SA515360233B1 - Inhibitors of histone demethylases - Google Patents

Inhibitors of histone demethylases

Info

Publication number
SA515360233B1
SA515360233B1 SA515360233A SA515360233A SA515360233B1 SA 515360233 B1 SA515360233 B1 SA 515360233B1 SA 515360233 A SA515360233 A SA 515360233A SA 515360233 A SA515360233 A SA 515360233A SA 515360233 B1 SA515360233 B1 SA 515360233B1
Authority
SA
Saudi Arabia
Prior art keywords
compounds
inhibitors
histone demethylases
present application
discloses
Prior art date
Application number
SA515360233A
Other languages
Arabic (ar)
Inventor
بويسين ثوماس
اولاه فارمان
خان قاسم
لابيل مارك
ميهروترا موكوند
Original Assignee
ابثيرابيوتيكس ايه بي اس
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2013/070457 external-priority patent/WO2014053491A1/en
Application filed by ابثيرابيوتيكس ايه بي اس filed Critical ابثيرابيوتيكس ايه بي اس
Publication of SA515360233B1 publication Critical patent/SA515360233B1/en

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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The present application discloses compounds capable of modulating the activity of histone demethylases (HDMEs), which are useful for prevention and/or treatment of diseases in which genomic dysregulation is involved in the pathogenesis, such as e.g. cancer. The present application also discloses pharmaceutical compositions comprising said compounds and the use of such compounds as a medicament. The compounds take the form (I). (I)
SA515360233A 2012-10-02 2015-04-02 Inhibitors of histone demethylases SA515360233B1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261708806P 2012-10-02 2012-10-02
DKPA201200599 2012-10-02
US201361770050P 2013-02-27 2013-02-27
DKPA201370112 2013-02-27
PCT/EP2013/070457 WO2014053491A1 (en) 2012-10-02 2013-10-01 Inhibitors of histone demethylases

Publications (1)

Publication Number Publication Date
SA515360233B1 true SA515360233B1 (en) 2017-11-12

Family

ID=71451029

Family Applications (1)

Application Number Title Priority Date Filing Date
SA515360233A SA515360233B1 (en) 2012-10-02 2015-04-02 Inhibitors of histone demethylases

Country Status (3)

Country Link
EC (1) ECSP15017165A (en)
HK (1) HK1247920A1 (en)
SA (1) SA515360233B1 (en)

Also Published As

Publication number Publication date
ECSP15017165A (en) 2016-01-29
HK1247920A1 (en) 2018-10-05

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