES401745A ES401745A1 (en) 1970-09-17 1972-04-14 Esters of {60 -amino penicillins
US05/339,364 US3939270A (en) 1970-09-17 1973-03-08 Pharmaceutical preparations containing α-aminopenicillins
SU731899287A SU1153830A3 (en) 1970-09-17 1973-03-27 Method of obtaining esters of alpha-aminopenicillins or their acid-additive salts
CA184,183A CA1008447A (en) 1970-09-17 1973-10-25 INTERMEDIATES FOR THE PREPARATION OF NEW .alpha.-AMINOPENICILLINS
DK509774A DK509774A (en) 1970-09-17 1974-09-27
DK509674A DK150200C (en) 1970-09-17 1974-09-27 6-AMINOPENICILLANIC ACID ESTES USED FOR PREPARING AN N-ACYL DERIVATIVE OF A 6-AMINOPENICILLANIC ACID ESTER
NO74744606A NO142670C (en) 1970-09-17 1974-12-19 BENZYLPENICILLINESTERS FOR USE AS BASIC MATERIAL IN THE PREPARATION OF A THERAPEUTIC ACTIVE ESTER OF ALFA-AMINOBENZYLPENICILLINES
FI3814/74A FI59600C (en) 1970-09-17 1974-12-31 MELLAN PRODUCTS FOR FRAMSTAELLNING AV ALFA-AMINOPENICILLINESTRAR
ES433637A ES433637A1 (en) 1970-09-17 1975-01-08 Esters of {60 -amino penicillins
AR258235A AR210991A1 (en) 1970-09-17 1975-04-08 1-ETOXICARBONYLOXYETHYL BENZYLPENICILANATE FOR ITS EXCLUSIVE USE AS AN INTERMEDIARY.
JP7921675A JPS5537996B2 (en) 1970-09-17 1975-06-24
DK375975A DK375975A (en) 1970-09-17 1975-08-20
CA240,891A CA1008446A (en) 1970-09-17 1975-12-02 INTERMEDIATES FOR THE PREPARATION OF NEW .alpha.-AMINOPENICILLINS
CH493776A CH613207A5 (en) 1970-09-17 1976-04-20
CH1155377A CH602745A5 (en) 1970-09-17 1977-09-21
FI773032A FI57951C (en) 1970-09-17 1977-10-13 MELLANPRODUKTER TILL ANVAENDNING VID FRAMSTAELLNING AV ESTRAR AV ALFA-AMINOPENICILLINER
NL7801086A NL7801086A (en) 1970-09-17 1978-01-31 PROCESS FOR PREPARING THE ETHOXYCARBONYLOXYETHYL ESTER OF BENZYL PENICILLIN AND THE ACID ADDITIONAL SALTS AND OPTICAL ISOMERS DERIVED FROM IT.
NO784144A NO142671C (en) 1970-09-17 1978-12-08 ALFA-AZIDOBENZYLPENICILLIN ESTERS FOR USE IN THE PREPARATION OF THERAPEUTIC EFFECTIVE ALFA-AMINOBENZYLPENICILLIN ESTERS
FI791386A FI59103C (en) 1970-09-17 1979-04-27 MELLANPRODUKTER TILL ANVAENDNING VID FRAMSTAELLNING AV ALFA-AMINOPENICILLINESTRAR
NLAANVRAGE8001563,A NL171160C (en) 1970-09-17 1980-03-17 METHOD FOR PREPARING OR MANUFACTURING A MEDICINAL PRODUCT WITH ANTIBIOTIC ACTION AND METHOD FOR PREPARING A SUBSTITUTED HYDROXYALKYL ESTER OF AN ALFA-AMINOARALKYLPENICILLIN
DK133380A DK150201C (en) 1970-09-17 1980-03-27 ALFA-AZIDO-N-ACYL-6-AMINOPENICILLANIC ACID ESTABLES USED FOR PREPARING THE SIMILAR ALFA-AMINO COMPOUND
DK163482A DK158519C (en) 1970-09-17 1982-04-07 BENZYLPENICILLIN DERIVATIVES USED AS THE BASIC MATERIAL OF THE PROCESS FOR THE PREPARATION OF ALFA-AMINOPENICILLIN ESTERS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE1572070A SE380806B (en) 1970-11-20 1970-11-20 PROCEDURE FOR MAKING NEW ESTRAS OF ALFA-AMINOPENICILLINS

Publications (1)

Publication Number Publication Date
SE380806B true SE380806B (en) 1975-11-17

Family

ID=20301115

Family Applications (1)

Application Number Title Priority Date Filing Date
SE1572070A SE380806B (en) 1970-09-17 1970-11-20 PROCEDURE FOR MAKING NEW ESTRAS OF ALFA-AMINOPENICILLINS

Country Status (1)

Country Link
SE (1) SE380806B (en)

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