SE0401464D0 - New disubstituted phenylpiperidines / piperazines as modulators of dopamine neurotransmission - Google Patents

New disubstituted phenylpiperidines / piperazines as modulators of dopamine neurotransmission

Info

Publication number
SE0401464D0
SE0401464D0 SE0401464A SE0401464A SE0401464D0 SE 0401464 D0 SE0401464 D0 SE 0401464D0 SE 0401464 A SE0401464 A SE 0401464A SE 0401464 A SE0401464 A SE 0401464A SE 0401464 D0 SE0401464 D0 SE 0401464D0
Authority
SE
Sweden
Prior art keywords
piperazines
modulators
dopamine neurotransmission
phenylpiperidines
new disubstituted
Prior art date
Application number
SE0401464A
Other languages
Swedish (sv)
Inventor
Clas Sonesson
Lars Swanson
Nicholas Waters
Original Assignee
Carlsson A Research Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Carlsson A Research Ab filed Critical Carlsson A Research Ab
Priority to SE0401464A priority Critical patent/SE0401464D0/en
Publication of SE0401464D0 publication Critical patent/SE0401464D0/en
Priority to KR1020077000513A priority patent/KR101245075B1/en
Priority to ZA200807949A priority patent/ZA200807949B/en
Priority to DK05760618.8T priority patent/DK1773772T3/en
Priority to CN200580023206.5A priority patent/CN1997630B/en
Priority to DE602005017784T priority patent/DE602005017784D1/en
Priority to UAA200700155A priority patent/UA87853C2/en
Priority to RU2006147243/04A priority patent/RU2366654C2/en
Priority to AU2005251906A priority patent/AU2005251906B2/en
Priority to MXPA06013941A priority patent/MXPA06013941A/en
Priority to NZ552409A priority patent/NZ552409A/en
Priority to ES05760618T priority patent/ES2346452T3/en
Priority to BRPI0511907A priority patent/BRPI0511907A8/en
Priority to CN 200580023251 priority patent/CN1997631A/en
Priority to JP2007526287A priority patent/JP4937124B2/en
Priority to JP2007526289A priority patent/JP2008501749A/en
Priority to NZ552411A priority patent/NZ552411A/en
Priority to EP10155758A priority patent/EP2204363A1/en
Priority to CA2569840A priority patent/CA2569840C/en
Priority to DE602005021641T priority patent/DE602005021641D1/en
Priority to AU2005251909A priority patent/AU2005251909A1/en
Priority to AT05746589T priority patent/ATE449070T1/en
Priority to PCT/EP2005/006147 priority patent/WO2005121087A1/en
Priority to PCT/EP2005/006154 priority patent/WO2005121088A1/en
Priority to MXPA06013944A priority patent/MXPA06013944A/en
Priority to AT05760618T priority patent/ATE469885T1/en
Priority to PL05760618T priority patent/PL1773772T3/en
Priority to EP05760618A priority patent/EP1773772B1/en
Priority to EP05746589A priority patent/EP1768958B1/en
Priority to CA002569843A priority patent/CA2569843A1/en
Priority to PT05760618T priority patent/PT1773772E/en
Priority to IL179790A priority patent/IL179790A0/en
Priority to US11/567,925 priority patent/US7851629B2/en
Priority to US11/608,313 priority patent/US7763639B2/en
Priority to NO20070124A priority patent/NO20070124L/en
Priority to US12/814,827 priority patent/US8314126B2/en

Links

Abstract

The present invention relates to compounds which have therapeutic effects against disorders in the central nervous system, and in particular new 4-(ortho, meta-disubstituted phenyl)-1-alkypiperidines and piperazines. (I) wherein R1, R2, R3 and Y are as defined.
SE0401464A 2004-06-08 2004-06-08 New disubstituted phenylpiperidines / piperazines as modulators of dopamine neurotransmission SE0401464D0 (en)

Priority Applications (36)

Application Number Priority Date Filing Date Title
SE0401464A SE0401464D0 (en) 2004-06-08 2004-06-08 New disubstituted phenylpiperidines / piperazines as modulators of dopamine neurotransmission
EP10155758A EP2204363A1 (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
NZ552411A NZ552411A (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
CA2569840A CA2569840C (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
DK05760618.8T DK1773772T3 (en) 2004-06-08 2005-06-08 Novel disubstituted phenylpiperidines / piperazines as modulators of dopamine neurotransmission
ZA200807949A ZA200807949B (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
DE602005017784T DE602005017784D1 (en) 2004-06-08 2005-06-08 NEW DISUBSTITUTED PHENYLPIPERIDINES AS MODULATORS OF DOPAMINE AND SEROTONINE NEUROTRANSMISSION
DE602005021641T DE602005021641D1 (en) 2004-06-08 2005-06-08 NEW DISUBSTITUTED PHENYLPIPERIDINES AND PIPERAZINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION
RU2006147243/04A RU2366654C2 (en) 2004-06-08 2005-06-08 New disubstituted phenyl piperidines/piperazines as modulators of dopamine neurotransmission
AU2005251906A AU2005251906B2 (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
MXPA06013941A MXPA06013941A (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines as modulators of dopamine and serotonin neurotransmission.
NZ552409A NZ552409A (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines as modulators of dopamine and serotonin neurotransmission
ES05760618T ES2346452T3 (en) 2004-06-08 2005-06-08 NEW DISABLED PHENYLPIPERIDINS / PIPERAZINS USED AS MODULATORS OF THE DOPAMINE NEUROTRANSMISSION.
BRPI0511907A BRPI0511907A8 (en) 2004-06-08 2005-06-08 new disubstituted phenylpiperidine / piperazine derivatives as modulators of dopamine neurotransmission
CN 200580023251 CN1997631A (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines as modulators of dopamine and serotonin neurotransmission
JP2007526287A JP4937124B2 (en) 2004-06-08 2005-06-08 Newly provided phenylpiperidine / piperazine as modulators of dopamine neurotransmission
JP2007526289A JP2008501749A (en) 2004-06-08 2005-06-08 Novel disubstituted phenylpiperidines as modulators of dopamine and serotonin neurotransmission
KR1020077000513A KR101245075B1 (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
PT05760618T PT1773772E (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
CN200580023206.5A CN1997630B (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines as modulators of dopamine neurotransmission
UAA200700155A UA87853C2 (en) 2004-06-08 2005-06-08 Disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
AU2005251909A AU2005251909A1 (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines as modulators of dopamine and serotonin neurotransmission
AT05746589T ATE449070T1 (en) 2004-06-08 2005-06-08 NEW DISUBSTITUTED PHENYLPIPERIDINES AS MODULATORS OF DOPAMINE AND SEROTONINE NEUROTRANSMISSION
PCT/EP2005/006147 WO2005121087A1 (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
PCT/EP2005/006154 WO2005121088A1 (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines as modulators of dopamine and serotonin neurotransmission
MXPA06013944A MXPA06013944A (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission.
AT05760618T ATE469885T1 (en) 2004-06-08 2005-06-08 NEW DISUBSTITUTED PHENYLPIPERIDINE AND PIPERAZINE AS MODULATORS OF DOPAMINE NEUROTRANSMISSION
PL05760618T PL1773772T3 (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
EP05760618A EP1773772B1 (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
EP05746589A EP1768958B1 (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines as modulators of dopamine and serotonin neurotransmission
CA002569843A CA2569843A1 (en) 2004-06-08 2005-06-08 New disubstituted phenylpiperidines as modulators of dopamine and serotonin neurotransmission
IL179790A IL179790A0 (en) 2004-06-08 2006-12-03 New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
US11/567,925 US7851629B2 (en) 2004-06-08 2006-12-07 Disubstituted phenylpiperidines as modulators of dopamine and serotonin neurotransmission
US11/608,313 US7763639B2 (en) 2004-06-08 2006-12-08 Disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission
NO20070124A NO20070124L (en) 2004-06-08 2007-01-08 New disubstituted phenylpiperidines / piperazines as modulators of dopamine neurotransmission
US12/814,827 US8314126B2 (en) 2004-06-08 2010-06-14 Disubstituted phenylpiperdines/piperazines as modulators of dopamine neurotransmission

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0401464A SE0401464D0 (en) 2004-06-08 2004-06-08 New disubstituted phenylpiperidines / piperazines as modulators of dopamine neurotransmission

Publications (1)

Publication Number Publication Date
SE0401464D0 true SE0401464D0 (en) 2004-06-08

Family

ID=32653559

Family Applications (1)

Application Number Title Priority Date Filing Date
SE0401464A SE0401464D0 (en) 2004-06-08 2004-06-08 New disubstituted phenylpiperidines / piperazines as modulators of dopamine neurotransmission

Country Status (4)

Country Link
CN (2) CN1997630B (en)
SE (1) SE0401464D0 (en)
UA (1) UA87853C2 (en)
ZA (1) ZA200807949B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103382187B (en) * 2013-08-06 2015-06-03 信实生物医药(上海)有限公司 3-chloro-7(5)-bromo-benzo-isoxazole compounding method

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9904723D0 (en) * 1999-12-22 1999-12-22 Carlsson A Research Ab New modulators of dopamine neurotransmission II

Also Published As

Publication number Publication date
UA87853C2 (en) 2009-08-25
CN1997630B (en) 2013-01-30
CN1997631A (en) 2007-07-11
CN1997630A (en) 2007-07-11
ZA200807949B (en) 2010-02-24

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