RU93050124A - NEW DERIVATIVES OF ERYTHROMYCIN, THE METHOD OF THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITION ON THEIR BASIS - Google Patents

NEW DERIVATIVES OF ERYTHROMYCIN, THE METHOD OF THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITION ON THEIR BASIS

Info

Publication number
RU93050124A
RU93050124A RU93050124/04A RU93050124A RU93050124A RU 93050124 A RU93050124 A RU 93050124A RU 93050124/04 A RU93050124/04 A RU 93050124/04A RU 93050124 A RU93050124 A RU 93050124A RU 93050124 A RU93050124 A RU 93050124A
Authority
RU
Russia
Prior art keywords
erythromycin
pharmaceutical composition
basis
production
new derivatives
Prior art date
Application number
RU93050124/04A
Other languages
Russian (ru)
Other versions
RU2114859C1 (en
Inventor
Агурида Константин
Боннефой Ален
Шанто Жан-Франсуа
Дени Олексис
Ле Мартрэ Одиль
Original Assignee
Руссель-Юклаф
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9213321A external-priority patent/FR2697524B1/en
Application filed by Руссель-Юклаф filed Critical Руссель-Юклаф
Publication of RU93050124A publication Critical patent/RU93050124A/en
Application granted granted Critical
Publication of RU2114859C1 publication Critical patent/RU2114859C1/en

Links

Claims (1)

Изобретение касается новых производных эритромицина, обладающих антибиотической активностью в отношении грамположительных бактерий, к способу получения новых соединений и к фармацевтической композиции на их основе.The invention relates to new derivatives of erythromycin with antibiotic activity against gram-positive bacteria, to a method for producing new compounds and to a pharmaceutical composition based on them.
RU93050124A 1992-11-05 1993-11-04 Erythromycin derivatives, pharmaceutical composition, method of synthesis of erythromycin derivatives RU2114859C1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9213321 1992-11-05
FR9213321A FR2697524B1 (en) 1992-11-05 1992-11-05 New erythromycin derivatives, their preparation process and their use as drugs.

Publications (2)

Publication Number Publication Date
RU93050124A true RU93050124A (en) 1997-02-20
RU2114859C1 RU2114859C1 (en) 1998-07-10

Family

ID=9435255

Family Applications (1)

Application Number Title Priority Date Filing Date
RU93050124A RU2114859C1 (en) 1992-11-05 1993-11-04 Erythromycin derivatives, pharmaceutical composition, method of synthesis of erythromycin derivatives

Country Status (15)

Country Link
US (1) US5543400A (en)
EP (1) EP0606024B1 (en)
JP (1) JP3334980B2 (en)
KR (1) KR100319358B1 (en)
CN (1) CN1033273C (en)
AT (1) ATE135709T1 (en)
AU (1) AU664122B2 (en)
CA (1) CA2102454C (en)
DE (1) DE69301907T2 (en)
DK (1) DK0606024T3 (en)
ES (1) ES2085129T3 (en)
FR (1) FR2697524B1 (en)
GR (1) GR3019384T3 (en)
HU (1) HU217977B (en)
RU (1) RU2114859C1 (en)

Families Citing this family (40)

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US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
HRP931480B1 (en) * 1993-12-08 1997-08-31 Sour Pliva 9a-N-(N'-CARBAMONYL) and 9a-N-(N'-THIOCARBAMONYL) DERIVATES OF 9-DEOXO-9a-HOMOERYTHROMYCIN A
FR2718450B1 (en) * 1994-04-08 1997-01-10 Roussel Uclaf New erythromycin derivatives, their preparation process and their use as drugs.
FR2719587B1 (en) * 1994-05-03 1996-07-12 Roussel Uclaf New erythromycin derivatives, their preparation process and their use as drugs.
FR2727969B1 (en) * 1994-12-09 1997-01-17 Roussel Uclaf NOVEL ERYTHROMYCIN DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS
FR2732023B1 (en) * 1995-03-22 1997-04-30 Roussel Uclaf NOVEL ERYTHROMYCIN DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS
FR2732684B1 (en) * 1995-04-06 1997-04-30 Roussel Uclaf NOVEL ERYTHROMYCIN DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS
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HUP0105190A3 (en) 1999-01-27 2003-03-28 Pfizer Prod Inc Ketolide antibiotics, medicaments containing them and their use
US6054435A (en) * 1999-03-19 2000-04-25 Abbott Laboratories 6-O-substituted macrolides having antibacterial activity
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CN1780846A (en) * 2003-03-05 2006-05-31 Rib－X医药品有限公司 Bifunctional heterocyclic compounds and methods of making and using the same
US7601695B2 (en) 2003-03-10 2009-10-13 Optimer Pharmaceuticals, Inc. Antibacterial agents
US20050014706A1 (en) * 2003-07-14 2005-01-20 Kanakeshwari Falzari Method of treating tuberculosis
US20070149463A1 (en) * 2003-10-30 2007-06-28 Oyelere Adegboyega K Bifunctional macrolide heterocyclic compounds and methods of making and using the same
WO2005049632A1 (en) * 2003-11-18 2005-06-02 Rib-X Pharmaceuticals, Inc. Bifunctional macrolide heterocyclic compounds and methods of making and using the same
US8202843B2 (en) * 2004-02-27 2012-06-19 Rib-X Pharmaceuticals, Inc. Macrocyclic compounds and methods of making and using the same
PT1836211E (en) * 2004-12-21 2010-04-08 Pfizer Prod Inc Macrolides
US20100035832A1 (en) * 2005-01-12 2010-02-11 Alpharma Aps Macrolides
CN101917850B (en) * 2007-10-25 2016-01-13 森普拉制药公司 The preparation method of macrolide antibacterial agents
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US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
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CN103080122A (en) 2010-03-22 2013-05-01 森普拉制药公司 Crystalline forms of a macrolide, and uses therefor
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WO1992009614A1 (en) * 1990-11-28 1992-06-11 Taisho Pharmaceutical Co., Ltd. 6-o-methylerythromycin a derivative

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