RU93058362A - METHODS FOR DIASTEROSELECTIVE SYNTHESIS OF NUCLEOSIDES, INTERMEDIATE COMPOUNDS, METHODS FOR PRODUCING INTERMEDIATE COMPOUNDS - Google Patents

METHODS FOR DIASTEROSELECTIVE SYNTHESIS OF NUCLEOSIDES, INTERMEDIATE COMPOUNDS, METHODS FOR PRODUCING INTERMEDIATE COMPOUNDS

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Publication number
RU93058362A
RU93058362A RU93058362/04A RU93058362A RU93058362A RU 93058362 A RU93058362 A RU 93058362A RU 93058362/04 A RU93058362/04 A RU 93058362/04A RU 93058362 A RU93058362 A RU 93058362A RU 93058362 A RU93058362 A RU 93058362A
Authority
RU
Russia
Prior art keywords
methods
intermediate compounds
nucleosides
diasteroselective
synthesis
Prior art date
Application number
RU93058362/04A
Other languages
Russian (ru)
Other versions
RU2140925C1 (en
Inventor
Мансур Тарек
Джин Хаолун
Х.Л.Тсе Аллан
Сиддики М.Арманд
Original Assignee
Биокем Фарма Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Биокем Фарма Инк. filed Critical Биокем Фарма Инк.
Priority claimed from PCT/CA1992/000211 external-priority patent/WO1992020669A1/en
Priority to TJ94000127A priority Critical patent/TJ267R3/en
Publication of RU93058362A publication Critical patent/RU93058362A/en
Application granted granted Critical
Publication of RU2140925C1 publication Critical patent/RU2140925C1/en

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Claims (1)

Изобретение относится к высоко диастереоселективным способам получения цис-нуклеозидов и аналогов и производных нуклеозидов с высокой оптической чистотой и к интермедиатам, пригодным для использования в этих способах.The invention relates to highly diastereoselective methods for producing cis-nucleosides and analogues and derivatives of nucleosides with high optical purity and to intermediates suitable for use in these methods.
RU93058362A 1991-05-21 1992-05-20 Method of diastereoselective synthesis of nucleosides, intermediate compounds, and method of preparing intermediate compounds RU2140925C1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
TJ94000127A TJ267R3 (en) 1992-05-20 1994-12-15 Methods of diastereoselective synthesis of nucleosides intermediate junctions methods of deriving of intermediate junctions

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US70337991A 1991-05-21 1991-05-21
US703,379 1991-05-21
PCT/CA1992/000211 WO1992020669A1 (en) 1991-05-21 1992-05-20 Processes for the diastereoselective synthesis of nucleosides

Related Child Applications (1)

Application Number Title Priority Date Filing Date
RU99115480/04A Division RU2223960C2 (en) 1991-05-21 1992-05-20 Diastereoselective method for preparing glycosylated purine or pyrimidine base

Publications (2)

Publication Number Publication Date
RU93058362A true RU93058362A (en) 1997-01-20
RU2140925C1 RU2140925C1 (en) 1999-11-10

Family

ID=24825144

Family Applications (4)

Application Number Title Priority Date Filing Date
RU96119766/04A RU2163909C2 (en) 1991-05-21 1992-05-20 Pyrimidine 2,3-didesoxynucleoside derivatives and method of preparing thereof
RU99115480/04A RU2223960C2 (en) 1991-05-21 1992-05-20 Diastereoselective method for preparing glycosylated purine or pyrimidine base
RU93058554A RU2105009C1 (en) 1991-05-21 1992-05-20 Method of diastereoselective synthesis of optically active cis-nucleosides, nucleoside analogs or derivatives and intermediate compounds for this method
RU93058362A RU2140925C1 (en) 1991-05-21 1992-05-20 Method of diastereoselective synthesis of nucleosides, intermediate compounds, and method of preparing intermediate compounds

Family Applications Before (3)

Application Number Title Priority Date Filing Date
RU96119766/04A RU2163909C2 (en) 1991-05-21 1992-05-20 Pyrimidine 2,3-didesoxynucleoside derivatives and method of preparing thereof
RU99115480/04A RU2223960C2 (en) 1991-05-21 1992-05-20 Diastereoselective method for preparing glycosylated purine or pyrimidine base
RU93058554A RU2105009C1 (en) 1991-05-21 1992-05-20 Method of diastereoselective synthesis of optically active cis-nucleosides, nucleoside analogs or derivatives and intermediate compounds for this method

Country Status (34)

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US (5) US5756706A (en)
EP (2) EP0515156B1 (en)
JP (3) JP3330972B2 (en)
KR (3) KR0160144B1 (en)
CN (6) CN1038591C (en)
AT (2) ATE157662T1 (en)
AU (4) AU655973B2 (en)
BG (2) BG61696B1 (en)
CA (2) CA2069063C (en)
CZ (3) CZ280857B6 (en)
DE (2) DE69208144T2 (en)
DK (2) DK0515156T3 (en)
EE (1) EE03044B1 (en)
ES (2) ES2104832T3 (en)
FI (3) FI109025B (en)
GR (2) GR3018941T3 (en)
GT (1) GT199800047A (en)
HK (2) HK132196A (en)
HU (2) HU221850B1 (en)
IE (2) IE76741B1 (en)
IL (6) IL116109A (en)
MD (1) MD1155C2 (en)
MX (2) MX9202404A (en)
NO (2) NO300593B1 (en)
NZ (2) NZ242818A (en)
OA (1) OA10212A (en)
PL (3) PL168910B1 (en)
RO (1) RO116812B1 (en)
RU (4) RU2163909C2 (en)
SG (1) SG43863A1 (en)
SK (2) SK279438B6 (en)
TW (4) TW467907B (en)
WO (2) WO1992020696A1 (en)
ZA (2) ZA923641B (en)

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