RU93043528A - 5- (2- (4- (1,2-BENZOTIAZOL-3-IL) -1-PIPERAZINYL) Ethyl MONOHYDRATE) -6-CHLOR-1,3-DIHYDRO-2H-INDOL-2-OH CHLOROHYDRATE, METHOD FOR ITS PREPARATION , PHARMACEUTICAL COMPOSITION, METHOD OF TREATMENT - Google Patents

5- (2- (4- (1,2-BENZOTIAZOL-3-IL) -1-PIPERAZINYL) Ethyl MONOHYDRATE) -6-CHLOR-1,3-DIHYDRO-2H-INDOL-2-OH CHLOROHYDRATE, METHOD FOR ITS PREPARATION , PHARMACEUTICAL COMPOSITION, METHOD OF TREATMENT

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Publication number
RU93043528A
RU93043528A RU93043528/04A RU93043528A RU93043528A RU 93043528 A RU93043528 A RU 93043528A RU 93043528/04 A RU93043528/04 A RU 93043528/04A RU 93043528 A RU93043528 A RU 93043528A RU 93043528 A RU93043528 A RU 93043528A
Authority
RU
Russia
Prior art keywords
piperazinyl
dihydro
preparation
benzotiazol
chlorohydrate
Prior art date
Application number
RU93043528/04A
Other languages
Russian (ru)
Other versions
RU2081116C1 (en
Inventor
Аллен Дуглас Д.М.
Р.Буш Фрэнк
А.Дирома Сабето
М.Годек Деннис
Original Assignee
Пфайзер Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US07/939,204 external-priority patent/US5312925A/en
Application filed by Пфайзер Инк. filed Critical Пфайзер Инк.
Publication of RU93043528A publication Critical patent/RU93043528A/en
Application granted granted Critical
Publication of RU2081116C1 publication Critical patent/RU2081116C1/en

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Claims (1)

Предложен моногидрат 5-(2-(4-(1,2-бензотиазол-3-ил)-1- пиперазинил)этил)-6-хлор-1,3-дигидро-2Н-индол-2-ОН хлоргидрата, обладающий повышенной стабильностью при получении композиций, обладающих нейролептическим действием.Proposed monohydrate 5- (2- (4- (1,2-benzothiazol-3-yl) -1-piperazinyl) ethyl) -6-chloro-1,3-dihydro-2H-indole-2-OH hydrochloride, with increased stability in the preparation of compositions having a neuroleptic effect.
RU9393043528A 1992-09-01 1993-08-31 5-(2-4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)ethyl)-6- -chloro-1,3-dihydro-2h-indol-2-one hydrochloride monohydrate and process for preparation thereof RU2081116C1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US939.204 1992-09-01
US07/939,204 US5312925A (en) 1992-09-01 1992-09-01 Monohydrate of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)-ethyl)-6-chloro-1,3-dihydro-2H-indol-2-one-hydrochloride
US939204 1992-09-01

Publications (2)

Publication Number Publication Date
RU93043528A true RU93043528A (en) 1996-09-20
RU2081116C1 RU2081116C1 (en) 1997-06-10

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Family Applications (1)

Application Number Title Priority Date Filing Date
RU9393043528A RU2081116C1 (en) 1992-09-01 1993-08-31 5-(2-4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)ethyl)-6- -chloro-1,3-dihydro-2h-indol-2-one hydrochloride monohydrate and process for preparation thereof

Country Status (21)

Country Link
US (1) US5312925A (en)
EP (1) EP0586191A1 (en)
JP (1) JP2742372B2 (en)
KR (2) KR100278321B1 (en)
CN (1) CN1033641C (en)
AU (1) AU657231B2 (en)
BR (1) BR9303014A (en)
CA (1) CA2105114C (en)
CZ (1) CZ285984B6 (en)
DE (1) DE9312903U1 (en)
EG (1) EG20251A (en)
FI (1) FI115460B (en)
HU (1) HU221725B1 (en)
IL (1) IL106777A (en)
MX (1) MX9305277A (en)
NO (1) NO300270B1 (en)
NZ (1) NZ248543A (en)
PL (2) PL173967B1 (en)
RU (1) RU2081116C1 (en)
TW (1) TW422845B (en)
ZA (1) ZA936394B (en)

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